Sfoglia per Autore
High-affinity sigma-1 (σ1) receptor ligands based on the σ1 antagonist PB212
2019-01-01 Niso, M.; Mosier, P. D.; Marottoli, Roberta; Ferorelli, S.; Cassano, G.; Gasparre, G.; Leopoldo, M.; Berardi, F.; Abate, C.
NO1, a new sigma 2 receptor/TMEM97 fluorescent ligand, downregulates SOCE and promotes apoptosis in the triple negative breast cancer cell lines
2020-01-01 Cantonero, C.; Camello, P. J.; Abate, C.; Berardi, F.; Salido, G. M.; Rosado, J. A.; Redondo, P. C.
Comparative host-coronavirus protein interaction networks reveal pan-viral disease mechanisms
2020-01-01 Gordon, David E; Hiatt, Joseph; Bouhaddou, Mehdi; Rezelj, Veronica V; Ulferts, Svenja; Braberg, Hannes; Jureka, Alexander S; Obernier, Kirsten; Guo, Jeffrey Z; Batra, Jyoti; Kaake, Robyn M; Weckstein, Andrew R; Owens, Tristan W; Gupta, Meghna; Pourmal, Sergei; Titus, Erron W; Cakir, Merve; Soucheray, Margaret; Mcgregor, Michael; Cakir, Zeynep; Jang, Gwendolyn; O'Meara, Matthew J; Tummino, Tia A; Zhang, Ziyang; Foussard, Helene; Rojc, Ajda; Zhou, Yuan; Kuchenov, Dmitry; Hüttenhain, Ruth; Xu, Jiewei; Eckhardt, Manon; Swaney, Danielle L; Fabius, Jacqueline M; Ummadi, Manisha; Tutuncuoglu, Beril; Rathore, Ujjwal; Modak, Maya; Haas, Paige; Haas, Kelsey M; Naing, Zun Zar Chi; Pulido, Ernst H; Shi, Ying; Barrio-Hernandez, Inigo; Memon, Danish; Petsalaki, Eirini; Dunham, Alistair; Marrero, Miguel Correa; Burke, David; Koh, Cassandra; Vallet, Thomas; Silvas, Jesus A; Azumaya, Caleigh M; Billesbølle, Christian; Brilot, Axel F; Campbell, Melody G; Diallo, Amy; Dickinson, Miles Sasha; Diwanji, Devan; Herrera, Nadia; Hoppe, Nick; Kratochvil, Huong T; Liu, Yanxin; Merz, Gregory E; Moritz, Michelle; Nguyen, Henry C; Nowotny, Carlos; Puchades, Cristina; Rizo, Alexandrea N; Schulze-Gahmen, Ursula; Smith, Amber M; Sun, Ming; Young, Iris D; Zhao, Jianhua; Asarnow, Daniel; Biel, Justin; Bowen, Alisa; Braxton, Julian R; Chen, Jen; Chio, Cynthia M; Chio, Un Seng; Deshpande, Ishan; Doan, Loan; Faust, Bryan; Flores, Sebastian; Jin, Mingliang; Kim, Kate; Lam, Victor L; Li, Fei; Li, Junrui; Li, Yen-Li; Li, Yang; Liu, Xi; Lo, Megan; Lopez, Kyle E; Melo, Arthur A; Moss, Frank R; Nguyen, Phuong; Paulino, Joana; Pawar, Komal Ishwar; Peters, Jessica K; Pospiech, Thomas H; Safari, Maliheh; Sangwan, Smriti; Schaefer, Kaitlin; Thomas, Paul V; Thwin, Aye C; Trenker, Raphael; Tse, Eric; Tsui, Tsz Kin Martin; Wang, Feng; Whitis, Natalie; Yu, Zanlin; Zhang, Kaihua; Zhang, Yang; Zhou, Fengbo; Saltzberg, Daniel; Hodder, Anthony J; Shun-Shion, Amber S; Williams, Daniel M; White, Kris M; Rosales, Romel; Kehrer, Thomas; Miorin, Lisa; Moreno, Elena; Patel, Arvind H; Rihn, Suzannah; Khalid, Mir M; Vallejo-Gracia, Albert; Fozouni, Parinaz; Simoneau, Camille R; Roth, Theodore L; Wu, David; Karim, Mohd