IACOBAZZI, ROSA MARIA
IACOBAZZI, ROSA MARIA
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
A model radiopharmaceutical agent targeted to translocator protein 18 kDa (TSPO)
2013-01-01 Piccinonna, S; Margiotta, Nicola; Denora, Nunzio; Iacobazzi, Rm; Pacifico, Concetta; Trapani, Giuseppe; Natile, Giovanni
A new complex of curcumin with sulfobutylether-β-cyclodextrin: characterization studies and in vitro evaluation of cytotoxic and antioxidant activity on HepG-2 cells
2014-01-01 Cutrignelli, Annalisa; Lopedota, Angela Assunta; Denora, Nunzio; Iacobazzi, Rm; Fanizza, Elisabetta; Laquintana, Valentino; Perrone, M; Maggi, V; Franco, Massimo
Antitumor Potential of Conjugable Valinomycins Bearing Hydroxyl Sites: In Vitro Studies
2013-01-01 Iacobazzi, R. M.; Annese, C; Azzariti, A; D'Accolti, Lucia; Franco, Massimo; Fusco, C; LA PIANA, Gianluigi; Laquintana, Valentino; Denora, Nunzio
Aurora kinase B inhibition reduces the proliferation of metastatic melanoma cells and enhances the response to chemotherapy
2015-01-01 Porcelli, L; Guida, Gabriella; Quatrale, Ae; Cocco, Tiziana Maria; Sidella, L; Maida, Immacolata; Iacobazzi, Rm; Ferretta, A; Stolfa, Da; Strippoli, S; Guida, S; Tommasi, S; Guida, M; Azzariti, A.
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitors
2018-01-01 Mangiatordi, G. F.; Trisciuzzi, D.; Iacobazzi, R.; Denora, N.; Pisani, L.; Catto, M.; Leonetti, F.; Alberga, D.; Nicolotti, O.
Bortezomib Aqueous Solubility in the Presence and Absence of D-Mannitol: A Clarification With Formulation Implications
2021-01-01 Lopalco, A.; Iacobazzi, R. M.; Denora, N.; Stella, V. J.
Bridging Pharmaceutical Chemistry with Drug and Nanoparticle Targeting to Investigate the Role of the 18-kDa Translocator Protein TSPO.
2017-01-01 Iacobazzi, R. M; Lopalco, A.; Cutrignelli, A.; Laquintana, V.; Lopedota, A.; Franco, M.; Denora, N.
CAFs and TGF-β Signaling Activation by Mast Cells Contribute to Resistance to Gemcitabine/Nabpaclitaxel in Pancreatic Cancer
2019-01-01 Porcelli, Letizia; Iacobazzi, Rosa Maria; Di Fonte, Roberta; Serrati', Simona; Intini, Angelica; Solimando, Antonio Giovanni; Brunetti, Oronzo; Calabrese, Angela; Leonetti, Francesco; Azzariti, Amalia; Silvestris, Nicola
Circulating extracellular vesicles expressing PD1 and PD-L1 predict response and mediate resistance to checkpoint inhibitors immunotherapy in metastatic melanoma
2022-01-01 Serratì, Simona; Guida, Michele; Di Fonte, Roberta; De Summa, Simona; Strippoli, Sabino; Iacobazzi, ROSA MARIA; Quarta, Alessandra; De Risi, Ivana; Guida, Gabriella; Paradiso, Angelo; Porcelli, Letizia; Azzariti, Amalia
Colonic budesonide delivery by multistimuli alginate/Eudragit® FS 30D/inulin-based microspheres as a paediatric formulation
