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1-[(1S)-(4-Fluorophenyl)-((1′S)-1′-naphthalen-1-yl-ethylamino)-methyl]-naphthalen-2-trifluoromethanesulfonate
2023-01-01 Cardellicchio, Cosimo; Capozzi, Maria Annunziata M.
1-Aryl-4-[(1-tetralinyl)alkyl]piperazines: alkylamido and alkylamino derivatives. Synthesis, 5-HT1A receptor affinity, and selectivity. 3
1996-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V; Fornaretto, Mg; Caccia, C; Mcarthur, Ra
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ(8)-Δ(7) Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity
2011-01-01 Abate, C; Niso, M; Contino, M; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, R; Berardi, Francesco
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Delta8─Delta7 sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activity
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Contino, Marialessandra; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto; Berardi, Francesco
1-Cyclohexylpiperazine and 3,3-Dimethylpiperidine Derivatives as Sigma-1 (σ1) and Sigma-2 (σ2) Receptor Ligands: A Review
2009-01-01 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
1-Cyclohexylpiperazine and 3,3-dimethylpiperidine derivatives as sigma-1 and sigma-2 receptor ligand: a review
2009-01-01 Berardi, Francesco; Abate, C; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
1-Oxa-2,6-Diazaspiro[3.3]heptane as a New Potential Piperazine Bioisostere – Flow-Assisted Preparation and Derivatisation by Strain-Release of Azabicyclo[1.1.0]butanes
2024-01-01 Graziano, Elena; Natho, Philipp; Andresini, Michael; Mastrolorito, Fabrizio; Mahdi, Iktedar; Mesto, Ernesto; Colella, Marco; Degennaro, Leonardo; Nicolotti, Orazio; Luisi, Renzo
1-Pentanoyl-N-{[2’-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}-pyrrolidine-2-carboxamide: Investigation of Structural Variations
2011-01-01 Catalano, Alessia; Carocci, Alessia; DI MOLA, A; Bruno, C; Vanderheyden, P. M. L.; Franchini, Carlo
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
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