Anisul; Ghoussaini, Maya; Dunham, Ian; Berardi, Francesco; Weigang, Sebastian; Chazal, Maxime; Park, Jisoo; Logue, James; Mcgrath, Marisa; Weston, Stuart; Haupt, Robert; Hastie, C James; Elliott, Matthew; Brown, Fiona; Burness, Kerry A; Reid, Elaine; Dorward, Mark; Johnson, Clare; Wilkinson, Stuart G; Geyer, Anna; Giesel, Daniel M; Baillie, Carla; Raggett, Samantha; Leech, Hannah; Toth, Rachel; Goodman, Nicola; Keough, Kathleen C; Lind, Abigail L; Klesh, Reyna J; Hemphill, Kafi R; Carlson-Stevermer, Jared; Oki, Jennifer; Holden, Kevin; Maures, Travis; Pollard, Katherine S; Sali, Andrej; Agard, David A; Cheng, Yifan; Fraser, James S; Frost, Adam; Jura, Natalia; Kortemme, Tanja; Manglik, Aashish; Southworth, Daniel R; Stroud, Robert M; Alessi, Dario R; Davies, Paul; Frieman, Matthew B; Ideker, Trey; Abate, Carmen; Jouvenet, Nolwenn; Kochs, Georg; Shoichet, Brian; Ott, Melanie; Palmarini, Massimo; Shokat, Kevan M; García-Sastre, Adolfo; Rassen, Jeremy A; Grosse, Robert; Rosenberg, Oren S; Verba, Kliment A; Basler, Christopher F; Vignuzzi, Marco; Peden, Andrew A; Beltrao, Pedro; Krogan, Nevan J
Mrp1-collateral sensitizers as a novel therapeutic approach in resistant cancer therapy: An in vitro and in vivo study in lung resistant tumor
2020-01-01 Riganti, C.; Giampietro, R.; Kopecka, J.; Costamagna, C.; Abatematteo, F. S.; Contino, M.; Abate, C.
Why PB28 Could Be a Covid 2019 Game Changer?
2020-01-01 Colabufo, Nicola Antonio; Leopoldo, Marcello; Ferorelli, Savina; Abate, Carmen; Contino, Marialessandra; Perrone, MARIA GRAZIA; Niso, Mauro; Perrone, Roberto; Berardi, Francesco
Cannabinoid Receptor Subtype 2 (CB2R) in a Multitarget Approach: Perspective of an Innovative Strategy in Cancer and Neurodegeneration
2020-01-01 Mangiatordi, Giuseppe Felice; Intranuovo, Francesca; Delre, Pietro; Abatematteo, Francesca Serena; Abate, Carmen; Niso, Mauro; Creanza, Teresa Maria; Ancona, Nicola; Stefanachi, Angela; Contino, Marialessandra
Design and synthesis of fluorescent ligands for the detection of cannabinoid type 2 receptor (CB2R)
2020-01-01 Spinelli, F.; Giampietro, R.; Stefanachi, A.; Riganti, C.; Kopecka, J.; Abatematteo, F. S.; Leonetti, F.; Colabufo, N. A.; Mangiatordi, G. F.; Nicolotti, O.; Perrone, M. G.; Brea, J.; Loza, M. I.; Infantino, V.; Abate, C.; Contino, M.
Proceedings from the Fourth International Symposium on sigma-2 Receptors: Role in Health and Disease
2020-01-01 Izzo, Nicholas J; Colom-Cadena, Martí; Riad, Aladdin A; Xu, Jinbin; Singh, Meharvan; Abate, Carmen; Cahill, Michael A; Spires-Jones, Tara L; Bowen, Wayne D; Mach, Robert H; Catalano, Susan M
PB28, the Sigma-1 and Sigma-2 Receptors Modulator With Potent Anti–SARS-CoV-2 Activity: A Review About Its Pharmacological Properties and Structure Affinity Relationships
2020-01-01 Abate, C.; Niso, M.; Abatematteo, F. S.; Contino, M.; Colabufo, N. A.; Berardi, F.
