LAVECCHIA, ANTONIO
LAVECCHIA, ANTONIO
A Chemical Modification of a Peroxisome Proliferator-Activated Receptor Pan Agonist Produced a Shift to a New Dual Alpha/Gamma Partial Agonist Endowed with Mitochondrial Pyruvate Carrier Inhibition and Antidiabetic Properties
2024-01-01 Laghezza, Antonio; Cerchia, Carmen; Genovese, Massimo; Montanari, Roberta; Capelli, Davide; Wackerlig, Judith; Simic, Stefan; Falbo, Emanuele; Pecora, Lucia; Leuci, Rosalba; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Biswas, Abanish; Singh, Ravi Pratap; Tambe, Suhas; Sudeep, C. A.; Pattnaik, Ashok Kumar; Jayaprakash, Venkatesan; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio
Discovery of a dual PPARα/γ partial agonist displaying antisteatotic and antidiabetic properties: in silico studies and X-ray structure determination
2024-01-01 Cerchia, Carmen; Laghezza, Antonio; Brunetti, Leonardo; Falbo, Emanuele; Tortorella, Paolo; Piemontese, Luca; Montanari, Roberta; Paoli, Paolo; Jayaprakash, Venkatesan; Loiodice, Fulvio; Lavecchia, Antonio
Sulfonimide and Amide Derivatives as Novel PPARα Antagonists: Synthesis, Antiproliferative Activity, and Docking Studies.
2020-01-01 Ammazzalorso, Alessandra; Bruno, Isabella; Florio, Rosalba; De Lellis, Laura; Laghezza, Antonio; Cerchia, Carmen; De Filippis, Barbara; Fantacuzzi, Marialuigia; Giampietro, Letizia; Maccallini, Cristina; Tortorella, Paolo; Veschi, Serena; Loiodice, Fulvio; Lavecchia, Antonio; Cama, Alessandro; Amoroso, Rosa
Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents
2020-01-01 Tilekar, Kalpana; Upadhyay, Neha; Meyer‐almes, Franz‐josef; Loiodice, Fulvio; Anisimova, Natalia Y.; Spirina, Tatiana S.; Sokolova, Darina V.; Smirnova, Galina B.; Choe, Jun‐yong; Pokrovsky, Vadim S.; Lavecchia, Antonio; Ramaa, C. S.
Synthesis and in vitro cytotoxicity of benzoxazole‐based PPARα/γ antagonists in colorectal cancer cell lines
2024-01-01 Moreno‐rodríguez, Nazaret; Laghezza, Antonio; Cerchia, Carmen; Sokolova, Darina V.; Spirina, Tatiana S.; De Filippis, Barbara; Romanelli, Virgilio; Recio, Rocío; Fernández, Inmaculada; Loiodice, Fulvio; Pokrovsky, Vadim S.; Ammazzalorso, Alessandra; Lavecchia, Antonio
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A Chemical Modification of a Peroxisome Proliferator-Activated Receptor Pan Agonist Produced a Shift to a New Dual Alpha/Gamma Partial Agonist Endowed with Mitochondrial Pyruvate Carrier Inhibition and Antidiabetic Properties | 1-gen-2024 | Laghezza, Antonio; Cerchia, Carmen; Genovese, Massimo; Montanari, Roberta; Capelli, Davide; Wackerlig, Judith; Simic, Stefan; Falbo, Emanuele; Pecora, Lucia; Leuci, Rosalba; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Biswas, Abanish; Singh, Ravi Pratap; Tambe, Suhas; Sudeep, C. A.; Pattnaik, Ashok Kumar; Jayaprakash, Venkatesan; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio | |
| Discovery of a dual PPARα/γ partial agonist displaying antisteatotic and antidiabetic properties: in silico studies and X-ray structure determination | 1-gen-2024 | Cerchia, Carmen; Laghezza, Antonio; Brunetti, Leonardo; Falbo, Emanuele; Tortorella, Paolo; Piemontese, Luca; Montanari, Roberta; Paoli, Paolo; Jayaprakash, Venkatesan; Loiodice, Fulvio; Lavecchia, Antonio | |
| Sulfonimide and Amide Derivatives as Novel PPARα Antagonists: Synthesis, Antiproliferative Activity, and Docking Studies. | 1-gen-2020 | Ammazzalorso, Alessandra; Bruno, Isabella; Florio, Rosalba; De Lellis, Laura; Laghezza, Antonio; Cerchia, Carmen; De Filippis, Barbara; Fantacuzzi, Marialuigia; Giampietro, Letizia; Maccallini, Cristina; Tortorella, Paolo; Veschi, Serena; Loiodice, Fulvio; Lavecchia, Antonio; Cama, Alessandro; Amoroso, Rosa | |
| Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents | 1-gen-2020 | Tilekar, Kalpana; Upadhyay, Neha; Meyer‐almes, Franz‐josef; Loiodice, Fulvio; Anisimova, Natalia Y.; Spirina, Tatiana S.; Sokolova, Darina V.; Smirnova, Galina B.; Choe, Jun‐yong; Pokrovsky, Vadim S.; Lavecchia, Antonio; Ramaa, C. S. | |
| Synthesis and in vitro cytotoxicity of benzoxazole‐based PPARα/γ antagonists in colorectal cancer cell lines | 1-gen-2024 | Moreno‐rodríguez, Nazaret; Laghezza, Antonio; Cerchia, Carmen; Sokolova, Darina V.; Spirina, Tatiana S.; De Filippis, Barbara; Romanelli, Virgilio; Recio, Rocío; Fernández, Inmaculada; Loiodice, Fulvio; Pokrovsky, Vadim S.; Ammazzalorso, Alessandra; Lavecchia, Antonio |