Sfoglia per Autore
Novel and Selective Fluorescent σ2-Receptor Ligand with a 3,4-Dihydroisoquinolin-1-one Scaffold: A Tool to Study σ2 Receptors in Living Cells
2015-01-01 Niso, Mauro; Riganti, Chiara; Pati, MARIA LAURA; Ghigo, Dario; Berardi, Francesco; Abate, CARMEN rosa
Deconstruction of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline moiety to separate Pglycoprotein (P-gp) activity from σ2 receptor affinity in mixed P-gp/σ2 receptor agents
2015-01-01 Pati, MARIA LAURA; Abate, CARMEN rosa; Contino, Marialessandra; Ferorelli, Savina; Luisi, Renzo; Laura, Carroccia; Niso, Mauro; Berardi, Francesco
Synthesis and pharmacological evaluation of 11C-labeled piperazine derivative as a PET probe for sigma-2 receptor imaging
2015-01-01 Svetlana V., Selivanova; Annamaria, Toscano; Abate, CARMEN rosa; Berardi, Francesco; Adrienne, Müller; Stefanie D., Krämer; Roger, Schibli; Simon M., Ametamey
Novel Metal Chelators Thiosemicarbazones with Activity at the sigma2 Receptors and P-glycoprotein: an Innovative Strategy for Resistant Tumors Treatment
2015-01-01 Pati, MARIA LAURA; Niso, Mauro; Ferorelli, Savina; Abate, CARMEN rosa; Berardi, Francesco
Elements in support of the 'non-identity' of the PGRMC1 protein with the σ2 receptor
2015-01-01 Abate, C; Niso, Mauro; Infantino, V; Menga, A; Berardi, Francesco
Live imaging reveals a new role for the sigma-1 (σ1) receptor in allowing microglia to leave brain injuries
2015-01-01 Moritz, Christian; Berardi, Francesco; Abate, CARMEN rosa; Peri, Francesca
Development of sigma-1 (σ1) receptor fluorescent ligands as versatile tools to study σ1 receptors
2016-01-01 Abate, CARMEN rosa; Riganti, Chiara; Pati, MARIA LAURA; Ghigo, Dario; Berardi, Francesco; Mavlyutov, Timur; Guo, Lian Wang; Ruoho, Arnold
Rigid versus flexible anilines or anilides confirm the bicyclic ring as the hydrophobic portion for optimal σ2 receptor binding and provide novel tools for the development of future σ2 receptor PET radiotracer
2016-01-01 Niso, Mauro; Pati, MARIA LAURA; Berardi, Francesco; Abate, CARMEN rosa
Society for Neuroscience Annual Meeting; Nanosymposium: Sigma-2/PGRMC1 Receptor Function in Disease and Therapeutics
2016-01-01 Pati, MARIA LAURA; Abate, CARMEN rosa; Niso, Mauro; Berardi, Francesco; Colabufo, Nicola Antonio
The σ1 receptor agonist (+)-pentazocine increases store-operated Ca2+ entry in MCF7σ1 and SK-N-SH cell lines
2017-01-01 Gasparre, Giuseppe; Abate, CARMEN rosa; Carlucci, Roberto; Berardi, Francesco; Cassano, Giuseppe
Sigma-2 receptor agonist derivatives of 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) induce cell death via mitochondrial superoxide production and caspase activation in pancreatic cancer
2017-01-01 Pati, MARIA LAURA; Hornick, John R.; Niso, Mauro; Berardi, Francesco; Spitzer, Dirk; Abate, CARMEN rosa; Hawkins, William
Perspectives of Cannabinoid Type 2 Receptor (CB2R) Ligands in Neurodegenerative Disorders: Structure–Affinity Relationship (SAfiR) and Structure–Activity Relationship (SAR) Studies
2017-01-01 Spinelli, F; Capparelli, E; Abate, C; Colabufo, Na; Contino, M.
Sigma 2 receptor expression levels in blood and bladder from healthy and bladder cancer cattle
2017-01-01 Russo, V; Inglese, C; Avallone, L; Roperto, F; Abate, C; Zizzo, N; Munday, J S; Berardi, F; Colabufo, N A; Roperto, S
Sigma-2 receptor and progesterone receptor membrane component 1 (PGRMC1) are two different proteins: Proofs by fluorescent labeling and binding of sigma-2 receptor ligands to PGRMC1
2017-01-01 Pati, MARIA LAURA; Groza, Diana; Riganti, Chiara; Kopecka, Joanna; Niso, Mauro; Berardi, Francesco; Hager, Sonja; Heffeter, Petra; Hirai, Miwa; Tsugawa, Hitoshi; Kabe, Yasuaki; Suematsu, Makoto; Abate, CARMEN rosa
Sigma-2 receptor: Past, present and perspectives on multiple therapeutic exploitations
2018-01-01 Abate, Carmen; Niso, Mauro; Berardi, Francesco
Synthesis, radiolabelling, and evaluation of [11C]PB212 as a radioligand for imaging sigma-1 receptors using PET.
