MICIACCIA, MORENA

MICIACCIA, MORENA  

DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO  

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A further pocket or conformational plasticity by mapping COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet behavior 1-gen-2024 Solidoro, Roberta; Miciaccia, Morena; Bonaccorso, Carmela; Fortuna, Cosimo Gianluca; Armenise, Domenico; Centonze, Antonella; Ferorelli, Savina; Vitale, Paola; Rodrigues, Pryscila; Guimarães, Renilda; de Oliveira, Alana; da Paz, Mariana; Rangel, Luciana; Sathler, Plínio Cunha; Altomare, Angela; Perrone, Maria Grazia; Scilimati, Antonio
A Simplified Direct O2 Consumption-Based Assay to Test COX Inhibition 1-gen-2022 Perrone, M. G.; Miciaccia, M.; Ferorelli, S.; Scilimati, A.
An attempt to chemically state the cross-talk between monomers of COX homodimers by double/hybrid inhibitors mofezolac-spacer-mofezolac and mofezolac-spacer-arachidonic acid 1-gen-2021 Perrone, M. G.; Miciaccia, M.; Vitale, P.; Ferorelli, S.; Araujo, C. D. C. B.; de Almeida, G. S.; Souza Domingos, T. F.; da Silva, L. C. R. P.; de Padula, M.; Cabral, L. M.; Sathler, P. C.; Bonaccorso, C.; Fortuna, C. G.; Scilimati, A.
CHALLENGE TRANSABILITY OF “IN VITRO” TO “IN VIVO”: GENE-EXPRESSION BIOMARKERS AND FLUORESCENT IMAGE-GUIDED SURGERY PROBES IDENTIFICATION FOR OVARIAN CANCER 1-gen-2022 Scilimati, A.; Ferorelli, S.; Centonze, A.; Miciaccia, M.; Solidoro, R.; De Grassi, A.; Perrone, M. G.
Comparative Structural Analysis of hCOX‑1 and oCOX‑1 Isoenzymes 1-gen-2021 Miciaccia, M.; Belviso, B. D.; Caliandro, R.; Ferorelli, S.; Perrone, M. G.; Scilimati, A.
COX-1 INHIBITORS AS ANTI-PLATELET AGENTS IN COVID-19 1-gen-2022 Solidoro, R.; Armenise, D.; Ferorelli, S.; Miciaccia, M.; Perrone, M. G.; Scilimati, A
Cyclooxygenase Inhibition Safety and Efficacy in Inflammation-Based Psychiatric Disorders 1-gen-2020 Perrone, M. G.; Centonze, A.; Miciaccia, M.; Ferorelli, S.; Scilimati, A.
Cyclooxygenase-1 Inhibition: A Promising Theragnostic Approach for Ovarian Cancer 1-gen-2023 Miciaccia, Morena; Ferorelli, Savina; Centonze, Antonella; Solidoro, Roberta; Munzone, Cristina; Bonaccorso, Carmela; Gianluca Fortuna, Cosimo; Kleinmanns, Katrin; Bjørge, Line; Perrone, MARIA GRAZIA; Scilimati, Antonio
Design and synthesis of new [4,5-b] and [4,5-c] imidazopyridines as potential fluorophores/inhibitors for Human Cyclooxygenase-1. 1-gen-2023 Munzone, C.; Fortuna, C. G.; Bonaccorso, C.; Perrone, M. G.; Miciaccia, M.
DIPG-27. Diffuse Intrinsic Pontine Glioma (DIPG) challenge: from gene expression profile to drug. 1-gen-2023 Scilimati, Antonio; Armenise, Domenico; Baldelli, Olga; Centonze, Antonella; Derri, Davide; Ferorelli, Savina; Miciaccia, Morena; Solidoro, Roberta; Perrone, MARIA GRAZIA
Fluorescent imaging probes for in vivo ovarian cancer targeted detection and surgery 1-gen-2024 Solidoro, Roberta; Centonze, Antonella; Miciaccia, Morena; Baldelli, Olga Maria; Armenise, Domenico; Ferorelli, Savina; Perrone, Maria Grazia; Scilimati, Antonio
