BERARDI, Francesco
BERARDI, Francesco
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
"Tritium radiolabeling of [3H]-1-cicloesil-4-[3-(5-methoxy-1,2, 3,4,-tetraidronaftalen-1-il)-n-propil] piperazine ([3H]-PB28)as potent sigma-2 receptor ligand
2008-01-01 Abate, C; Berardi, Francesco; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto
1-(2-Methoxyphenyl)-4-alkylpiperazines: effect of the N-4 substituent on the affinity and selectivity for dopamine D4 receptor
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Aryl-4-[(1-tetralinyl)alkyl]piperazines: alkylamido and alkylamino derivatives. Synthesis, 5-HT1A receptor affinity, and selectivity. 3
1996-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V; Fornaretto, Mg; Caccia, C; Mcarthur, Ra
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Delta8─Delta7 sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activity
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Contino, Marialessandra; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto; Berardi, Francesco
1-Cyclohexylpiperazine and 3,3-Dimethylpiperidine Derivatives as Sigma-1 (σ1) and Sigma-2 (σ2) Receptor Ligands: A Review
2009-01-01 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
1-Cyclohexylpiperazine and 3,3-dimethylpiperidine derivatives as sigma-1 and sigma-2 receptor ligand: a review
2009-01-01 Berardi, Francesco; Abate, C; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
1-Phenylalkoxy-2-beta-phenylethyl derivatives as P-gP inhibitors useful in drug resistance events
2007-01-01 Berardi, Francesco; Colabufo, Nicola Antonio; Perrone, Roberto; A., Balsamo; S., Rapposelli
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors
2005-01-01 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
2-(Aryloxy)ethylamine derivatives: ring opened congeners of long chain 1-arylpiperazines with high 5-HT1A receptor affinity and selectivity versus D2 and a1 receptors
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
2-[(3-Methoxyphenylethyl)phenoxy]-based ABCB1 inhibitors: effect of different basic side-chains on their biological properties
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A.
2-Aminopyridine derivatives as potential sigma2 receptor antagonists
2012-01-01 Abate, CARMEN rosa; Ferorelli, Savina; Niso, Mauro; Lovicario, C; Infantino, V; Convertini, P; Perrone, Roberto; Berardi, Francesco
4-(Tetralin-1-yl)- and 4-(Naphthalen-1-yl)alkyl Derivatives of 1-Cycloheylpiperazine as sigma receptor Ligands with Agonist sigma 2 Activity
2004-01-01 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, N. C.; Contino, Marialessandra; Perrone, Roberto; Tortorella, V.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
4-[omega-Tetralin-1-yl]-1-benzylpiperazines and related compounds as 5-HT1A/D-2 ligands
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lograno, M.; Tortorella, V.
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo
5 HT1A receptor, an old target for new therapeutic agents
2008-01-01 Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Perrone, R.
5-HT and DA receptor affinity of arylpiperazine derivatives with terminal benzamide fragment
1994-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V.; Lograno, Marcello Diego; Daniele, E.; Govoni, S.
5-HT1A and D-2 receptor affinity of o-methoxyphenyl derivatives with terminal benzamide fragment on N-4 alkyl chain. 2
1995-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V; Lograno, Marcello Diego; Daniele, E; Govoni, S.