2018-01-01 Francesco, Spinelli; Ahmed, Haider; Toscano, Annamaria; Pati, MARIA LAURA; Claudia, Keller; Berardi, Francesco; Colabufo, Nicola Antonio; Abate, Carmen; Simon, M Ametamey:
Quantum Dot Based Luminescent Nanoprobes for Sigma-2 Receptor Imaging
2018-01-01 Pati, Maria Laura; Fanizza, Elisabetta; Hager, Sonja; Groza, Diana; Heffeter, Petra; Laurenza, Amelita Grazia; Laquintana, Valentino; Curri, Maria Lucia; Depalo, Nicoletta; Abate, Carmen; Denora, Nunzio
Multifunctional thiosemicarbazones and deconstructed analogues as a strategy to study the involvement of metal chelation, Sigma-2 (Ï 2) receptor and P-gp protein in the cytotoxic action: In vitro and in vivo activity in pancreatic tumors
2018-01-01 Pati, Maria Laura; Niso, Mauro; Spitzer, Dirk; Berardi, Francesco; Contino, Marialessandra; Riganti, Chiara; Hawkins, William G.; Abate, Carmen
Validation of Thiosemicarbazone Compounds as P-Glycoprotein Inhibitors in Human Primary Brain-Blood Barrier and Glioblastoma Stem Cells
2019-01-01 Salaroglio, Iris Chiara; Abate, Carmen; Rolando, Barbara; Battaglia, Luigi; Gazzano, Elena; Colombino, Elena; Costamagna, Costanzo; Annovazzi, Laura; Mellai, Marta; Berardi, Francesco; Capucchio, Maria Teresa; Schiffer, Davide; Riganti, Chiara
High-affinity sigma-1 (σ1) receptor ligands based on the σ1 antagonist PB212
2019-01-01 Niso, M.; Mosier, P. D.; Marottoli, Roberta; Ferorelli, S.; Cassano, G.; Gasparre, G.; Leopoldo, M.; Berardi, F.; Abate, C.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel and Selective Fluorescent σ2-Receptor Ligand with a 3,4-Dihydroisoquinolin-1-one Scaffold: A Tool to Study σ2 Receptors in Living Cells | 1-gen-2015 | Niso, Mauro; Riganti, Chiara; Pati, MARIA LAURA; Ghigo, Dario; Berardi, Francesco; Abate, CARMEN rosa | |
Deconstruction of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline moiety to separate Pglycoprotein (P-gp) activity from σ2 receptor affinity in mixed P-gp/σ2 receptor agents | 1-gen-2015 | Pati, MARIA LAURA; Abate, CARMEN rosa; Contino, Marialessandra; Ferorelli, Savina; Luisi, Renzo; Laura, Carroccia; Niso, Mauro; Berardi, Francesco | |
Synthesis and pharmacological evaluation of 11C-labeled piperazine derivative as a PET probe for sigma-2 receptor imaging | 1-gen-2015 | Svetlana V., Selivanova; Annamaria, Toscano; Abate, CARMEN rosa; Berardi, Francesco; Adrienne, Müller; Stefanie D., Krämer; Roger, Schibli; Simon M., Ametamey | |
Novel Metal Chelators Thiosemicarbazones with Activity at the sigma2 Receptors and P-glycoprotein: an Innovative Strategy for Resistant Tumors Treatment | 1-gen-2015 | Pati, MARIA LAURA; Niso, Mauro; Ferorelli, Savina; Abate, CARMEN rosa; Berardi, Francesco | |
Elements in support of the 'non-identity' of the PGRMC1 protein with the σ2 receptor | 1-gen-2015 | Abate, C; Niso, Mauro; Infantino, V; Menga, A; Berardi, Francesco | |
Live imaging reveals a new role for the sigma-1 (σ1) receptor in allowing microglia to leave brain injuries | 1-gen-2015 | Moritz, Christian; Berardi, Francesco; Abate, CARMEN rosa; Peri, Francesca | |
Development of sigma-1 (σ1) receptor fluorescent ligands as versatile tools to study σ1 receptors | 1-gen-2016 | Abate, CARMEN rosa; Riganti, Chiara; Pati, MARIA LAURA; Ghigo, Dario; Berardi, Francesco; Mavlyutov, Timur; Guo, Lian Wang; Ruoho, Arnold | |
Rigid versus flexible anilines or anilides confirm the bicyclic ring as the hydrophobic portion for optimal σ2 receptor binding and provide novel tools for the development of future σ2 receptor PET radiotracer | 1-gen-2016 | Niso, Mauro; Pati, MARIA LAURA; Berardi, Francesco; Abate, CARMEN rosa | |
Society for Neuroscience Annual Meeting; Nanosymposium: Sigma-2/PGRMC1 Receptor Function in Disease and Therapeutics | 1-gen-2016 | Pati, MARIA LAURA; Abate, CARMEN rosa; Niso, Mauro; Berardi, Francesco; Colabufo, Nicola Antonio | |
The σ1 receptor agonist (+)-pentazocine increases store-operated Ca2+ entry in MCF7σ1 and SK-N-SH cell lines | 1-gen-2017 | Gasparre, Giuseppe; Abate, CARMEN rosa; Carlucci, Roberto; Berardi, Francesco; Cassano, Giuseppe | |
Sigma-2 receptor agonist derivatives of 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) induce cell death via mitochondrial superoxide production and caspase activation in pancreatic cancer | 1-gen-2017 | Pati, MARIA LAURA; Hornick, John R.; Niso, Mauro; Berardi, Francesco; Spitzer, Dirk; Abate, CARMEN rosa; Hawkins, William | |
Perspectives of Cannabinoid Type 2 Receptor (CB2R) Ligands in Neurodegenerative Disorders: Structure–Affinity Relationship (SAfiR) and Structure–Activity Relationship (SAR) Studies | 1-gen-2017 | Spinelli, F; Capparelli, E; Abate, C; Colabufo, Na; Contino, M. | |
Sigma 2 receptor expression levels in blood and bladder from healthy and bladder cancer cattle | 1-gen-2017 | Russo, V; Inglese, C; Avallone, L; Roperto, F; Abate, C; Zizzo, N; Munday, J S; Berardi, F; Colabufo, N A; Roperto, S | |
Sigma-2 receptor and progesterone receptor membrane component 1 (PGRMC1) are two different proteins: Proofs by fluorescent labeling and binding of sigma-2 receptor ligands to PGRMC1 | 1-gen-2017 | Pati, MARIA LAURA; Groza, Diana; Riganti, Chiara; Kopecka, Joanna; Niso, Mauro; Berardi, Francesco; Hager, Sonja; Heffeter, Petra; Hirai, Miwa; Tsugawa, Hitoshi; Kabe, Yasuaki; Suematsu, Makoto; Abate, CARMEN rosa | |
Sigma-2 receptor: Past, present and perspectives on multiple therapeutic exploitations | 1-gen-2018 | Abate, Carmen; Niso, Mauro; Berardi, Francesco | |
Synthesis, radiolabelling, and evaluation of [11C]PB212 as a radioligand for imaging sigma-1 receptors using PET. | 1-gen-2018 | Francesco, Spinelli; Ahmed, Haider; Toscano, Annamaria; Pati, MARIA LAURA; Claudia, Keller; Berardi, Francesco; Colabufo, Nicola Antonio; Abate, Carmen; Simon, M Ametamey: | |
Quantum Dot Based Luminescent Nanoprobes for Sigma-2 Receptor Imaging | 1-gen-2018 | Pati, Maria Laura; Fanizza, Elisabetta; Hager, Sonja; Groza, Diana; Heffeter, Petra; Laurenza, Amelita Grazia; Laquintana, Valentino; Curri, Maria Lucia; Depalo, Nicoletta; Abate, Carmen; Denora, Nunzio | |
Multifunctional thiosemicarbazones and deconstructed analogues as a strategy to study the involvement of metal chelation, Sigma-2 (Ï 2) receptor and P-gp protein in the cytotoxic action: In vitro and in vivo activity in pancreatic tumors | 1-gen-2018 | Pati, Maria Laura; Niso, Mauro; Spitzer, Dirk; Berardi, Francesco; Contino, Marialessandra; Riganti, Chiara; Hawkins, William G.; Abate, Carmen | |
Validation of Thiosemicarbazone Compounds as P-Glycoprotein Inhibitors in Human Primary Brain-Blood Barrier and Glioblastoma Stem Cells | 1-gen-2019 | Salaroglio, Iris Chiara; Abate, Carmen; Rolando, Barbara; Battaglia, Luigi; Gazzano, Elena; Colombino, Elena; Costamagna, Costanzo; Annovazzi, Laura; Mellai, Marta; Berardi, Francesco; Capucchio, Maria Teresa; Schiffer, Davide; Riganti, Chiara | |
High-affinity sigma-1 (σ1) receptor ligands based on the σ1 antagonist PB212 | 1-gen-2019 | Niso, M.; Mosier, P. D.; Marottoli, Roberta; Ferorelli, S.; Cassano, G.; Gasparre, G.; Leopoldo, M.; Berardi, F.; Abate, C. |
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