LACIVITA, ENZA
LACIVITA, ENZA
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors
2005-01-01 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
3-(1H-indol-3-yl)-2-[3-(4-nitrophenyl)ureido]propanamide enantiomers with human formyl-peptide receptor agonist activity: Molecular modeling of chiral recognition by FPR2.
2013-01-01 Schepetkin, Ia; Kirpotina, Ln; Khlebnikov, Ai; Leopoldo, Marcello; Lucente, E; Lacivita, Enza; De Giorgio, P; Quinn, M. T.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
5 HT1A receptor, an old target for new therapeutic agents
2008-01-01 Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Perrone, R.
5-HT7 receptor activation: procognitive and antiamnesic effects
2015-01-01 Meneses, A; Perez Garcia, G; Liy Salmeron, G; Ponce López, T; Lacivita, Enza; Leopoldo, Marcello
5-HT7 receptor modulators: a medicinal chemistry survey of recent patent literature (2004 - 2009)
2010-01-01 Leopoldo, Marcello; Lacivita, Enza; Berardi, Francesco; Perrone, Roberto
5-HT7 Receptors Regulate Excitatory-Inhibitory Balance in Mouse Spinal Cord Dorsal Horn
2022-01-01 Comitato, Antonella; Lacivita, Enza; Leopoldo, Marcello; Bardoni, Rita
Activatable fluorescent probes: a new concept in optical molecular imaging
2012-01-01 Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Perrone, R.
Activation of 5-HT7 receptor by administration of its selective agonist, LP-211, modifies explorative-curiosity behavior in rats in two paradigms which differ in visuospatial parameters
2018-01-01 Carbone, Cristiana; Adinolfi, Annalisa; Cinque, Stefano; Lacivita, Enza; Alleva, Enrico; Leopoldo, Marcello; Adriani, Walter
Activation of 5-HT7 receptor stimulates neurite elongation through mTOR, Cdc42 and actin filaments dynamics.
2015-01-01 Speranza, L; Giuliano, T; Volpicelli, F; De Stefano, Me; Lombardi, L; Chambery, A; Lacivita, Enza; Leopoldo, Marcello; Bellenchi, Gc; di Porzio, U; Crispino, M; Perrone Capano, C.
Activation of 5-HT7 serotonin receptors reverses metabotropic glutamate receptor-mediated synaptic plasticity in wild-type and Fmr1 knockout mice, a model of Fragile X Syndrome
2012-01-01 Costa, L; Spatuzza, M; D'Antoni, S; Bonaccorso, Cm; Trovato, C; Musumeci, Sa; Leopoldo, Marcello; Lacivita, Enza; Catania, Mv; Ciranna, L.
Activation of Serotonin 5-HT7 Receptors Modulates Hippocampal Synaptic Plasticity by Stimulation of Adenylate Cyclases and Rescues Learning and Behavior in a Mouse Model of Fragile X Syndrome
2018-01-01 Costa, Lara; Sardone, Lara Maria; Bonaccorso, Carmela Maria; D’Antoni, Simona; Spatuzza, Michela; Gulisano, Walter; Tropea, Maria Rosaria; Puzzo, Daniela; Leopoldo, Marcello; Lacivita, Enza; Catania, Maria Vincenza; Ciranna, Lucia
Allosteric Modulators of Serotonin Receptors: A Medicinal Chemistry Survey
2024-01-01 Brunetti, Leonardo; Francavilla, Fabio; Leopoldo, Marcello; Lacivita, Enza
Analogues of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Lacivita, Enza; Mosier, P. D.; Toscano, A.; Perrone, Roberto
Arylpiperazine agonists of the serotonin 5-HT1A receptor preferentially activate cAMP signaling versus recruitment of β-arrestin-2
2015-01-01 Stroth, Nikolas; Niso, Mauro; Colabufo, Nicola Antonio; Perrone, Roberto; Svenningsson, Per; Lacivita, Enza; Leopoldo, Marcello
Aurantiamide-related dipeptide derivatives are formyl peptide receptor 1 antagonists
2019-01-01 Mastromarino, Margherita; Kirpotina, Liliya N.; Schepetkin, Igor A.; Quinn, Mark T.; Lacivita, Enza; Leopoldo, Marcello
Behavioral, Anti-Inflammatory, and Neuroprotective Effects of a Novel FPR2 Agonist in Two Mouse Models of Autism
2022-01-01 Cristiano, C.; Volpicelli, F.; Crispino, M.; Lacivita, E.; Russo, R.; Leopoldo, M.; Calignano, A.; Perrone-Capano, C.
BEHAVIOURAL EFFECTS OF TWO NOVEL AGONISTS FOR SEROTONIN RECEPTOR 7 IN MICE
2011-01-01 Adriani, W; Travaglini, D; Lacivita, Enza; Leopoldo, Marcello; Laviola, G.
Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: Synthesis and binding affinities for 5-HT7 and 5-HT1A receptors
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Design and Synthesis of Arylpiperazine Serotonergic/ Dopaminergic Ligands with Neuroprotective Properties
2022-01-01 Mastromarino, M.; Niso, M.; Abate, C.; Proschak, E.; Dubiel, M.; Stark, H.; Castro, M.; Lacivita, E.; Leopoldo, M.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors | 1-gen-2005 | Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto | |
| 3-(1H-indol-3-yl)-2-[3-(4-nitrophenyl)ureido]propanamide enantiomers with human formyl-peptide receptor agonist activity: Molecular modeling of chiral recognition by FPR2. | 1-gen-2013 | Schepetkin, Ia; Kirpotina, Ln; Khlebnikov, Ai; Leopoldo, Marcello; Lucente, E; Lacivita, Enza; De Giorgio, P; Quinn, M. T. | |
| 4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization | 1-gen-2007 | Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R. | |
| 5 HT1A receptor, an old target for new therapeutic agents | 1-gen-2008 | Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Perrone, R. | |
| 5-HT7 receptor activation: procognitive and antiamnesic effects | 1-gen-2015 | Meneses, A; Perez Garcia, G; Liy Salmeron, G; Ponce López, T; Lacivita, Enza; Leopoldo, Marcello | |
| 5-HT7 receptor modulators: a medicinal chemistry survey of recent patent literature (2004 - 2009) | 1-gen-2010 | Leopoldo, Marcello; Lacivita, Enza; Berardi, Francesco; Perrone, Roberto | |
| 5-HT7 Receptors Regulate Excitatory-Inhibitory Balance in Mouse Spinal Cord Dorsal Horn | 1-gen-2022 | Comitato, Antonella; Lacivita, Enza; Leopoldo, Marcello; Bardoni, Rita | |
| Activatable fluorescent probes: a new concept in optical molecular imaging | 1-gen-2012 | Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Perrone, R. | |
| Activation of 5-HT7 receptor by administration of its selective agonist, LP-211, modifies explorative-curiosity behavior in rats in two paradigms which differ in visuospatial parameters | 1-gen-2018 | Carbone, Cristiana; Adinolfi, Annalisa; Cinque, Stefano; Lacivita, Enza; Alleva, Enrico; Leopoldo, Marcello; Adriani, Walter | |
| Activation of 5-HT7 receptor stimulates neurite elongation through mTOR, Cdc42 and actin filaments dynamics. | 1-gen-2015 | Speranza, L; Giuliano, T; Volpicelli, F; De Stefano, Me; Lombardi, L; Chambery, A; Lacivita, Enza; Leopoldo, Marcello; Bellenchi, Gc; di Porzio, U; Crispino, M; Perrone Capano, C. | |
| Activation of 5-HT7 serotonin receptors reverses metabotropic glutamate receptor-mediated synaptic plasticity in wild-type and Fmr1 knockout mice, a model of Fragile X Syndrome | 1-gen-2012 | Costa, L; Spatuzza, M; D'Antoni, S; Bonaccorso, Cm; Trovato, C; Musumeci, Sa; Leopoldo, Marcello; Lacivita, Enza; Catania, Mv; Ciranna, L. | |
| Activation of Serotonin 5-HT7 Receptors Modulates Hippocampal Synaptic Plasticity by Stimulation of Adenylate Cyclases and Rescues Learning and Behavior in a Mouse Model of Fragile X Syndrome | 1-gen-2018 | Costa, Lara; Sardone, Lara Maria; Bonaccorso, Carmela Maria; D’Antoni, Simona; Spatuzza, Michela; Gulisano, Walter; Tropea, Maria Rosaria; Puzzo, Daniela; Leopoldo, Marcello; Lacivita, Enza; Catania, Maria Vincenza; Ciranna, Lucia | |
| Allosteric Modulators of Serotonin Receptors: A Medicinal Chemistry Survey | 1-gen-2024 | Brunetti, Leonardo; Francavilla, Fabio; Leopoldo, Marcello; Lacivita, Enza | |
| Analogues of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers | 1-gen-2011 | Abate, CARMEN rosa; Niso, Mauro; Lacivita, Enza; Mosier, P. D.; Toscano, A.; Perrone, Roberto | |
| Arylpiperazine agonists of the serotonin 5-HT1A receptor preferentially activate cAMP signaling versus recruitment of β-arrestin-2 | 1-gen-2015 | Stroth, Nikolas; Niso, Mauro; Colabufo, Nicola Antonio; Perrone, Roberto; Svenningsson, Per; Lacivita, Enza; Leopoldo, Marcello | |
| Aurantiamide-related dipeptide derivatives are formyl peptide receptor 1 antagonists | 1-gen-2019 | Mastromarino, Margherita; Kirpotina, Liliya N.; Schepetkin, Igor A.; Quinn, Mark T.; Lacivita, Enza; Leopoldo, Marcello | |
| Behavioral, Anti-Inflammatory, and Neuroprotective Effects of a Novel FPR2 Agonist in Two Mouse Models of Autism | 1-gen-2022 | Cristiano, C.; Volpicelli, F.; Crispino, M.; Lacivita, E.; Russo, R.; Leopoldo, M.; Calignano, A.; Perrone-Capano, C. | |
| BEHAVIOURAL EFFECTS OF TWO NOVEL AGONISTS FOR SEROTONIN RECEPTOR 7 IN MICE | 1-gen-2011 | Adriani, W; Travaglini, D; Lacivita, Enza; Leopoldo, Marcello; Laviola, G. | |
| Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: Synthesis and binding affinities for 5-HT7 and 5-HT1A receptors | 1-gen-2007 | Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
| Design and Synthesis of Arylpiperazine Serotonergic/ Dopaminergic Ligands with Neuroprotective Properties | 1-gen-2022 | Mastromarino, M.; Niso, M.; Abate, C.; Proschak, E.; Dubiel, M.; Stark, H.; Castro, M.; Lacivita, E.; Leopoldo, M. |