σ2 receptor and its role in cancer with focus on a multitarget directed ligand (Mtdl) approach
2021-01-01 Abatematteo, F. S.; Niso, M.; Lacivita, E.; Abate, C.
Multifunctional thiosemicarbazones targeting sigma receptors: in vitro and in vivo antitumor activities in pancreatic cancer models
2021-01-01 Niso, M.; Kopecka, J.; Abatematteo, F. S.; Berardi, F.; Riganti, C.; Abate, C.
DEVELOPMENT OF PHENOXYALKYLPIPERIDINES AS HIGH-AFFINITY SIGMA-1 (s1) RECEPTOR LIGANDS WITH POTENT ANTI-AMNESIC ACTIVITY
2021-01-01 Laghezza, Antonio; Abatematteo, Francesca S.; Mosier, Philip D.; Niso, Mauro; Brunetti, Leonardo; Berardi, Francesco; Loiodice, Fulvio; Contino, Marialessandra; Delprat, Benjamin; Maurice, Tangui; Abate, Carmen
Multi‐target directed ligands (Mtdls) binding the σ1 receptor as promising therapeutics: State of the art and perspectives
2021-01-01 Abatematteo, F. S.; Niso, M.; Contino, M.; Leopoldo, M.; Abate, C.
P-Glycoprotein, a biological and medicinal chemistry/radiochemistry point of view
2021-01-01 Abate, C.; Colabufo, N. A.; Contino, M.
New Pharmacological Strategies against Pancreatic Adenocarcinoma: The Multifunctional Thiosemicarbazone FA4
2022-01-01 Anobile, D. P.; Niso, M.; Puerta, A.; Fraga Rodrigues, S. M.; Abatematteo, F. S.; Avan, A.; Abate, C.; Riganti, C.; Giovannetti, E.
Development of novel phenoxyalkylpiperidines as high-affinity Sigma-1 (σ1) receptor ligands with potent anti-amnesic effect
2022-01-01 Abatematteo, F. S.; Mosier, P. D.; Niso, M.; Brunetti, L.; Berardi, F.; Loiodice, F.; Contino, M.; Delprat, B.; Maurice, T.; Laghezza, A.; Abate, C.
Design and Synthesis of Arylpiperazine Serotonergic/ Dopaminergic Ligands with Neuroprotective Properties
2022-01-01 Mastromarino, M.; Niso, M.; Abate, C.; Proschak, E.; Dubiel, M.; Stark, H.; Castro, M.; Lacivita, E.; Leopoldo, M.
The Intriguing Sigma-1 and Sigma-2 Receptors and Their Potential Therapeutic Roles 2.0
2023-01-01 Abate, Carmen; Maurice, Tangui
Synthesis and Biological Evaluation of Enantiomerically Pure (R)- and (S)-[18F]OF-NB1 for Imaging the GluN2B Subunit-Containing NMDA Receptors
2023-01-01 Korff, Marvin; Chaudhary, Ahmad; Li, Yinlong; Zhou, Xin; Zhao, Chunyu; Rong, Jian; Chen, Jiahui; Xiao, Zhiwei; Elghazawy, Nehal H.; Sippl, Wolfgang; Davenport, April T.; Daunais, James B.; Wang, Lu; Abate, Carmen; Ahmed, Hazem; Crowe, Ron; Schmidt, Thomas J.; Liang, Steven H.; Ametamey, Simon M.; Wünsch, Bernhard; Haider, Ahmed
Sigma-2 Receptor Ligand Binding Modulates Association between TSPO and TMEM97
2023-01-01 Thejer, B. M.; Infantino, V.; Santarsiero, A.; Pappalardo, I.; Abatematteo, F. S.; Teakel, S.; Van Oosterum, A.; Mach, R. H.; Denora, N.; Lee, B. C.; Resta, N.; Bagnulo, R.; Niso, M.; Contino, M.; Montsch, B.; Heffeter, P.; Abate, C.; Cahill, M. A.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| High-affinity sigma-1 (σ1) receptor ligands based on the σ1 antagonist PB212 | 1-gen-2019 | Niso, M.; Mosier, P. D.; Marottoli, Roberta; Ferorelli, S.; Cassano, G.; Gasparre, G.; Leopoldo, M.; Berardi, F.; Abate, C. | |
