Sfoglia per Autore
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitors
2018-01-01 Mangiatordi, G. F.; Trisciuzzi, D.; Iacobazzi, R.; Denora, N.; Pisani, L.; Catto, M.; Leonetti, F.; Alberga, D.; Nicolotti, O.
Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT 1A receptor agonists for CNS disorders and neuropathic pain
2018-01-01 Franchini, S.; Bencheva, L. I.; Battisti, U. M.; Tait, A.; Sorbi, C.; Fossa, P.; Cichero, E.; Ronsisvalle, S.; Arico, G.; Denora, N.; Iacobazzi, R. M.; Cilia, A.; Pirona, L.; Brasili, L.
NEW HORIZONS IN TREATMENTS OF METASTATIC MELANOMA: THE ROLE OF TOMATINE
2018-01-01 Guida, Stefania; Ferretta, Anna; Serratì, Simona; Cocco, Tiziana Maria; Maida, Immacolata; Iacobazzi, ROSA MARIA; Porcelli, Letizia; Azzariti, Amalia; Tommasi, Stefania; Tamasi, Gabriella; Rossi, Claudio; Pellacani, Giovanni; Guida, Gabriella
CAFs and TGF-β Signaling Activation by Mast Cells Contribute to Resistance to Gemcitabine/Nabpaclitaxel in Pancreatic Cancer
2019-01-01 Porcelli, Letizia; Iacobazzi, Rosa Maria; Di Fonte, Roberta; Serrati', Simona; Intini, Angelica; Solimando, Antonio Giovanni; Brunetti, Oronzo; Calabrese, Angela; Leonetti, Francesco; Azzariti, Amalia; Silvestris, Nicola
Plasma-activated medium triggers cell death and the presentation of immune activating danger signals in melanoma and pancreatic cancer cells
2019-01-01 Azzariti, Amalia; Iacobazzi, Rosa Maria; Di Fonte, Roberta; Porcelli, Letizia; Gristina, Roberto; Favia, Pietro; Fracassi, Francesco; Trizio, Ilaria; Silvestris, Nicola; Guida, Gabriella; Tommasi, Stefania; Sardella, Eloisa
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity
2019-01-01 Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L.
Investigating alkyl nitrates as nitric oxide releasing precursors of multitarget acetylcholinesterase-monoamine oxidase B inhibitors
2019-01-01 Pisani, Leonardo; Iacobazzi, Rosa Maria; Catto, Marco; Rullo, Mariagrazia; Farina, Roberta; Denora, Nunzio; Cellamare, Saverio; Altomare, Cosimo Damiano
Gene Expression Comparison between the Lymph Node-Positive and -Negative Reveals a Peculiar Immune Microenvironment Signature and a Theranostic Role for WNT Targeting in Pancreatic Ductal Adenocarcinoma: A Pilot Study
2019-01-01 Argentiero, Antonella; De Summa, Simona; Di Fonte, Roberta; Iacobazzi, Rosa Maria; Porcelli, Letizia; Da Vià, Matteo; Brunetti, Oronzo; Azzariti, Amalia; Silvestris, Nicola; Solimando, Antonio Giovanni
TSPO-targeted NIR-fluorescent ultra-small iron oxide nanoparticles for glioblastoma imaging
2019-01-01 Denora, N.; Lee, C.; Iacobazzi, R. M.; Choi, J. Y.; Song, I. H.; Yoo, J. S.; Piao, Y.; Lopalco, A.; Leonetti, F.; Lee, B. C.; Kim, S. E.
Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
2019-01-01 Oukoloff, Killian; Coquelle, Nicolas; Bartolini, Manuela; Naldi, Marina; Le Guevel, Rémy; Bach, Stéphane; Josselin, Béatrice; Ruchaud, Sandrine; Catto, Marco; Pisani, Leonardo; Denora, Nunzio; Iacobazzi, Rosa Maria; Silman, Israel; Sussman, Joel L.; Buron, Frédéric; Colletier, Jacques-Philippe; Jean, Ludovic; Routier, Sylvain; Renard, Pierre-Yves
Green fluorescent terbium (III) complex doped silica nanoparticles
2019-01-01 Fanizza, E.; Depalo, N.; Fedorenko, S.; Iacobazzi, R. M.; Mukhametshina, A.; Zairov, R.; Salatino, A.; Vischio, F.; Panniello, A.; Laquintana, V.; Lucia Curri, M.; Mustafina, A.; Denora, N.; Striccoli, M.