Fluorochrome Selection for Imaging Intraoperative Ovarian Cancer Probes 1-gen-2022 Perrone, Maria Grazia; Vitale, Paola; Miciaccia, Morena; Ferorelli, Savina; Centonze, Antonella; Solidoro, Roberta; Munzone, Cristina; Bonaccorso, Carmela; Fortuna, Cosimo Gianluca; Kleinmanns, Katrin; Bjørge, Line; Scilimati, Antonio
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment 1-gen-2024 Miciaccia, M.; Rizzo, F.; Centonze, A.; Cavallaro, G.; Contino, M.; Armenise, D.; Baldelli, O. M.; Solidoro, R.; Ferorelli, S.; Scarcia, P.; Agrimi, G.; Zingales, V.; Cimetta, E.; Ronsisvalle, S.; Sipala, F. M.; Polosa, P. L.; Fortuna, C. G.; Perrone, M. G.; Scilimati, A.
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment 1-gen-2024 Miciaccia, Morena; Rizzo, Francesca; Centonze, Antonella; Cavallaro, Gianfranco; Contino, Marialessandra; Armenise, Domenico; Baldelli, OLGA MARIA; Solidoro, Roberta; Ferorelli, Savina; Scarcia, Pasquale; Agrimi, Gennaro; Zingales, Veronica; Cimetta, Elisa; Ronsisvalle, Simone; Maria Sipala, Federica; LOGUERCIO POLOSA, Paola Anna Maria; Gianluca Fortuna, Cosimo; Perrone, MARIA GRAZIA; Scilimati, Antonio
Harmaline-based scaffold as Human Caseinolytic Protease P (hClpP) inducers for Diffuse Intrinsic Pontine Glioma (DIPG) treatment 1-gen-2023 Miciaccia, Morena; Centonze, Antonella; Baldelli, Olga; Solidoro, Roberta; Armenise, Domenico; Cavallaro, Gianfranco; Gianluca Fortuna, Cosimo; Ferorelli, Savina; Perrone, MARIA GRAZIA; Scilimati, Antonio
Human Caseinolytic Protease P (hClpP) Activity Modulating Agents For The Treatment Of DIPG/DMG 1-gen-2023 Perrone, M. G.; Centonze, A.; Miciaccia, M.; Baldelli, O.; Cavallaro, G.; Ferorelli, S.; Fortuna, C.; Scilimati, A.
Inside circular economy challenges: “green” application to valorise olive mill wastewater 1-gen-2022 Foti, Paola; Occhipinti, Paride S.; Russo, Nunziatina; Scilimati, Antonio; Miciaccia, Morena; Ferorelli, Savina; Caggia, Cinzia; Perrone, MARIA GRAZIA; Randazzo, Cinzia L.; Romeo, Flora V.
Learning from Nature: From a Marine Natural Product to Synthetic Cyclooxygenase-1 Inhibitors by Automated De Novo Design 1-gen-2021 Friedrich, L.; Cingolani, G.; Ko, Y. -H.; Iaselli, M.; Miciaccia, M.; Perrone, M. G.; Neukirch, K.; Bobinger, V.; Merk, D.; Hofstetter, R. K.; Werz, O.; Koeberle, A.; Scilimati, A.; Schneider, G.
m-Terphenylamines, Acting as Selective COX-1 Inhibitors, Block Microglia Inflammatory Response and Exert Neuroprotective Activity 1-gen-2023 Rocchi, Damiano; González, Juan F.; Martín-Cámara, Olmo; Perrone, MARIA GRAZIA; Miciaccia, Morena; Scilimati, Antonio; Decouty-Pérez, Celine; Parada, Esther; Egea, Javier; Carlos Menéndez, J.
Modulation of the activity of human mitochondrial protease complex ClpXP as potential therapeutic strategy for cancer 1-gen-2023 Rizzo, Francesca; Miciaccia, Morena; Cormio, Antonella; Ferorelli, Savina; Perrone, MARIA GRAZIA; Scilimati, Antonio; LOGUERCIO POLOSA, Paola Anna Maria