Sfoglia per Autore
Arylamides hybrids of two high-affinity sigma-2 receptor ligands as tools for the development of PET radiotracers
2011-01-01 Abate, CARMEN rosa; Ferorelli, Savina; Contino, Marialessandra; Marottoli, R; Colabufo, Nicola Antonio; Perrone, Roberto; Berardi, Francesco
Fluorescent Derivatives of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) as a Tool for Uptake and Cellular Localization Studies in Pancreatic Tumor Cells
2011-01-01 Abate, CARMEN rosa; Hornick, J; Spitzer, D; Hawkins, W; Niso, Mauro; Perrone, Roberto; Berardi, Francesco
Analogues of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Lacivita, Enza; Mosier, P. D.; Toscano, A.; Perrone, Roberto
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Delta8─Delta7 sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activity
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Contino, Marialessandra; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto; Berardi, Francesco
Synthesis and binding assays of novel 3,3-dimethylpiperidine derivatives with various lipophilicities as sigma-1 receptor ligands
2011-01-01 Ferorelli, Savina; Abate, CARMEN rosa; Pedone, Mp; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, Roberto; Berardi, Francesco
Effects of PB190 and PB212, new sigma receptor ligands, on glucocorticoid receptor-mediated gene transcription in LMCAT cells
2011-01-01 Skuza, G; Szymańska, M; Budziszewska, B; Abate, CARMEN rosa; Berardi, Francesco
Synthesis and pharmacological evaluation of methyl and fluoroethyl piperazine analogues as PET probes for sigma receptor imaging.
2012-01-01 Sv, Selivanova; A., Toscano; Abate, CARMEN rosa; Berardi, Francesco; A., Müller; S‐d, Krämer; R., Schibli; Sm, Ametamey
Classes of sigma2 ( o-2) receptor ligands: structure affinity relationship (SAfiR) studies and antiproliferative activity
2012-01-01 Abate, CARMEN rosa; Perrone, R; Berardi, Francesco
The sigma-1 receptor antagonist PB212 reduces the Ca2+-release through the inositol (1, 4, 5)-triphosphate receptor in SK-N-SH cells
2012-01-01 Gasparre, Giuseppe; Abate, CARMEN rosa; Berardi, Francesco; Cassano, Giuseppe
2-Aminopyridine derivatives as potential sigma2 receptor antagonists
2012-01-01 Abate, CARMEN rosa; Ferorelli, Savina; Niso, Mauro; Lovicario, C; Infantino, V; Convertini, P; Perrone, Roberto; Berardi, Francesco
Lysosomial membrane permeabilization is an early event in sigma-2 receptor ligand mediated cell death in pancreatic cancer
2012-01-01 Hornick, Jr; Vangveravong, S; Spitzer, D; Abate, CARMEN rosa; Berardi, Francesco; Goedegebuure, P; Mach, Rh; Hawkins, W. G.
Sigma Receptor Research: Progress Towards Diagnostic and Therapeutic Uses of Sigma Ligands
2012-01-01 Abate, CARMEN rosa
Investigation of sigma receptors agonist/antagonist activity through N-(6-methoxytetralin-1-yl)- and N-(6-methoxynaphthalen-1-yl)alkyl derivatives of polymethylpiperidines
2013-01-01 Niso, Mauro; Abate, CARMEN rosa; Ferorelli, Savina; Cassano, Giuseppe; Gasparre, Giuseppe; Perrone, Roberto; Berardi, Francesco
Development of 3,4-dihydroisoquinolin-1(2H)-one derivatives for the Positron Emission Tomography (PET) imaging of sigma-2 receptors
2013-01-01 Abate, CARMEN rosa; Selivanova, S. V.; Müller, ; Krämer, S. D.; Schibli, R; Marottoli, R; Perrone, R; Berardi, Francesco; Niso, Mauro; Ametamey, S. M.
Sigma-2 receptor agonists as possible antitumor agents in resistant tumors: Hints for collateral sensitivity
2013-01-01 Niso, Mauro; Abate, CARMEN rosa; Contino, Marialessandra; Ferorelli, Savina; Azzariti, Amalia; Perrone, Roberto; Colabufo, Nicola Antonio; Berardi, Francesco
Collateral Sensitivity of sigma2 Receptor ligands: Potentials in the Treatment of Multidrug Resistant Tumors
2014-01-01 Niso, Mauro; Chiara, Riganti; Abate, CARMEN rosa
The effects of new sigma (σ) receptor ligands, PB190 and PB212, in the models predictive of antidepressant activity.
2014-01-01 Skuza, G; Sadaj, W; Kabziński, M; Cassano, Giuseppe; Gasparre, Giuseppe; Abate, CARMEN rosa; Berardi, Francesco
Novel Derivatives of 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Improved Fluorescent and σ Receptors Binding Properties
2014-01-01 Abate, CARMEN rosa; Niso, Mauro; Marottoli, R; Riganti, C; Ghigo, D; Ferorelli, Savina; Ossato, G; Perrone, R; Lacivita, Enza; Lamb, Dc; Berardi, Francesco
The controversial identity of the sigma-2 receptor with PGRMC1: is the PGRMC1/sigma-2 protein, that binds Abeta oligomer, made of two independent molecular entities?
2015-01-01 Abate, CARMEN rosa; Niso, Mauro; Pati, MARIA LAURA; Colabufo, Nicola Antonio; Berardi, Francesco
From mixed sigma-2 receptor/P-glycoprotein targeting agents to selective P-glycoprotein modulators: small structural changes address the mechanism of interaction at the efflux pump
2015-01-01 Abate, C; Pati, Maria Laura; Contino, M; Colabufo, N A; Perrone, R; Niso, M; Berardi, F
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