Induced expression of P-gp and BCRP transporters on brain endothelial cells using transferrin functionalized nanostructured lipid carriers: A first step of a potential strategy for the treatment of Alzheimer's disease
2020-01-01 Arduino, I.; Iacobazzi, R. M.; Riganti, C.; Lopedota, A. A.; Perrone, M. G.; Lopalco, A.; Cutrignelli, A.; Cantore, M.; Laquintana, V.; Franco, M.; Colabufo, N. A.; Luurtsema, G.; Contino, M.; Denora, N.
Tomatine displays antitumor potential in in vitro models of metastatic melanoma
2020-01-01 Serrati, S.; Porcelli, L.; Guida, S.; Ferretta, A.; Iacobazzi, R. M.; Cocco, T.; Maida, I.; Tamasi, G.; Rossi, C.; Manganelli, M.; Tommasi, S.; Azzariti, A.; Guida, G.
Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents
2020-01-01 Franchini, S.; Linciano, P.; Puja, G.; Tait, A.; Borsari, C.; Denora, N.; Iacobazzi, R. M.; Brasili, L.; Sorbi, C.
Reproducibility warning: The curious case of polyethylene glycol 6000 and spheroid cell culture
2020-01-01 Serrati, S.; Martinelli, C.; Palazzo, A.; Iacobazzi, R. M.; Perrone, M.; Ong, Q. K.; Luo, Z.; Bekdemir, A.; Pinto, G.; Cavalleri, O.; Cutrignelli, A.; Laquintana, V.; Denora, N.; Stellacci, F.; Krol, S.
Hydroxy-propil-β-cyclodextrin inclusion complexes of two biphenylnicotinamide derivatives: Formulation and anti-proliferative activity evaluation in pancreatic cancer cell models
2020-01-01 Iacobazzi, R. M.; Cutrignelli, A.; Stefanachi, A.; Porcelli, L.; Lopedota, A. A.; Di Fonte, R.; Lopalco, A.; Serrati, S.; Laquintana, V.; Silvestris, N.; Franco, M.; Cellamare, S.; Leonetti, F.; Azzariti, A.; Denora, N.
Gold-Speckled SPION@SiO2 Nanoparticles Decorated with Thiocarbohydrates for ASGPR1 Targeting: Towards HCC Dual Mode Imaging Potential Applications
2020-01-01 Siciliano, G.; Corricelli, M.; Iacobazzi, R. M.; Canepa, F.; Comegna, D.; Fanizza, E.; Del Gatto, A.; Saviano, M.; Laquintana, V.; Comparelli, R.; Mascolo, G.; Murgolo, S.; Striccoli, M.; Agostiano, A.; Denora, N.; Zaccaro, L.; Curri, M. L.; Depalo, N.
New Oxaliplatin-Pyrophosphato Analogs with Improved In Vitro Cytotoxicity
2021-01-01 Barbanente, Alessandra; Maria Iacobazzi, Rosa; Azzariti, Amalia; Hoeschele, James D.; Denora, Nunzio; Papadia, Paride; Pacifico, Concetta; Natile, Giovanni; Margiotta, Nicola
Bortezomib Aqueous Solubility in the Presence and Absence of D-Mannitol: A Clarification With Formulation Implications
2021-01-01 Lopalco, A.; Iacobazzi, R. M.; Denora, N.; Stella, V. J.