| NO1, a new sigma 2 receptor/TMEM97 fluorescent ligand, downregulates SOCE and promotes apoptosis in the triple negative breast cancer cell lines | 1-gen-2020 | Cantonero, C.; Camello, P. J.; Abate, C.; Berardi, F.; Salido, G. M.; Rosado, J. A.; Redondo, P. C. | |
| Comparative host-coronavirus protein interaction networks reveal pan-viral disease mechanisms | 1-gen-2020 | Gordon, David E; Hiatt, Joseph; Bouhaddou, Mehdi; Rezelj, Veronica V; Ulferts, Svenja; Braberg, Hannes; Jureka, Alexander S; Obernier, Kirsten; Guo, Jeffrey Z; Batra, Jyoti; Kaake, Robyn M; Weckstein, Andrew R; Owens, Tristan W; Gupta, Meghna; Pourmal, Sergei; Titus, Erron W; Cakir, Merve; Soucheray, Margaret; Mcgregor, Michael; Cakir, Zeynep; Jang, Gwendolyn; O'Meara, Matthew J; Tummino, Tia A; Zhang, Ziyang; Foussard, Helene; Rojc, Ajda; Zhou, Yuan; Kuchenov, Dmitry; Hüttenhain, Ruth; Xu, Jiewei; Eckhardt, Manon; Swaney, Danielle L; Fabius, Jacqueline M; Ummadi, Manisha; Tutuncuoglu, Beril; Rathore, Ujjwal; Modak, Maya; Haas, Paige; Haas, Kelsey M; Naing, Zun Zar Chi; Pulido, Ernst H; Shi, Ying; Barrio-Hernandez, Inigo; Memon, Danish; Petsalaki, Eirini; Dunham, Alistair; Marrero, Miguel Correa; Burke, David; Koh, Cassandra; Vallet, Thomas; Silvas, Jesus A; Azumaya, Caleigh M; Billesbølle, Christian; Brilot, Axel F; Campbell, Melody G; Diallo, Amy; Dickinson, Miles Sasha; Diwanji, Devan; Herrera, Nadia; Hoppe, Nick; Kratochvil, Huong T; Liu, Yanxin; Merz, Gregory E; Moritz, Michelle; Nguyen, Henry C; Nowotny, Carlos; Puchades, Cristina; Rizo, Alexandrea N; Schulze-Gahmen, Ursula; Smith, Amber M; Sun, Ming; Young, Iris D; Zhao, Jianhua; Asarnow, Daniel; Biel, Justin; Bowen, Alisa; Braxton, Julian R; Chen, Jen; Chio, Cynthia M; Chio, Un Seng; Deshpande, Ishan; Doan, Loan; Faust, Bryan; Flores, Sebastian; Jin, Mingliang; Kim, Kate; Lam, Victor L; Li, Fei; Li, Junrui; Li, Yen-Li; Li, Yang; Liu, Xi; Lo, Megan; Lopez, Kyle E; Melo, Arthur A; Moss, Frank R; Nguyen, Phuong; Paulino, Joana; Pawar, Komal Ishwar; Peters, Jessica K; Pospiech, Thomas H; Safari, Maliheh; Sangwan, Smriti; Schaefer, Kaitlin; Thomas, Paul V; Thwin, Aye C; Trenker, Raphael; Tse, Eric; Tsui, Tsz Kin Martin; Wang, Feng; Whitis, Natalie; Yu, Zanlin; Zhang, Kaihua; Zhang, Yang; Zhou, Fengbo; Saltzberg, Daniel; Hodder, Anthony J; Shun-Shion, Amber S; Williams, Daniel M; White, Kris M; Rosales, Romel; Kehrer, Thomas; Miorin, Lisa; Moreno, Elena; Patel, Arvind H; Rihn, Suzannah; Khalid, Mir M; Vallejo-Gracia, Albert; Fozouni, Parinaz; Simoneau, Camille R; Roth, Theodore L; Wu, David; Karim, Mohd Anisul; Ghoussaini, Maya; Dunham, Ian; Berardi, Francesco; Weigang, Sebastian; Chazal, Maxime; Park, Jisoo; Logue, James; Mcgrath, Marisa; Weston, Stuart; Haupt, Robert; Hastie, C