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Novel and Selective Fluorescent σ2-Receptor Ligand with a 3,4-Dihydroisoquinolin-1-one Scaffold: A Tool to Study σ2 Receptors in Living Cells 1-gen-2015 Niso, Mauro; Riganti, Chiara; Pati, MARIA LAURA; Ghigo, Dario; Berardi, Francesco; Abate, CARMEN rosa
Deconstruction of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline moiety to separate Pglycoprotein (P-gp) activity from σ2 receptor affinity in mixed P-gp/σ2 receptor agents 1-gen-2015 Pati, MARIA LAURA; Abate, CARMEN rosa; Contino, Marialessandra; Ferorelli, Savina; Luisi, Renzo; Laura, Carroccia; Niso, Mauro; Berardi, Francesco
Synthesis and pharmacological evaluation of 11C-labeled piperazine derivative as a PET probe for sigma-2 receptor imaging 1-gen-2015 Svetlana V., Selivanova; Annamaria, Toscano; Abate, CARMEN rosa; Berardi, Francesco; Adrienne, Müller; Stefanie D., Krämer; Roger, Schibli; Simon M., Ametamey
Novel Metal Chelators Thiosemicarbazones with Activity at the sigma2 Receptors and P-glycoprotein: an Innovative Strategy for Resistant Tumors Treatment 1-gen-2015 Pati, MARIA LAURA; Niso, Mauro; Ferorelli, Savina; Abate, CARMEN rosa; Berardi, Francesco
Elements in support of the 'non-identity' of the PGRMC1 protein with the σ2 receptor 1-gen-2015 Abate, C; Niso, Mauro; Infantino, V; Menga, A; Berardi, Francesco
Live imaging reveals a new role for the sigma-1 (σ1) receptor in allowing microglia to leave brain injuries 1-gen-2015 Moritz, Christian; Berardi, Francesco; Abate, CARMEN rosa; Peri, Francesca
Development of sigma-1 (σ1) receptor fluorescent ligands as versatile tools to study σ1 receptors 1-gen-2016 Abate, CARMEN rosa; Riganti, Chiara; Pati, MARIA LAURA; Ghigo, Dario; Berardi, Francesco; Mavlyutov, Timur; Guo, Lian Wang; Ruoho, Arnold
Rigid versus flexible anilines or anilides confirm the bicyclic ring as the hydrophobic portion for optimal σ2 receptor binding and provide novel tools for the development of future σ2 receptor PET radiotracer 1-gen-2016 Niso, Mauro; Pati, MARIA LAURA; Berardi, Francesco; Abate, CARMEN rosa
Society for Neuroscience Annual Meeting; Nanosymposium: Sigma-2/PGRMC1 Receptor Function in Disease and Therapeutics 1-gen-2016 Pati, MARIA LAURA; Abate, CARMEN rosa; Niso, Mauro; Berardi, Francesco; Colabufo, Nicola Antonio
The σ1 receptor agonist (+)-pentazocine increases store-operated Ca2+ entry in MCF7σ1 and SK-N-SH cell lines 1-gen-2017 Gasparre, Giuseppe; Abate, CARMEN rosa; Carlucci, Roberto; Berardi, Francesco; Cassano, Giuseppe
Sigma-2 receptor agonist derivatives of 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) induce cell death via mitochondrial superoxide production and caspase activation in pancreatic cancer 1-gen-2017 Pati, MARIA LAURA; Hornick, John R.; Niso, Mauro; Berardi, Francesco; Spitzer, Dirk; Abate, CARMEN rosa; Hawkins, William
Perspectives of Cannabinoid Type 2 Receptor (CB2R) Ligands in Neurodegenerative Disorders: Structure–Affinity Relationship (SAfiR) and Structure–Activity Relationship (SAR) Studies 1-gen-2017 Spinelli, F; Capparelli, E; Abate, C; Colabufo, Na; Contino, M.
Sigma 2 receptor expression levels in blood and bladder from healthy and bladder cancer cattle 1-gen-2017 Russo, V; Inglese, C; Avallone, L; Roperto, F; Abate, C; Zizzo, N; Munday, J S; Berardi, F; Colabufo, N A; Roperto, S
Sigma-2 receptor and progesterone receptor membrane component 1 (PGRMC1) are two different proteins: Proofs by fluorescent labeling and binding of sigma-2 receptor ligands to PGRMC1 1-gen-2017 Pati, MARIA LAURA; Groza, Diana; Riganti, Chiara; Kopecka, Joanna; Niso, Mauro; Berardi, Francesco; Hager, Sonja; Heffeter, Petra; Hirai, Miwa; Tsugawa, Hitoshi; Kabe, Yasuaki; Suematsu, Makoto; Abate, CARMEN rosa
Sigma-2 receptor: Past, present and perspectives on multiple therapeutic exploitations 1-gen-2018 Abate, Carmen; Niso, Mauro; Berardi, Francesco
Synthesis, radiolabelling, and evaluation of [11C]PB212 as a radioligand for imaging sigma-1 receptors using PET. 1-gen-2018 Francesco, Spinelli; Ahmed, Haider; Toscano, Annamaria; Pati, MARIA LAURA; Claudia, Keller; Berardi, Francesco; Colabufo, Nicola Antonio; Abate, Carmen; Simon, M Ametamey:
Quantum Dot Based Luminescent Nanoprobes for Sigma-2 Receptor Imaging 1-gen-2018 Pati, Maria Laura; Fanizza, Elisabetta; Hager, Sonja; Groza, Diana; Heffeter, Petra; Laurenza, Amelita Grazia; Laquintana, Valentino; Curri, Maria Lucia; Depalo, Nicoletta; Abate, Carmen; Denora, Nunzio
Multifunctional thiosemicarbazones and deconstructed analogues as a strategy to study the involvement of metal chelation, Sigma-2 (Ï 2) receptor and P-gp protein in the cytotoxic action: In vitro and in vivo activity in pancreatic tumors 1-gen-2018 Pati, Maria Laura; Niso, Mauro; Spitzer, Dirk; Berardi, Francesco; Contino, Marialessandra; Riganti, Chiara; Hawkins, William G.; Abate, Carmen
Validation of Thiosemicarbazone Compounds as P-Glycoprotein Inhibitors in Human Primary Brain-Blood Barrier and Glioblastoma Stem Cells 1-gen-2019 Salaroglio, Iris Chiara; Abate, Carmen; Rolando, Barbara; Battaglia, Luigi; Gazzano, Elena; Colombino, Elena; Costamagna, Costanzo; Annovazzi, Laura; Mellai, Marta; Berardi, Francesco; Capucchio, Maria Teresa; Schiffer, Davide; Riganti, Chiara
High-affinity sigma-1 (σ1) receptor ligands based on the σ1 antagonist PB212 1-gen-2019 Niso, M.; Mosier, P. D.; Marottoli, Roberta; Ferorelli, S.; Cassano, G.; Gasparre, G.; Leopoldo, M.; Berardi, F.; Abate, C.
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