PERRONE, MARIA GRAZIA
PERRONE, MARIA GRAZIA
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes
2015-01-01 Schininà, B; Martorana, A; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Perrone, MARIA GRAZIA; de Guidi, G; Catalfo, A; Rappazzo, G; Zuccarello, E; Prezzavento, O; Amata, E; Rescifina, A; Marrazzo, A.
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers
2020-01-01 Braconi, Laura; Bartolucci, Gianluca; Contino, Marialessandra; Chiaramonte, Niccolò; Giampietro, Roberta; Manetti, Dina; Perrone, Maria Grazia; Romanelli, Maria Novella; Colabufo, Nicola Antonio; Riganti, Chiara; Dei, Silvia; Teodori, Elisabetta
[18F]-P6 AS A CYCLOOXYGENASE-1 TARGETED IMAGING AGENT
2012-01-01 Malerba, P.; Uddin, J; Perrone, MARIA GRAZIA; Vitale, P.; Crews, B. C.; Daniel, C. K.; Ghebreselasie, K.; Nickels, M.; Manning, H. C.; Marnett, L. J.; Scilimati, Antonio
A chemoenzymatic scalable route to optically active (R)-1-(pyridin-3-yl)-2-aminoethanol, valuable moiety of beta3-adrenergic receptor agonists
2006-01-01 Perrone, MARIA GRAZIA; Santandrea, E.; Giorgio, E.; Bleve, L.; Scilimati, Antonio; Tortorella, Paolo
A Benzopyrane Derivative as a P-Glycoprotein Stimulator: A Potential Agent to Decrease β-Amyloid Accumulation in Alzheimer's Disease
2012-01-01 Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A.
A Benzopyrane derivative as P-glycoprotein stimulator: a potential agent to decrease beta-amyloid accumulation in Alzheimer’s disease
2012-01-01 Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A.
A Combined HPLC and LC-MS Approach for Evaluating Drug Stability in Elastomeric Devices: A Challenge for the Sustainability in Pharmacoeconomics
2014-01-01 Nardulli, Patrizia; Capparelli, Elena; Perrone, MARIA GRAZIA; Ferraiuolo1, Simona; Rita Laforgia1, Maria; Crapolicchio1 and Nicola Antonio Colabufo2, Claudia
A further pocket or conformational plasticity by mapping COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet behavior
2024-01-01 Solidoro, Roberta; Miciaccia, Morena; Bonaccorso, Carmela; Fortuna, Cosimo Gianluca; Armenise, Domenico; Centonze, Antonella; Ferorelli, Savina; Vitale, Paola; Rodrigues, Pryscila; Guimarães, Renilda; de Oliveira, Alana; da Paz, Mariana; Rangel, Luciana; Sathler, Plínio Cunha; Altomare, Angela; Perrone, Maria Grazia; Scilimati, Antonio
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression
2016-01-01 Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, MARIA GRAZIA; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio
A Simplified Direct O2 Consumption-Based Assay to Test COX Inhibition
2022-01-01 Perrone, M. G.; Miciaccia, M.; Ferorelli, S.; Scilimati, A.
Acridone derivatives and small molecules as P-gp inhibitors
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, MARIA GRAZIA; Cantore, M; Niso, M; Perrone, R.
Activity-lipophilicity relationship studies on P-gp ligands designed as simplified tariquidar bulky fragments
2013-01-01 Contino, Marialessandra; Zinzi, Laura; Cantore, Mariangela; Perrone, Maria Grazia; Leopoldo, Marcello; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio
An attempt to chemically state the cross-talk between monomers of COX homodimers by double/hybrid inhibitors mofezolac-spacer-mofezolac and mofezolac-spacer-arachidonic acid
2021-01-01 Perrone, M. G.; Miciaccia, M.; Vitale, P.; Ferorelli, S.; Araujo, C. D. C. B.; de Almeida, G. S.; Souza Domingos, T. F.; da Silva, L. C. R. P.; de Padula, M.; Cabral, L. M.; Sathler, P. C.; Bonaccorso, C.; Fortuna, C. G.; Scilimati, A.
Arylamino Esters As P-Glycoprotein Modulators: SAR Studies to Establish Requirements for Potency and Selectivity
2015-01-01 Teodori, Elisabetta; Dei, Silvia; Floriddia, Elisa; Perrone, MARIA GRAZIA; Manetti, Dina; Romanelli, Maria Novella; Contino, Marialessandra; Colabufo, Nicola Antonio
Baker's yeast-mediated reduction of ethyl 2-(4-chlorophenoxy)-3-oxoalkanoates intermediates for potential PPARa ligands
2004-01-01 Perrone, MARIA GRAZIA; Santandrea, E; Scilimati, Antonio; Tortorella, V; Capitelli, F; Bertolasi, V.
Beta 3-Adrenoceptor Agonists and (Antagonists as) Inverse Agonists: History, Perspective, Constitutive Activity, and Stereospecific Binding
2010-01-01 Perrone, Mg; Scilimati, Antonio
Beta 3-adrenoceptor ligand development history through patent review
2011-01-01 Perrone, MARIA GRAZIA; Scilimati, Antonio
BETA-3 RECEPTOR LIGANDS AND THEIR USE IN THERAPY
2010-01-01 Scilimati, Antonio; Perrone, MARIA GRAZIA; Santandrea, E.
