COLABUFO, Nicola Antonio
COLABUFO, Nicola Antonio
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
"Tritium radiolabeling of [3H]-1-cicloesil-4-[3-(5-methoxy-1,2, 3,4,-tetraidronaftalen-1-il)-n-propil] piperazine ([3H]-PB28)as potent sigma-2 receptor ligand
2008-01-01 Abate, C; Berardi, Francesco; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto
1,2,3,4-Tetrahydroisoquinoline/2H-chromen-2-one conjugates as nanomolar P-glycoprotein inhibitors: Molecular determinants for affinity and selectivity over multidrug resistance associated protein 1
2019-01-01 Rullo, Mariagrazia; Niso, Mauro; Pisani, Leonardo; Carrieri, Antonio; Colabufo, Nicola Antonio; Cellamare, Saverio; Altomare, Cosimo Damiano
1-(2-Methoxyphenyl)-4-alkylpiperazines: effect of the N-4 substituent on the affinity and selectivity for dopamine D4 receptor
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Arylpiperazinic ligands of 5-HT7 receptor and use threreof
2011-01-01 Leopoldo, Marcello; Lacivita, E; Colabufo, Nicola Antonio; De Giorgio, P; Berardi, Francesco; Perrone, R.
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ(8)-Δ(7) Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity
2011-01-01 Abate, C; Niso, M; Contino, M; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, R; Berardi, Francesco
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Delta8─Delta7 sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activity
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Contino, Marialessandra; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto; Berardi, Francesco
1-Cyclohexylpiperazine and 3,3-Dimethylpiperidine Derivatives as Sigma-1 (σ1) and Sigma-2 (σ2) Receptor Ligands: A Review
2009-01-01 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
1-Cyclohexylpiperazine and 3,3-dimethylpiperidine derivatives as sigma-1 and sigma-2 receptor ligand: a review
2009-01-01 Berardi, Francesco; Abate, C; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
1-Phenylalkoxy-2-beta-phenylethyl derivatives as P-gP inhibitors useful in drug resistance events
2007-01-01 Berardi, Francesco; Colabufo, Nicola Antonio; Perrone, Roberto; A., Balsamo; S., Rapposelli
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
11C- and 18F-Labeled Radioligands for P-Glycoprotein Imaging by Positron Emission Tomography
2016-01-01 Cantore, M; Benadiba, M; Elsinga, Ph; Kwizera, C; Dierckx, R. A.; Colabufo, Nicola Antonio; Luurtsema, G.
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors
2005-01-01 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
2-(Aryloxy)ethylamine derivatives: ring opened congeners of long chain 1-arylpiperazines with high 5-HT1A receptor affinity and selectivity versus D2 and a1 receptors
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
2-[(3-Methoxyphenylethyl)phenoxy]-based ABCB1 inhibitors: effect of different basic side-chains on their biological properties
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A.
3-benzazecine-based cyclic allene derivatives as highly potent P-glycoprotein inhibitors overcoming doxorubicin multidrug resistance
2019-01-01 Titov, A. A.; Niso, M.; Candia, M.; Kobzev, M. S.; Varlamov, A. V.; Borisova, T. N.; Voskressensky, L. G.; Colabufo, N. A.; Cellamare, S.; Pisani, L.; Altomare, C. D.
34. Methyl substitution on the piperidine ring of N-[ -(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma-1 receptor
2005-01-01 Berardi, Francesco; Ferorelli, Savina; Abate, C; Pedone, Mp; Colabufo, Nicola Antonio; Contino, M; Perrone, R.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
4-[omega-Tetralin-1-yl]-1-benzylpiperazines and related compounds as 5-HT1A/D-2 ligands
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lograno, M.; Tortorella, V.
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo