CAROTTI, Angelo
CAROTTI, Angelo
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
"One-step" Synthesis of an Indeno-Indolizine Nucleus
1985-01-01 Carotti, Angelo; Casini, G.; Gavuzzo, E.; Mazza, F.
(EN) GALLOYL BENZAMIDE-BASED COMPOUNDS AS JNK MODULATORS (FR) COMPOSES A BASE DE GALLOYL BENZAMIDE UTILISES EN TANT QUE MODULATEURS DE JNK
2014-01-01 Cellamare, Saverio; Carotti, Angelo; Stefanachi, Angela; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Tardia, Piero; Introcaso, Antonellina; Valentina, Leo; Addabbo, Francesco; Montagnani, Monica; Nacci, Carmela
1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships
2008-01-01 Stefanachi, Angela; Nicolotti, Orazio; Leonetti, Francesco; Cellamare, Saverio; Campagna, Francesco; Loza, Mi; Brea, Jm; Mazza, F; Gavuzzo, E; Carotti, Angelo
1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships
2009-01-01 Fernandez, F; Caamano, O; Nieto, Mi; Lopez, C; Garcia Mera, X; Stefanachi, Angela; Nicolotti, Orazio; Loza, Mi; Brea, J; Esteve, C; Segarra, V; Vidal, B; Carotti, Angelo
17β-Hydroxysteroid Dehydrogenase Type 2 Inhibition: Discovery of Selective and Metabolically Stable Compounds Inhibiting both the Human Enzyme and its Murine Ortholog
2015-01-01 Gargano, Emanuele; Allegretta, Giuseppe; Perspicace, Enrico; Carotti, Angelo; Van Koppen, Chris; Frotscher, Martin; Marchais Oberwinkler, Sandrine; Hartmann, Rolf
2-(2-Phenylcyclopropyl)-Imidazolines: Reversed Enantioselective Interaction At I1 and I2 Imidazoline Receptors
1999-01-01 Quaglia, W.; Bousquet, P.; Pigini, M.; Carotti, Angelo; Carrieri, Antonio; Dontemwill, M.; Gentili, F.; Giannella, M.; Piergentili, A.; Brasili, L.
2-Aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones: novel rigid planar benzodiazepine receptor ligands
1993-01-01 Campagna, F; Carotti, Angelo; Casini, G; Palluotto, F; Genchi, G; De Sarro, G. B.
2-D and 3-D modeling of imadazoline receptor ligands: insights into pharmacophore
1997-01-01 Carrieri, Antonio; L., Brasili; Leonetti, Francesco; M., Pigini; M., Giannella; P., Bousquet; Carotti, Angelo
3,4-Dihydroquinazoline derivatives as T-type Ca2+ channel blockers inhibit the activities of cholinesterase enzymes
2017-01-01 Park, B; Nam, Jh; Kim, Jh; Kim, Hj; Onnis, V; Balboni, G; Lee, Kt; Jeong Ho Park, Jh; Catto, Marco; Carotti, Angelo; Lee, Jy
6-Substituted-(E)-2-(benzofuran-3(2H)-ylidene)-N-methylacetamides as novel, potent and selective MAO inhibitors
2011-01-01 Barletta, M.; Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Soto Otero, R.; Carotti, Angelo
8-Aminomethyl-7-hydroxy-4-methylcoumarins as Multitarget Leads for Alzheimer's Disease
2016-01-01 Dominguez, J. L.; Fernandez-Nieto, F.; Brea, J. M.; Catto, M.; Paleo, M. R.; Porto, S.; Sardina, F. J.; Castro, M.; Pisani, L.; Carotti, A.; Soto-Otero, R.; Mendez-Alvarez, E.; Villaverde, M. C.; Sussman, F.
8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B
2004-01-01 Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio
9,10-Anthraquinone hinders beta-aggregation: how does a small molecule interfere with Abeta-peptide amyloid fibrillation?
2009-01-01 Convertino, M; Pellarin, R; Catto, Marco; Carotti, Angelo; Caflisch, A.
A chemocentric approach to the identification of cancer targets
2012-01-01 Flachner, B; Lorincz, Z; Carotti, Angelo; Nicolotti, Orazio; Kuchipudi, P; Remez, N; Sanz, F; Tovari, J; Szabo, Mj; Bertok, B; Cseh, S; Mestres, J; Dorman, G.
A convenient synthesis of nitriles from primary amides under mild conditions
1977-01-01 Campagna, F; Carotti, Angelo; Casini, G.
A k-NN algorithm for predicting oral sub-chronic toxicity in the rat
2014-01-01 Gadaleta, Domenico; Pizzo, Fabiola; Lombardo, Anna; Carotti, Angelo; Escher, Sylvia E.; Nicolotti, Orazio; Benfenati, Emilio
A natural prothrombin mutant reveals an unexpected influence of the A-chain’s structure on the activity of human alpha-thrombin
2004-01-01 DE CRISTOFARO, R.; Akhavan, S.; Altomare, Cosimo Damiano; Carotti, Angelo; Peyvandi, F.; Mannucci, P. M.
A Round Trip from Medicinal Chemistry to Predictive Toxicology
2016-01-01 Mangiatordi, Giuseppe Felice; Carotti, Angelo; Novellino, Ettore; Nicolotti, Orazio
A simple and Mild Procedure for the Preparation of Bile Acid Methyl Esters
1983-01-01 Ballini, R.; Carotti, Angelo
A simple Synthesis of Heterocyclic Ring Systems Containing the 1,3-oxazine Nucleus
1984-01-01 Altomare, Cosimo Damiano; Carotti, Angelo; Casini, G.; Ferappi, M.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| "One-step" Synthesis of an Indeno-Indolizine Nucleus | 1-gen-1985 | Carotti, Angelo; Casini, G.; Gavuzzo, E.; Mazza, F. | |
| (EN) GALLOYL BENZAMIDE-BASED COMPOUNDS AS JNK MODULATORS (FR) COMPOSES A BASE DE GALLOYL BENZAMIDE UTILISES EN TANT QUE MODULATEURS DE JNK | 1-gen-2014 | Cellamare, Saverio; Carotti, Angelo; Stefanachi, Angela; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Tardia, Piero; Introcaso, Antonellina; Valentina, Leo; Addabbo, Francesco; Montagnani, Monica; Nacci, Carmela | |
| 1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships | 1-gen-2008 | Stefanachi, Angela; Nicolotti, Orazio; Leonetti, Francesco; Cellamare, Saverio; Campagna, Francesco; Loza, Mi; Brea, Jm; Mazza, F; Gavuzzo, E; Carotti, Angelo | |
| 1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships | 1-gen-2009 | Fernandez, F; Caamano, O; Nieto, Mi; Lopez, C; Garcia Mera, X; Stefanachi, Angela; Nicolotti, Orazio; Loza, Mi; Brea, J; Esteve, C; Segarra, V; Vidal, B; Carotti, Angelo | |
| 17β-Hydroxysteroid Dehydrogenase Type 2 Inhibition: Discovery of Selective and Metabolically Stable Compounds Inhibiting both the Human Enzyme and its Murine Ortholog | 1-gen-2015 | Gargano, Emanuele; Allegretta, Giuseppe; Perspicace, Enrico; Carotti, Angelo; Van Koppen, Chris; Frotscher, Martin; Marchais Oberwinkler, Sandrine; Hartmann, Rolf | |
| 2-(2-Phenylcyclopropyl)-Imidazolines: Reversed Enantioselective Interaction At I1 and I2 Imidazoline Receptors | 1-gen-1999 | Quaglia, W.; Bousquet, P.; Pigini, M.; Carotti, Angelo; Carrieri, Antonio; Dontemwill, M.; Gentili, F.; Giannella, M.; Piergentili, A.; Brasili, L. | |
