PURGATORIO, ROSA

PURGATORIO, ROSA  

DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO  

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Risultati 1 - 20 di 54 (tempo di esecuzione: 0.038 secondi).
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1,3,5-triazine derivatives as dual inhibitors of 5-HT6R/FAAH in search of new therapy for Alzheimer's disease 1-gen-2022 Czarnota-Łydka, Kinga; Satała, Grzegorz; Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; DE CANDIA, Modesto; Purgatorio, Rosa; Gumułka, Magdalena; Kucwaj-Brysz, Katarzyna; Carrieri, Antonio; Handzlik, Jadwiga
3D-QSAR and pharmacophore mapping of 1H-indole-2,3-dione adducts inhibiting beta-amyloid aggregation and other major targets related to Alzheimer’s Disease. 1-gen-2021 Purgatorio, R.; Gambacorta, N.; Catto, M.; de Candia, M.; Pisani, L.; Rullo, M.; Nicolotti, O.; Altomare, C. D.
A Critical Appraisal of the Protecting Activity of Polyphenolic Antioxidants Against Iatrogenic Effects of Anticancer Chemotherapeutics§ 1-gen-2024 Purgatorio, Rosa; Boccarelli, Angelina; Pisani, Leonardo; De Candia, Modesto; Catto, Marco; Altomare, Cosimo Damiano
A new class of 1-aryl-5,6-dihydropyrrolo[2,1-a]isoquinoline derivatives as reversers of P-glycoprotein-mediated multidrug resistance in tumor cells 1-gen-2018 Altomare, Cosimo Damiano; Nevskaya, Alisa A.; Matveeva, Maria D.; Borisova, Tatiana N.; Niso, Mauro; Colabufo, Nicola Antonio; Boccarelli, Angelina; Purgatorio, Rosa; de Candia, Modesto; Cellamare, Saverio; Voskressensky, Leonid G.
A Prospective Repurposing of Dantrolene as a Multitarget Agent for Alzheimer’s Disease 1-gen-2019 Bolognino, I; Giangregorio, N; Pisani, L; de Candia, M; Purgatorio, R; Tonazzi, A; Altomare, Cd; Cellamare, S; Catto, M
A second life for MAO inhibitors? From CNS diseases to anticancer therapy 1-gen-2024 Sblano, Sabina; Boccarelli, Angelina; Mesiti, Francesco; Purgatorio, Rosa; de Candia, Modesto; Catto, Marco; Altomare, Cosimo D.
Annelated medium-sized azaheterocycles as attractive scaffolds for CNS targeted leads. 1-gen-2019 Altomare, C. D.; de Candia, M.; Purgatorio, R.; Pisani, L.; Catto, M.; Cellamare, S.; Titov, A. A.; Voskressensky, L. G.
Assessing the Role of a Malonamide Linker in the Design of Potent Dual Inhibitors of Factor Xa and Cholinesterases 1-gen-2022 Purgatorio, Rosa; Gambacorta, Nicola; Samarelli, Francesco; Lopopolo, Gianfranco; DE CANDIA, Modesto; Catto, Marco; Nicolotti, Orazio; Altomare, Cosimo D.
Biophysical Characterization of Inhibition of A-beta Fibril Formation by Isatin-3-arylhydrazones 1-gen-2010 Campagna, Francesco; Purgatorio, R; Catto, Marco; Carotti, A; De, Stradisa; Palazzo, Gerardo
Biophysical Characterization of Inhibition of A-beta Fibril Formation by Isatin-3-arylhydrazones 1-gen-2010 Campagna, F; Purgatorio, R; Catto, M; Carotti, A; Stradisa, De; Palazzo, G
Biophysical characterization of inhibition of Aβ fibril formation by isatin-3-arylhydrazones 1-gen-2010 Campagna, F; Purgatorio, R; Catto, Marco; Carotti, A; De Stradis, A; Palazzo, Gerardo
Chemical and Biological Evaluation of Novel 1H-Chromeno[3,2-c]pyridine Derivatives as MAO Inhibitors Endowed with Potential Anticancer Activity 1-gen-2023 Kulikova, Larisa N.; Purgatorio, Rosa; Beloglazkin, Andrey A.; Tafeenko, Viktor A.; Reza, Raesi Gh.; Levickaya, Daria D.; Sblano, Sabina; Boccarelli, Angelina; DE CANDIA, Modesto; Catto, Marco; Voskressensky, Leonid G.; Altomare, Cosimo D.
Design, synthesis and biological evaluation of indane 2-arylhydrazinylmethylene-1,3-diones and indol-2-aryldiazenylmethylene-3-ones as b-amyloid aggregation inhibitors 1-gen-2010 Catto, Marco; Aliano, R; Carotti, Angelo; Cellamare, Saverio; Palluotto, Fausta; Purgatorio, R; DE STRADIS, A; Campagna, Francesco
Development of a continuous flow synthesis of propranolol: tackling a competitive side reaction 1-gen-2019 De Angelis, S.; Celestini, P.; Purgatorio, R.; Degennaro, L.; Rebuzzini, G.; Luisi, R.; Carlucci, C.
Enantiomeric Separation and Molecular Modelling of Bioactive 4-Aryl-3,4-dihydropyrimidin-2(1H)-one Ester Derivatives on Teicoplanin-Based Chiral Stationary Phase 1-gen-2022 Bolognino, Isabella; Carrieri, Antonio; Purgatorio, Rosa; Catto, Marco; Caliandro, Rocco; Carrozzini, Benedetta; Belviso, BENNY DANILO; Majellaro, Maria; Sotelo, Eddy; Cellamare, Saverio; Altomare, Cosimo Damiano
Evaluation of Novel Guanidino-Containing Isonipecotamide Inhibitors of Blood Coagulation Factors against SARS-CoV-2 Virus Infection 1-gen-2022 Maio, F. D.; Rullo, M.; de Candia, M.; Purgatorio, R.; Lopopolo, G.; Santarelli, G.; Palmieri, V.; Papi, M.; Elia, G.; De Candia, E.; Sanguinetti, M.; Altomare, C. D.
Evaluation of water‐soluble Mannich base prodrugs of 2,3,4,5‐tetrahydroazepino[4,3‐b]indol‐1(6H)‐one as multitarget‐directed agents for Alzheimer’s disease 1-gen-2021 Purgatorio, Rosa; de Candia, Modesto; Catto, Marco; Rullo, Mariagrazia; Pisani, Leonardo; Denora, Nunzio; Carrieri, Antonio; Nevskaya, Alisa A.; Voskressensky, Leonid G.; Altomare, Cosimo D.
First-in-Class Isonipecotamide-Based Thrombin and Cholinesterase Dual Inhibitors with Potential for Alzheimer Disease 1-gen-2021 Purgatorio, Rosa; Gambacorta, Nicola; DE CANDIA, Modesto; Catto, Marco; Rullo, Mariagrazia; Pisani, Leonardo; Nicolotti, Orazio; Altomare, Cosimo Damiano
HISTONE ACETYLTRANSFERASE ACTIVATORS AND COMPOSITIONS AND USES THEREOF 1-gen-2018 O'Connor Owen, Anthony; Deng Shi, Xian; Scotto, Luigi; Purgatorio, Rosa; Arancio, Ottavio; Fiorito, Jole; Amengual Jennifer, Effie; Landry Donald, W.
HISTONE ACETYLTRANSFERASE ACTIVATORS AND USES THEREOF 1-gen-2015 Arancio, Ottavio; Deng Shi, Xian; Landry Donald, W; Fiorito, Jole; Purgatorio, Rosa; O'Connor Owen, Anthony; Amengual Jennifer, Effie