2023-01-01 D'Amico, Vita; Arduino, Ilaria; Vacca, Mirco; Iacobazzi, Rosa Maria; Altamura, Davide; Lopalco, Antonio; Rizzi, Rosanna; Cutrignelli, Annalisa; Laquintana, Valentino; Franco, Massimo; De Angelis, Maria; Denora, Nunzio; Lopedota, Angela Assunta
Delivery of proapoptotic agents in glioma cell lines by TSPO ligand–dextran nanogels
2018-01-01 Lopalco, Antonio; Cutrignelli, Annalisa; Denora, Nunzio; Perrone, Mara; Iacobazzi, Rosa Maria; Fanizza, Elisabetta; Lopedota, Angela; Depalo, Nicoletta; De Candia, Modesto; Franco, Massimo; Laquintana, Valentino
Design and synthesis of grafted TSPO ligand-amino functionalized silica-coated quantum dots
2013-01-01 Denora, Nunzio; Iacobazzi, Rm; Laquintana, Valentino; Fanizza, Elisabetta; Depalo, N; Sriccoli, M; Curri, Ml; Cutrignelli, Annalisa; Lopedota, Angela Assunta; Franco, Massimo
Design and synthesis of grafted TSPO ligand-amino functionalized silica-coated quantum dots
2013-01-01 Denora, Nunzio; Iacobazzi, R. M.; Laquintana, Valentino; Fanizza, F.; Depalo, N.; Striccoli, M.; Curri, M. L.; Cutrignelli, Annalisa; Lopedota, Angela Assunta; Franco, Massimo
Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
2019-01-01 Oukoloff, Killian; Coquelle, Nicolas; Bartolini, Manuela; Naldi, Marina; Le Guevel, Rémy; Bach, Stéphane; Josselin, Béatrice; Ruchaud, Sandrine; Catto, Marco; Pisani, Leonardo; Denora, Nunzio; Iacobazzi, Rosa Maria; Silman, Israel; Sussman, Joel L.; Buron, Frédéric; Colletier, Jacques-Philippe; Jean, Ludovic; Routier, Sylvain; Renard, Pierre-Yves
DEVELOPMENT OF MUCOADHESIVE MICROSPHERES AS CELECOXIB DELIVERY SYSTEMS IN THE BLADDER
2013-01-01 Lopedota, Angela Assunta; Iacobazzi, R. M.; Denora, Nunzio; Cutrignelli, Annalisa; Laquintana, Valentino; Franco, Massimo
Development of mucoadhesive microspheres as celecoxib delivery systems in the bladder
2013-01-01 Lopedota, Angela Assunta; Iacobazzi, R. M.; Denora, Nunzio; Cutrignelli, Annalisa; Laquintana, Valentino; Franco, Massimo
Development of New Theranostic Nanosystems Composed of Semiconducting-Magnetic Heterostructures and Cyclic RGD Peptide for Integrin Targeting
2014-01-01 Depalo, N; Valente, G; De Paola, I; Comparelli, R; Striccoli, M; Agostiano, Angela; Denora, Nunzio; Laquintana, Valentino; Iacobazzi, Rm; Saviano, M; Del Gatto, A; Curri, Ml; Zaccaro, L.
Direct cyclodextrin based powder extrusion 3D printing of budesonide loaded mini-tablets for the treatment of eosinophilic colitis in paediatric patients
2023-01-01 Pistone, M.; Racaniello, G. F.; Rizzi, R.; Iacobazzi, R. M.; Arduino, I.; Lopalco, A.; Lopedota, A. A.; Denora, N.
Drug delivery nanovectors based on SPIONS for targeted therapy of hepatocellular carcinoma
2017-01-01 Depalo, N.; Striccoli, M.; Curri, M. L.; Iacobazzi, R. M.; Arduino, Ilaria; Laquintana, V.; Cutrignelli, A.; Lopedota, A.; Franco, M.; Denora, N.; Porcelli, L.; Azzariti, A.; Valente, G.; Fanizza, E.; Villa, S.; Canepa, F.