| 2-Aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones: novel rigid planar benzodiazepine receptor ligands | 1-gen-1993 | Campagna, F; Carotti, Angelo; Casini, G; Palluotto, F; Genchi, G; De Sarro, G. B. | |
| 2-D and 3-D modeling of imadazoline receptor ligands: insights into pharmacophore | 1-gen-1997 | Carrieri, Antonio; L., Brasili; Leonetti, Francesco; M., Pigini; M., Giannella; P., Bousquet; Carotti, Angelo | |
| 3,4-Dihydroquinazoline derivatives as T-type Ca2+ channel blockers inhibit the activities of cholinesterase enzymes | 1-gen-2017 | Park, B; Nam, Jh; Kim, Jh; Kim, Hj; Onnis, V; Balboni, G; Lee, Kt; Jeong Ho Park, Jh; Catto, Marco; Carotti, Angelo; Lee, Jy | |
| 6-Substituted-(E)-2-(benzofuran-3(2H)-ylidene)-N-methylacetamides as novel, potent and selective MAO inhibitors | 1-gen-2011 | Barletta, M.; Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Soto Otero, R.; Carotti, Angelo | |
| 8-Aminomethyl-7-hydroxy-4-methylcoumarins as Multitarget Leads for Alzheimer's Disease | 1-gen-2016 | Dominguez, J. L.; Fernandez-Nieto, F.; Brea, J. M.; Catto, M.; Paleo, M. R.; Porto, S.; Sardina, F. J.; Castro, M.; Pisani, L.; Carotti, A.; Soto-Otero, R.; Mendez-Alvarez, E.; Villaverde, M. C.; Sussman, F. | |
| 8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B | 1-gen-2004 | Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio | |
| 9,10-Anthraquinone hinders beta-aggregation: how does a small molecule interfere with Abeta-peptide amyloid fibrillation? | 1-gen-2009 | Convertino, M; Pellarin, R; Catto, Marco; Carotti, Angelo; Caflisch, A. | |
| A chemocentric approach to the identification of cancer targets | 1-gen-2012 | Flachner, B; Lorincz, Z; Carotti, Angelo; Nicolotti, Orazio; Kuchipudi, P; Remez, N; Sanz, F; Tovari, J; Szabo, Mj; Bertok, B; Cseh, S; Mestres, J; Dorman, G. | |
| A convenient synthesis of nitriles from primary amides under mild conditions | 1-gen-1977 | Campagna, F; Carotti, Angelo; Casini, G. | |
| A k-NN algorithm for predicting oral sub-chronic toxicity in the rat | 1-gen-2014 | Gadaleta, Domenico; Pizzo, Fabiola; Lombardo, Anna; Carotti, Angelo; Escher, Sylvia E.; Nicolotti, Orazio; Benfenati, Emilio | |
| A natural prothrombin mutant reveals an unexpected influence of the A-chain’s structure on the activity of human alpha-thrombin | 1-gen-2004 | DE CRISTOFARO, R.; Akhavan, S.; Altomare, Cosimo Damiano; Carotti, Angelo; Peyvandi, F.; Mannucci, P. M. | |
| A Round Trip from Medicinal Chemistry to Predictive Toxicology | 1-gen-2016 | Mangiatordi, Giuseppe Felice; Carotti, Angelo; Novellino, Ettore; Nicolotti, Orazio | |
| A simple and Mild Procedure for the Preparation of Bile Acid Methyl Esters | 1-gen-1983 | Ballini, R.; Carotti, Angelo | |
| A simple Synthesis of Heterocyclic Ring Systems Containing the 1,3-oxazine Nucleus | 1-gen-1984 | Altomare, Cosimo Damiano; Carotti, Angelo; Casini, G.; Ferappi, M. |