From oil to microparticulate by prilling technique: Production of polynucleate alginate beads loading Serenoa Repens oil as intestinal delivery systems
2021-01-01 Lopedota, A. A.; Arduino, I.; Lopalco, A.; Iacobazzi, R. M.; Cutrignelli, A.; Laquintana, V.; Racaniello, G. F.; Franco, M.; la Forgia, F.; Fontana, S.; Denora, N.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitors | 1-gen-2018 | Mangiatordi, G. F.; Trisciuzzi, D.; Iacobazzi, R.; Denora, N.; Pisani, L.; Catto, M.; Leonetti, F.; Alberga, D.; Nicolotti, O. | |
Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT 1A receptor agonists for CNS disorders and neuropathic pain | 1-gen-2018 | Franchini, S.; Bencheva, L. I.; Battisti, U. M.; Tait, A.; Sorbi, C.; Fossa, P.; Cichero, E.; Ronsisvalle, S.; Arico, G.; Denora, N.; Iacobazzi, R. M.; Cilia, A.; Pirona, L.; Brasili, L. | |
NEW HORIZONS IN TREATMENTS OF METASTATIC MELANOMA: THE ROLE OF TOMATINE | 1-gen-2018 | Guida, Stefania; Ferretta, Anna; Serratì, Simona; Cocco, Tiziana Maria; Maida, Immacolata; Iacobazzi, ROSA MARIA; Porcelli, Letizia; Azzariti, Amalia; Tommasi, Stefania; Tamasi, Gabriella; Rossi, Claudio; Pellacani, Giovanni; Guida, Gabriella | |
CAFs and TGF-β Signaling Activation by Mast Cells Contribute to Resistance to Gemcitabine/Nabpaclitaxel in Pancreatic Cancer | 1-gen-2019 | Porcelli, Letizia; Iacobazzi, Rosa Maria; Di Fonte, Roberta; Serrati', Simona; Intini, Angelica; Solimando, Antonio Giovanni; Brunetti, Oronzo; Calabrese, Angela; Leonetti, Francesco; Azzariti, Amalia; Silvestris, Nicola | |
Plasma-activated medium triggers cell death and the presentation of immune activating danger signals in melanoma and pancreatic cancer cells | 1-gen-2019 | Azzariti, Amalia; Iacobazzi, Rosa Maria; Di Fonte, Roberta; Porcelli, Letizia; Gristina, Roberto; Favia, Pietro; Fracassi, Francesco; Trizio, Ilaria; Silvestris, Nicola; Guida, Gabriella; Tommasi, Stefania; Sardella, Eloisa | |
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity | 1-gen-2019 | Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L. | |
Investigating alkyl nitrates as nitric oxide releasing precursors of multitarget acetylcholinesterase-monoamine oxidase B inhibitors | 1-gen-2019 | Pisani, Leonardo; Iacobazzi, Rosa Maria; Catto, Marco; Rullo, Mariagrazia; Farina, Roberta; Denora, Nunzio; Cellamare, Saverio; Altomare, Cosimo Damiano | |
Gene Expression Comparison between the Lymph Node-Positive and -Negative Reveals a Peculiar Immune Microenvironment Signature and a Theranostic Role for WNT Targeting in Pancreatic Ductal Adenocarcinoma: A Pilot Study | 1-gen-2019 | Argentiero, Antonella; De Summa, Simona; Di Fonte, Roberta; Iacobazzi, Rosa Maria; Porcelli, Letizia; Da Vià, Matteo; Brunetti, Oronzo; Azzariti, Amalia; Silvestris, Nicola; Solimando, Antonio Giovanni | |
TSPO-targeted NIR-fluorescent ultra-small iron oxide nanoparticles for glioblastoma imaging | 1-gen-2019 | Denora, N.; Lee, C.; Iacobazzi, R. M.; Choi, J. Y.; Song, I. H.; Yoo, J. S.; Piao, Y.; Lopalco, A.; Leonetti, F.; Lee, B. C.; Kim, S. E. | |
Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3 | 1-gen-2019 | Oukoloff, Killian; Coquelle, Nicolas; Bartolini, Manuela; Naldi, Marina; Le Guevel, Rémy; Bach, Stéphane; Josselin, Béatrice; Ruchaud, Sandrine; Catto, Marco; Pisani, Leonardo; Denora, Nunzio; Iacobazzi, Rosa Maria; Silman, Israel; Sussman, Joel L.; Buron, Frédéric; Colletier, Jacques-Philippe; Jean, Ludovic; Routier, Sylvain; Renard, Pierre-Yves | |
Green fluorescent terbium (III) complex doped silica nanoparticles | 1-gen-2019 | Fanizza, E.; Depalo, N.; Fedorenko, S.; Iacobazzi, R. M.; Mukhametshina, A.; Zairov, R.; Salatino, A.; Vischio, F.; Panniello, A.; Laquintana, V.; Lucia Curri, M.; Mustafina, A.; Denora, N.; Striccoli, M. | |
Induced expression of P-gp and BCRP transporters on brain endothelial cells using transferrin functionalized nanostructured lipid carriers: A first step of a potential strategy for the treatment of Alzheimer's disease | 1-gen-2020 | Arduino, I.; Iacobazzi, R. M.; Riganti, C.; Lopedota, A. A.; Perrone, M. G.; Lopalco, A.; Cutrignelli, A.; Cantore, M.; Laquintana, V.; Franco, M.; Colabufo, N. A.; Luurtsema, G.; Contino, M.; Denora, N. | |
Tomatine displays antitumor potential in in vitro models of metastatic melanoma | 1-gen-2020 | Serrati, S.; Porcelli, L.; Guida, S.; Ferretta, A.; Iacobazzi, R. M.; Cocco, T.; Maida, I.; Tamasi, G.; Rossi, C.; Manganelli, M.; Tommasi, S.; Azzariti, A.; Guida, G. | |
Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents | 1-gen-2020 | Franchini, S.; Linciano, P.; Puja, G.; Tait, A.; Borsari, C.; Denora, N.; Iacobazzi, R. M.; Brasili, L.; Sorbi, C. | |
Reproducibility warning: The curious case of polyethylene glycol 6000 and spheroid cell culture | 1-gen-2020 | Serrati, S.; Martinelli, C.; Palazzo, A.; Iacobazzi, R. M.; Perrone, M.; Ong, Q. K.; Luo, Z.; Bekdemir, A.; Pinto, G.; Cavalleri, O.; Cutrignelli, A.; Laquintana, V.; Denora, N.; Stellacci, F.; Krol, S. | |
Hydroxy-propil-β-cyclodextrin inclusion complexes of two biphenylnicotinamide derivatives: Formulation and anti-proliferative activity evaluation in pancreatic cancer cell models | 1-gen-2020 | Iacobazzi, R. M.; Cutrignelli, A.; Stefanachi, A.; Porcelli, L.; Lopedota, A. A.; Di Fonte, R.; Lopalco, A.; Serrati, S.; Laquintana, V.; Silvestris, N.; Franco, M.; Cellamare, S.; Leonetti, F.; Azzariti, A.; Denora, N. | |
Gold-Speckled SPION@SiO2 Nanoparticles Decorated with Thiocarbohydrates for ASGPR1 Targeting: Towards HCC Dual Mode Imaging Potential Applications | 1-gen-2020 | Siciliano, G.; Corricelli, M.; Iacobazzi, R. M.; Canepa, F.; Comegna, D.; Fanizza, E.; Del Gatto, A.; Saviano, M.; Laquintana, V.; Comparelli, R.; Mascolo, G.; Murgolo, S.; Striccoli, M.; Agostiano, A.; Denora, N.; Zaccaro, L.; Curri, M. L.; Depalo, N. | |
New Oxaliplatin-Pyrophosphato Analogs with Improved In Vitro Cytotoxicity | 1-gen-2021 | Barbanente, Alessandra; Maria Iacobazzi, Rosa; Azzariti, Amalia; Hoeschele, James D.; Denora, Nunzio; Papadia, Paride; Pacifico, Concetta; Natile, Giovanni; Margiotta, Nicola | |
Bortezomib Aqueous Solubility in the Presence and Absence of D-Mannitol: A Clarification With Formulation Implications | 1-gen-2021 | Lopalco, A.; Iacobazzi, R. M.; Denora, N.; Stella, V. J. | |
From oil to microparticulate by prilling technique: Production of polynucleate alginate beads loading Serenoa Repens oil as intestinal delivery systems | 1-gen-2021 | Lopedota, A. A.; Arduino, I.; Lopalco, A.; Iacobazzi, R. M.; Cutrignelli, A.; Laquintana, V.; Racaniello, G. F.; Franco, M.; la Forgia, F.; Fontana, S.; Denora, N. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile