CAMPAGNA, Francesco

CAMPAGNA, Francesco  

DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO  

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Titolo Data di pubblicazione Autore(i) File
1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships 1-gen-2008 Stefanachi, Angela; Nicolotti, Orazio; Leonetti, Francesco; Cellamare, Saverio; Campagna, Francesco; Loza, Mi; Brea, Jm; Mazza, F; Gavuzzo, E; Carotti, Angelo
4-(ALKYL)AMINOMETHYL-SUBSTITUTED COUMARINS AS POTENT AND SELECTIVE ACHE AND MAO-B DUAL INHIBITORS WITH A THERAPEUTIC POTENTIAL IN NEURODEGENERATIVE DISORDERS 1-gen-2013 Pisani, Leonardo; Catto, Marco; Stefanachi, Angela; Leonetti, F; Campagna, Francesco; Nicolotti, O; SOTO OTERO, R; Carotti, A.
Benzodiazepine receptor affinities, behavioural and anticonvulsant activity of 2-aryl-2,5-dihydropyridazino[4,3-b]indol-3(3H)-ones in mice 1-gen-2000 DE SARRO, G.; Carotti, Angelo; Campagna, Francesco; Palluotto, Fausta; Mckernan, R.; Quirk, K.; Rizzo, M.; Giusti, P.; Rettore, C.; DE SARRO, A.
Biophysical Characterization of Inhibition of A-beta Fibril Formation by Isatin-3-arylhydrazones 1-gen-2010 Campagna, Francesco; Purgatorio, R; Catto, Marco; Carotti, A; De, Stradisa; Palazzo, Gerardo
Design, synthesis and biological evaluation of benzo[e][1,2,4]triazin-7(1H)-one and [1,2,4]-triazino[5,6,1-jk]carbazol-6-one derivatives as dual inhibitors of beta-amyloid aggregation and acetyl/butyryl cholinesterases 1-gen-2012 Catto, Marco; Berezin, A. A.; Lo Re, D; Loizou, G; Demetriades, M; De Stradis, A; Campagna, Francesco; Koutentis, P. A.; Carotti, Angelo
Design, synthesis and biological evaluation of indane 2-arylhydrazinylmethylene-1,3-diones and indol-2-aryldiazenylmethylene-3-ones as b-amyloid aggregation inhibitors 1-gen-2010 Catto, Marco; Aliano, R; Carotti, Angelo; Cellamare, Saverio; Palluotto, Fausta; Purgatorio, R; DE STRADIS, A; Campagna, Francesco
Design, synthesis, and biological evaluation of glycine-based molecular tongs as inhibitors of Aβ40 aggregation in vitro 1-gen-2008 Cellamare, Saverio; Stefanachi, Angela; Stolfa, D. A.; Basile, T; Catto, Marco; Campagna, Francesco; Sotelo, E; Acquafredda, Pasquale; Carotti, Angelo
Indol-3-ylidene, pyridazino[4,3-b]indole and indeno[1,2-c]pyrazole derivatives:synthesis and biological evaluation as inhibitors of GSK-3 and CDKs 1-gen-2005 Campagna, Francesco; Aliano, R; Carotti, A; Palluotto, Fausta; Lozach, O; Meijer, L.
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications 1-gen-2007 Campagna, Francesco; Cellamare, Saverio; Stefanachi, Angela; Stolfa, D. A.; Basile, T; Ferappi, M; Catto, Marco; Carotti, A.
Insights into Structure-Activity Relationships of 3-Arylhydrazonoindolin-2-One Derivatives for Their Multitarget Activity on β-Amyloid Aggregation and Neurotoxicity 1-gen-2018 Purgatorio, Rosa; de Candia, M; De Palma, A; DE SANTIS, Francesco; Pisani, L; Campagna, F; Cellamare, S; Altomare, Cd; Catto, M
Investigation on the influence of (Z)-3-(2-(3-chlorophenyl)hydrazono)-5,6-dihydroxyindolin-2-one (PT2) on β-amyloid(1-40) aggregation and toxicity 1-gen-2014 Catto, Marco; Arnesano, Fabio; Palazzo, Gerardo; De Stradis, A; Calò, V; Losacco, M; Purgatorio, R; Campagna, Francesco
Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: a water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity 1-gen-2017 Pisani, Leonardo; DE PALMA, Annalisa; Giangregorio, Nicola; Miniero, DANIELA VALERIA; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo Damiano; Catto, Marco
New N-arylmethyl derivatives of some cyclic amino acids and new peptidomimetics: synthesis and inhibition activity of insulin amyloid formation 1-gen-2005 Campagna, Francesco; Cellamare, Saverio; Aliano, R; Carotti, A; Ferappi, M.
NOVEL GLUCOSE-CONJUGATED HIGHLY POTENT DUAL THROMBIN AND FACTOR Xa INHIBITORS AS POTENTIAL ANTITHROMBOTICS 1-gen-2013 Zaetta, G; DE CANDIA, Modesto; Campagna, Francesco; Belviso, B. D.; Caliandro, R; Incampo, F; Carrieri, C; Colucci, M; Altomare, Cosimo Damiano
Synthesis and antibacterial activity of 2-aryl-2,5-dihydro-3(3H)-oxo-pyridazino4,3-bindole-4-carboxylic acids 1-gen-1999 Palluotto, Fausta; Carotti, Angelo; Casini, G.; Ferappi, M; Rosato, Antonio; Vitali, C.; Campagna, Francesco
Synthesis and antibacterial activity of pyridazino[4,3-b]indole-4-carboxylic acids carrying different substituents at N-2 1-gen-2002 Palluotto, Fausta; Campagna, Francesco; Carotti, Angelo; Ferappi, M.; Rosato, Antonio; Vitali, C.
Synthesis and biological evaluation of arylhydrazone derivatives of indoles and indolin-2-ones as b-amyloid aggregation inhibitors 1-gen-2009 Campagna, Francesco; Catto, Marco; Carotti, A; Cellamare, Saverio; Palluotto, Fausta; Purgatorio, R.
Synthesis and biological evaluation of arylhydrazone derivatives of indoles and indolin-2-ones as b-amyloid aggregation inhibitors 1-gen-2009 Campagna, F; Catto, M; Carotti, A; Cellamare, S; Palluotto, F; Purgatorio, R
Synthesis and biological evaluation of pyrazoles and pyrazole-containing polycyclic derivatives as new ligands of central and peripheral benzodiazepine receptors 1-gen-2004 Campagna, Francesco; Palluotto, F.; Carotti, Angelo; Maciocco, E.
Synthesis and biophysical evaluation of arylhydrazono-1H-2-indolinones as beta-amyloid aggregation inhibitors 1-gen-2011 Campagna, Francesco; Catto, Marco; Purgatorio, R; Altomare, Cosimo Damiano; Carotti, Angelo; DE STRADIS, A; Palazzo, Gerardo