LACIVITA, ENZA

LACIVITA, ENZA  

DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO  

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11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors 1-gen-2005 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
3-(1H-indol-3-yl)-2-[3-(4-nitrophenyl)ureido]propanamide enantiomers with human formyl-peptide receptor agonist activity: Molecular modeling of chiral recognition by FPR2. 1-gen-2013 Schepetkin, Ia; Kirpotina, Ln; Khlebnikov, Ai; Leopoldo, Marcello; Lucente, E; Lacivita, Enza; De Giorgio, P; Quinn, M. T.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization 1-gen-2007 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
5 HT1A receptor, an old target for new therapeutic agents 1-gen-2008 Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Perrone, R.
5-HT7 receptor activation: procognitive and antiamnesic effects 1-gen-2015 Meneses, A; Perez Garcia, G; Liy Salmeron, G; Ponce López, T; Lacivita, Enza; Leopoldo, Marcello
5-HT7 receptor modulators: a medicinal chemistry survey of recent patent literature (2004 - 2009) 1-gen-2010 Leopoldo, Marcello; Lacivita, Enza; Berardi, Francesco; Perrone, Roberto
5-HT7 Receptors Regulate Excitatory-Inhibitory Balance in Mouse Spinal Cord Dorsal Horn 1-gen-2022 Comitato, Antonella; Lacivita, Enza; Leopoldo, Marcello; Bardoni, Rita
Activatable fluorescent probes: a new concept in optical molecular imaging 1-gen-2012 Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Perrone, R.
Activation of 5-HT7 receptor by administration of its selective agonist, LP-211, modifies explorative-curiosity behavior in rats in two paradigms which differ in visuospatial parameters 1-gen-2018 Carbone, Cristiana; Adinolfi, Annalisa; Cinque, Stefano; Lacivita, Enza; Alleva, Enrico; Leopoldo, Marcello; Adriani, Walter
Activation of 5-HT7 receptor stimulates neurite elongation through mTOR, Cdc42 and actin filaments dynamics. 1-gen-2015 Speranza, L; Giuliano, T; Volpicelli, F; De Stefano, Me; Lombardi, L; Chambery, A; Lacivita, Enza; Leopoldo, Marcello; Bellenchi, Gc; di Porzio, U; Crispino, M; Perrone Capano, C.
Activation of 5-HT7 serotonin receptors reverses metabotropic glutamate receptor-mediated synaptic plasticity in wild-type and Fmr1 knockout mice, a model of Fragile X Syndrome 1-gen-2012 Costa, L; Spatuzza, M; D'Antoni, S; Bonaccorso, Cm; Trovato, C; Musumeci, Sa; Leopoldo, Marcello; Lacivita, Enza; Catania, Mv; Ciranna, L.
Activation of Serotonin 5-HT7 Receptors Modulates Hippocampal Synaptic Plasticity by Stimulation of Adenylate Cyclases and Rescues Learning and Behavior in a Mouse Model of Fragile X Syndrome 1-gen-2018 Costa, Lara; Sardone, Lara Maria; Bonaccorso, Carmela Maria; D’Antoni, Simona; Spatuzza, Michela; Gulisano, Walter; Tropea, Maria Rosaria; Puzzo, Daniela; Leopoldo, Marcello; Lacivita, Enza; Catania, Maria Vincenza; Ciranna, Lucia
Analogues of σ Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers 1-gen-2011 Abate, CARMEN rosa; Niso, Mauro; Lacivita, Enza; Mosier, P. D.; Toscano, A.; Perrone, Roberto
Arylpiperazine agonists of the serotonin 5-HT1A receptor preferentially activate cAMP signaling versus recruitment of β-arrestin-2 1-gen-2015 Stroth, Nikolas; Niso, Mauro; Colabufo, Nicola Antonio; Perrone, Roberto; Svenningsson, Per; Lacivita, Enza; Leopoldo, Marcello
Aurantiamide-related dipeptide derivatives are formyl peptide receptor 1 antagonists 1-gen-2019 Mastromarino, Margherita; Kirpotina, Liliya N.; Schepetkin, Igor A.; Quinn, Mark T.; Lacivita, Enza; Leopoldo, Marcello
Behavioral, Anti-Inflammatory, and Neuroprotective Effects of a Novel FPR2 Agonist in Two Mouse Models of Autism 1-gen-2022 Cristiano, C.; Volpicelli, F.; Crispino, M.; Lacivita, E.; Russo, R.; Leopoldo, M.; Calignano, A.; Perrone-Capano, C.
BEHAVIOURAL EFFECTS OF TWO NOVEL AGONISTS FOR SEROTONIN RECEPTOR 7 IN MICE 1-gen-2011 Adriani, W; Travaglini, D; Lacivita, Enza; Leopoldo, Marcello; Laviola, G.
Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: Synthesis and binding affinities for 5-HT7 and 5-HT1A receptors 1-gen-2007 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Design and Synthesis of Arylpiperazine Serotonergic/ Dopaminergic Ligands with Neuroprotective Properties 1-gen-2022 Mastromarino, M.; Niso, M.; Abate, C.; Proschak, E.; Dubiel, M.; Stark, H.; Castro, M.; Lacivita, E.; Leopoldo, M.
Design and synthesis of arylpiperazine-based fluorescent ligands for serotonin 5-HT1A and dopamine D3 receptors. 1-gen-2007 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.