Bioassisted synthesis of 3-hydroxyacids resembling antilipidemic clofibric acid molecular structure
2003-01-01 Perrone, MARIA GRAZIA; E., Santandrea; Tortorella, Paolo; Scilimati, Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo | |
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes | 1-gen-2015 | Schininà, B; Martorana, A; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Perrone, MARIA GRAZIA; de Guidi, G; Catalfo, A; Rappazzo, G; Zuccarello, E; Prezzavento, O; Amata, E; Rescifina, A; Marrazzo, A. | |
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers | 1-gen-2020 | Braconi, Laura; Bartolucci, Gianluca; Contino, Marialessandra; Chiaramonte, Niccolò; Giampietro, Roberta; Manetti, Dina; Perrone, Maria Grazia; Romanelli, Maria Novella; Colabufo, Nicola Antonio; Riganti, Chiara; Dei, Silvia; Teodori, Elisabetta | |
[18F]-P6 AS A CYCLOOXYGENASE-1 TARGETED IMAGING AGENT | 1-gen-2012 | Malerba, P.; Uddin, J; Perrone, MARIA GRAZIA; Vitale, P.; Crews, B. C.; Daniel, C. K.; Ghebreselasie, K.; Nickels, M.; Manning, H. C.; Marnett, L. J.; Scilimati, Antonio | |
A chemoenzymatic scalable route to optically active (R)-1-(pyridin-3-yl)-2-aminoethanol, valuable moiety of beta3-adrenergic receptor agonists | 1-gen-2006 | Perrone, MARIA GRAZIA; Santandrea, E.; Giorgio, E.; Bleve, L.; Scilimati, Antonio; Tortorella, Paolo | |
A Benzopyrane Derivative as a P-Glycoprotein Stimulator: A Potential Agent to Decrease β-Amyloid Accumulation in Alzheimer's Disease | 1-gen-2012 | Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A. | |
A Benzopyrane derivative as P-glycoprotein stimulator: a potential agent to decrease beta-amyloid accumulation in Alzheimer’s disease | 1-gen-2012 | Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A. | |
A Combined HPLC and LC-MS Approach for Evaluating Drug Stability in Elastomeric Devices: A Challenge for the Sustainability in Pharmacoeconomics | 1-gen-2014 | Nardulli, Patrizia; Capparelli, Elena; Perrone, MARIA GRAZIA; Ferraiuolo1, Simona; Rita Laforgia1, Maria; Crapolicchio1 and Nicola Antonio Colabufo2, Claudia | |
A further pocket or conformational plasticity by mapping COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet behavior | 1-gen-2024 | Solidoro, Roberta; Miciaccia, Morena; Bonaccorso, Carmela; Fortuna, Cosimo Gianluca; Armenise, Domenico; Centonze, Antonella; Ferorelli, Savina; Vitale, Paola; Rodrigues, Pryscila; Guimarães, Renilda; de Oliveira, Alana; da Paz, Mariana; Rangel, Luciana; Sathler, Plínio Cunha; Altomare, Angela; Perrone, Maria Grazia; Scilimati, Antonio | |
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression | 1-gen-2016 | Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, MARIA GRAZIA; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio | |
A Simplified Direct O2 Consumption-Based Assay to Test COX Inhibition | 1-gen-2022 | Perrone, M. G.; Miciaccia, M.; Ferorelli, S.; Scilimati, A. | |
Acridone derivatives and small molecules as P-gp inhibitors | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, MARIA GRAZIA; Cantore, M; Niso, M; Perrone, R. | |
Activity-lipophilicity relationship studies on P-gp ligands designed as simplified tariquidar bulky fragments | 1-gen-2013 | Contino, Marialessandra; Zinzi, Laura; Cantore, Mariangela; Perrone, Maria Grazia; Leopoldo, Marcello; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio | |
An attempt to chemically state the cross-talk between monomers of COX homodimers by double/hybrid inhibitors mofezolac-spacer-mofezolac and mofezolac-spacer-arachidonic acid | 1-gen-2021 | Perrone, M. G.; Miciaccia, M.; Vitale, P.; Ferorelli, S.; Araujo, C. D. C. B.; de Almeida, G. S.; Souza Domingos, T. F.; da Silva, L. C. R. P.; de Padula, M.; Cabral, L. M.; Sathler, P. C.; Bonaccorso, C.; Fortuna, C. G.; Scilimati, A. | |
Arylamino Esters As P-Glycoprotein Modulators: SAR Studies to Establish Requirements for Potency and Selectivity | 1-gen-2015 | Teodori, Elisabetta; Dei, Silvia; Floriddia, Elisa; Perrone, MARIA GRAZIA; Manetti, Dina; Romanelli, Maria Novella; Contino, Marialessandra; Colabufo, Nicola Antonio | |
Baker's yeast-mediated reduction of ethyl 2-(4-chlorophenoxy)-3-oxoalkanoates intermediates for potential PPARa ligands | 1-gen-2004 | Perrone, MARIA GRAZIA; Santandrea, E; Scilimati, Antonio; Tortorella, V; Capitelli, F; Bertolasi, V. | |
Beta 3-Adrenoceptor Agonists and (Antagonists as) Inverse Agonists: History, Perspective, Constitutive Activity, and Stereospecific Binding | 1-gen-2010 | Perrone, Mg; Scilimati, Antonio | |
Beta 3-adrenoceptor ligand development history through patent review | 1-gen-2011 | Perrone, MARIA GRAZIA; Scilimati, Antonio | |
BETA-3 RECEPTOR LIGANDS AND THEIR USE IN THERAPY | 1-gen-2010 | Scilimati, Antonio; Perrone, MARIA GRAZIA; Santandrea, E. | |
Bioassisted synthesis of 3-hydroxyacids resembling antilipidemic clofibric acid molecular structure | 1-gen-2003 | Perrone, MARIA GRAZIA; E., Santandrea; Tortorella, Paolo; Scilimati, Antonio |