Exploring Basic Tail Modifications of Coumarin-based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-soluble, Brain-permeant Neuroprotective Multitarget Agents
2016-01-01 Pisani, Leonardo; Farina, Roberta; Catto, Marco; Iacobazzi, ROSA MARIA; Nicolotti, Orazio; Cellamare, Saverio; Mangiatordi, Giuseppe Felice; Denora, Nunzio; Soto Otero, R; Siragusa, L; Altomare, Cosimo Damiano; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A model radiopharmaceutical agent targeted to translocator protein 18 kDa (TSPO) | 1-gen-2013 | Piccinonna, S; Margiotta, Nicola; Denora, Nunzio; Iacobazzi, Rm; Pacifico, Concetta; Trapani, Giuseppe; Natile, Giovanni | |
A new complex of curcumin with sulfobutylether-β-cyclodextrin: characterization studies and in vitro evaluation of cytotoxic and antioxidant activity on HepG-2 cells | 1-gen-2014 | Cutrignelli, Annalisa; Lopedota, Angela Assunta; Denora, Nunzio; Iacobazzi, Rm; Fanizza, Elisabetta; Laquintana, Valentino; Perrone, M; Maggi, V; Franco, Massimo | |
Antitumor Potential of Conjugable Valinomycins Bearing Hydroxyl Sites: In Vitro Studies | 1-gen-2013 | Iacobazzi, R. M.; Annese, C; Azzariti, A; D'Accolti, Lucia; Franco, Massimo; Fusco, C; LA PIANA, Gianluigi; Laquintana, Valentino; Denora, Nunzio | |
Aurora kinase B inhibition reduces the proliferation of metastatic melanoma cells and enhances the response to chemotherapy | 1-gen-2015 | Porcelli, L; Guida, Gabriella; Quatrale, Ae; Cocco, Tiziana Maria; Sidella, L; Maida, Immacolata; Iacobazzi, Rm; Ferretta, A; Stolfa, Da; Strippoli, S; Guida, S; Tommasi, S; Guida, M; Azzariti, A. | |
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitors | 1-gen-2018 | Mangiatordi, G. F.; Trisciuzzi, D.; Iacobazzi, R.; Denora, N.; Pisani, L.; Catto, M.; Leonetti, F.; Alberga, D.; Nicolotti, O. | |
Bortezomib Aqueous Solubility in the Presence and Absence of D-Mannitol: A Clarification With Formulation Implications | 1-gen-2021 | Lopalco, A.; Iacobazzi, R. M.; Denora, N.; Stella, V. J. | |
Bridging Pharmaceutical Chemistry with Drug and Nanoparticle Targeting to Investigate the Role of the 18-kDa Translocator Protein TSPO. | 1-gen-2017 | Iacobazzi, R. M; Lopalco, A.; Cutrignelli, A.; Laquintana, V.; Lopedota, A.; Franco, M.; Denora, N. | |
CAFs and TGF-β Signaling Activation by Mast Cells Contribute to Resistance to Gemcitabine/Nabpaclitaxel in Pancreatic Cancer | 1-gen-2019 | Porcelli, Letizia; Iacobazzi, Rosa Maria; Di Fonte, Roberta; Serrati', Simona; Intini, Angelica; Solimando, Antonio Giovanni; Brunetti, Oronzo; Calabrese, Angela; Leonetti, Francesco; Azzariti, Amalia; Silvestris, Nicola | |
Circulating extracellular vesicles expressing PD1 and PD-L1 predict response and mediate resistance to checkpoint inhibitors immunotherapy in metastatic melanoma | 1-gen-2022 | Serratì, Simona; Guida, Michele; Di Fonte, Roberta; De Summa, Simona; Strippoli, Sabino; Iacobazzi, ROSA MARIA; Quarta, Alessandra; De Risi, Ivana; Guida, Gabriella; Paradiso, Angelo; Porcelli, Letizia; Azzariti, Amalia | |
Colonic budesonide delivery by multistimuli alginate/Eudragit® FS 30D/inulin-based microspheres as a paediatric formulation | 1-gen-2023 | D'Amico, Vita; Arduino, Ilaria; Vacca, Mirco; Iacobazzi, Rosa Maria; Altamura, Davide; Lopalco, Antonio; Rizzi, Rosanna; Cutrignelli, Annalisa; Laquintana, Valentino; Franco, Massimo; De Angelis, Maria; Denora, Nunzio; Lopedota, Angela Assunta | |
Delivery of proapoptotic agents in glioma cell lines by TSPO ligand–dextran nanogels | 1-gen-2018 | Lopalco, Antonio; Cutrignelli, Annalisa; Denora, Nunzio; Perrone, Mara; Iacobazzi, Rosa Maria; Fanizza, Elisabetta; Lopedota, Angela; Depalo, Nicoletta; De Candia, Modesto; Franco, Massimo; Laquintana, Valentino | |
Design and synthesis of grafted TSPO ligand-amino functionalized silica-coated quantum dots | 1-gen-2013 | Denora, Nunzio; Iacobazzi, Rm; Laquintana, Valentino; Fanizza, Elisabetta; Depalo, N; Sriccoli, M; Curri, Ml; Cutrignelli, Annalisa; Lopedota, Angela Assunta; Franco, Massimo | |
Design and synthesis of grafted TSPO ligand-amino functionalized silica-coated quantum dots | 1-gen-2013 | Denora, Nunzio; Iacobazzi, R. M.; Laquintana, Valentino; Fanizza, F.; Depalo, N.; Striccoli, M.; Curri, M. L.; Cutrignelli, Annalisa; Lopedota, Angela Assunta; Franco, Massimo | |
Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3 | 1-gen-2019 | Oukoloff, Killian; Coquelle, Nicolas; Bartolini, Manuela; Naldi, Marina; Le Guevel, Rémy; Bach, Stéphane; Josselin, Béatrice; Ruchaud, Sandrine; Catto, Marco; Pisani, Leonardo; Denora, Nunzio; Iacobazzi, Rosa Maria; Silman, Israel; Sussman, Joel L.; Buron, Frédéric; Colletier, Jacques-Philippe; Jean, Ludovic; Routier, Sylvain; Renard, Pierre-Yves | |
DEVELOPMENT OF MUCOADHESIVE MICROSPHERES AS CELECOXIB DELIVERY SYSTEMS IN THE BLADDER | 1-gen-2013 | Lopedota, Angela Assunta; Iacobazzi, R. M.; Denora, Nunzio; Cutrignelli, Annalisa; Laquintana, Valentino; Franco, Massimo | |
Development of mucoadhesive microspheres as celecoxib delivery systems in the bladder | 1-gen-2013 | Lopedota, Angela Assunta; Iacobazzi, R. M.; Denora, Nunzio; Cutrignelli, Annalisa; Laquintana, Valentino; Franco, Massimo | |
Development of New Theranostic Nanosystems Composed of Semiconducting-Magnetic Heterostructures and Cyclic RGD Peptide for Integrin Targeting | 1-gen-2014 | Depalo, N; Valente, G; De Paola, I; Comparelli, R; Striccoli, M; Agostiano, Angela; Denora, Nunzio; Laquintana, Valentino; Iacobazzi, Rm; Saviano, M; Del Gatto, A; Curri, Ml; Zaccaro, L. | |
Direct cyclodextrin based powder extrusion 3D printing of budesonide loaded mini-tablets for the treatment of eosinophilic colitis in paediatric patients | 1-gen-2023 | Pistone, M.; Racaniello, G. F.; Rizzi, R.; Iacobazzi, R. M.; Arduino, I.; Lopalco, A.; Lopedota, A. A.; Denora, N. | |
Drug delivery nanovectors based on SPIONS for targeted therapy of hepatocellular carcinoma | 1-gen-2017 | Depalo, N.; Striccoli, M.; Curri, M. L.; Iacobazzi, R. M.; Arduino, Ilaria; Laquintana, V.; Cutrignelli, A.; Lopedota, A.; Franco, M.; Denora, N.; Porcelli, L.; Azzariti, A.; Valente, G.; Fanizza, E.; Villa, S.; Canepa, F. | |
Exploring Basic Tail Modifications of Coumarin-based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-soluble, Brain-permeant Neuroprotective Multitarget Agents | 1-gen-2016 | Pisani, Leonardo; Farina, Roberta; Catto, Marco; Iacobazzi, ROSA MARIA; Nicolotti, Orazio; Cellamare, Saverio; Mangiatordi, Giuseppe Felice; Denora, Nunzio; Soto Otero, R; Siragusa, L; Altomare, Cosimo Damiano; Carotti, Angelo |