James; Elliott, Matthew; Brown, Fiona; Burness, Kerry A; Reid, Elaine; Dorward, Mark; Johnson, Clare; Wilkinson, Stuart G; Geyer, Anna; Giesel, Daniel M; Baillie, Carla; Raggett, Samantha; Leech, Hannah; Toth, Rachel; Goodman, Nicola; Keough, Kathleen C; Lind, Abigail L; Klesh, Reyna J; Hemphill, Kafi R; Carlson-Stevermer, Jared; Oki, Jennifer; Holden, Kevin; Maures, Travis; Pollard, Katherine S; Sali, Andrej; Agard, David A; Cheng, Yifan; Fraser, James S; Frost, Adam; Jura, Natalia; Kortemme, Tanja; Manglik, Aashish; Southworth, Daniel R; Stroud, Robert M; Alessi, Dario R; Davies, Paul; Frieman, Matthew B; Ideker, Trey; Abate, Carmen; Jouvenet, Nolwenn; Kochs, Georg; Shoichet, Brian; Ott, Melanie; Palmarini, Massimo; Shokat, Kevan M; García-Sastre, Adolfo; Rassen, Jeremy A; Grosse, Robert; Rosenberg, Oren S; Verba, Kliment A; Basler, Christopher F; Vignuzzi, Marco; Peden, Andrew A; Beltrao, Pedro; Krogan, Nevan J | |
| Mrp1-collateral sensitizers as a novel therapeutic approach in resistant cancer therapy: An in vitro and in vivo study in lung resistant tumor | 1-gen-2020 | Riganti, C.; Giampietro, R.; Kopecka, J.; Costamagna, C.; Abatematteo, F. S.; Contino, M.; Abate, C. | |
| Why PB28 Could Be a Covid 2019 Game Changer? | 1-gen-2020 | Colabufo, Nicola Antonio; Leopoldo, Marcello; Ferorelli, Savina; Abate, Carmen; Contino, Marialessandra; Perrone, MARIA GRAZIA; Niso, Mauro; Perrone, Roberto; Berardi, Francesco | |
| Cannabinoid Receptor Subtype 2 (CB2R) in a Multitarget Approach: Perspective of an Innovative Strategy in Cancer and Neurodegeneration | 1-gen-2020 | Mangiatordi, Giuseppe Felice; Intranuovo, Francesca; Delre, Pietro; Abatematteo, Francesca Serena; Abate, Carmen; Niso, Mauro; Creanza, Teresa Maria; Ancona, Nicola; Stefanachi, Angela; Contino, Marialessandra | |
| Design and synthesis of fluorescent ligands for the detection of cannabinoid type 2 receptor (CB2R) | 1-gen-2020 | Spinelli, F.; Giampietro, R.; Stefanachi, A.; Riganti, C.; Kopecka, J.; Abatematteo, F. S.; Leonetti, F.; Colabufo, N. A.; Mangiatordi, G. F.; Nicolotti, O.; Perrone, M. G.; Brea, J.; Loza, M. I.; Infantino, V.; Abate, C.; Contino, M. | |
| Proceedings from the Fourth International Symposium on sigma-2 Receptors: Role in Health and Disease | 1-gen-2020 | Izzo, Nicholas J; Colom-Cadena, Martí; Riad, Aladdin A; Xu, Jinbin; Singh, Meharvan; Abate, Carmen; Cahill, Michael A; Spires-Jones, Tara L; Bowen, Wayne D; Mach, Robert H; Catalano, Susan M | |
| PB28, the Sigma-1 and Sigma-2 Receptors Modulator With Potent Anti–SARS-CoV-2 Activity: A Review About Its Pharmacological Properties and Structure Affinity Relationships | 1-gen-2020 | Abate, C.; Niso, M.; Abatematteo, F. S.; Contino, M.; Colabufo, N. A.; Berardi, F. | |
| σ2 receptor and its role in cancer with focus on a multitarget directed ligand (Mtdl) approach | 1-gen-2021 | Abatematteo, F. S.; Niso, M.; Lacivita, E.; Abate, C. | |
| Multifunctional thiosemicarbazones targeting sigma receptors: in vitro and in vivo antitumor activities in pancreatic cancer models | 1-gen-2021 | Niso, M.; Kopecka, J.; Abatematteo, F. S.; Berardi, F.; Riganti, C.; Abate, C. | |
| DEVELOPMENT OF PHENOXYALKYLPIPERIDINES AS HIGH-AFFINITY SIGMA-1 (s1) RECEPTOR LIGANDS WITH POTENT ANTI-AMNESIC ACTIVITY | 1-gen-2021 | Laghezza, Antonio; Abatematteo, Francesca S.; Mosier, Philip D.; Niso, Mauro; Brunetti, Leonardo; Berardi, Francesco; Loiodice, Fulvio; Contino, Marialessandra; Delprat, Benjamin; Maurice, Tangui; Abate, Carmen | |
| Multi‐target directed ligands (Mtdls) binding the σ1 receptor as promising therapeutics: State of the art and perspectives | 1-gen-2021 | Abatematteo, F. S.; Niso, M.; Contino, M.; Leopoldo, M.; Abate, C. | |
| P-Glycoprotein, a biological and medicinal chemistry/radiochemistry point of view | 1-gen-2021 | Abate, C.; Colabufo, N. A.; Contino, M. | |
| New Pharmacological Strategies against Pancreatic Adenocarcinoma: The Multifunctional Thiosemicarbazone FA4 | 1-gen-2022 | Anobile, D. P.; Niso, M.; Puerta, A.; Fraga Rodrigues, S. M.; Abatematteo, F. S.; Avan, A.; Abate, C.; Riganti, C.; Giovannetti, E. | |
| Development of novel phenoxyalkylpiperidines as high-affinity Sigma-1 (σ1) receptor ligands with potent anti-amnesic effect | 1-gen-2022 | Abatematteo, F. S.; Mosier, P. D.; Niso, M.; Brunetti, L.; Berardi, F.; Loiodice, F.; Contino, M.; Delprat, B.; Maurice, T.; Laghezza, A.; Abate, C. | |
| Design and Synthesis of Arylpiperazine Serotonergic/ Dopaminergic Ligands with Neuroprotective Properties | 1-gen-2022 | Mastromarino, M.; Niso, M.; Abate, C.; Proschak, E.; Dubiel, M.; Stark, H.; Castro, M.; Lacivita, E.; Leopoldo, M. | |
| The Intriguing Sigma-1 and Sigma-2 Receptors and Their Potential Therapeutic Roles 2.0 | 1-gen-2023 | Abate, Carmen; Maurice, Tangui | |
| Synthesis and Biological Evaluation of Enantiomerically Pure (R)- and (S)-[18F]OF-NB1 for Imaging the GluN2B Subunit-Containing NMDA Receptors | 1-gen-2023 | Korff, Marvin; Chaudhary, Ahmad; Li, Yinlong; Zhou, Xin; Zhao, Chunyu; Rong, Jian; Chen, Jiahui; Xiao, Zhiwei; Elghazawy, Nehal H.; Sippl, Wolfgang; Davenport, April T.; Daunais, James B.; Wang, Lu; Abate, Carmen; Ahmed, Hazem; Crowe, Ron; Schmidt, Thomas J.; Liang, Steven H.; Ametamey, Simon M.; Wünsch, Bernhard; Haider, Ahmed | |
| Sigma-2 Receptor Ligand Binding Modulates Association between TSPO and TMEM97 | 1-gen-2023 | Thejer, B. M.; Infantino, V.; Santarsiero, A.; Pappalardo, I.; Abatematteo, F. S.; Teakel, S.; Van Oosterum, A.; Mach, R. H.; Denora, N.; Lee, B. C.; Resta, N.; Bagnulo, R.; Niso, M.; Contino, M.; Montsch, B.; Heffeter, P.; Abate, C.; Cahill, M. A. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile