Sfoglia per Autore
Synthesis, antiarrhythmic activity, and toxicological evaluation of mexiletine analogues
2016-01-01 Roselli, Mariagrazia; Carocci, Alessia; Budriesi, Roberta; Micucci, Matteo; Toma, Maddalena; Di Cesare Mannelli, Lorenzo; Lovece, Angelo; Catalano, Alessia; Cavalluzzi, MARIA MADDALENA; Bruno, Claudio; DE PALMA, Annalisa; Contino, Marialessandra; Perrone, MARIA GRAZIA; Colabufo, Nicola Antonio; Chiarini, Alberto; Franchini, Carlo; Ghelardini, Carla; Habtemariam, Solomon; Lentini, Giovanni
The mitochondrial carnitine/acylcarnitine carrier is regulated by hydrogen sulfide via interaction with C136 and C155
2016-01-01 Giangregorio, Nicola; Tonazzi, Annamaria; Console, Lara; Lorusso, Imma; DE PALMA, Annalisa; Indiveri, Cesare
Nitric oxide inhibits the mitochondrial carnitine/acylcarnitine carrier through reversible S-nitrosylation of cysteine 136
2017-01-01 Tonazzi, Annamaria; Giangregorio, Nicola; Console, Lara; DE PALMA, Annalisa; Indiveri, Cesare
Nitro-substituted tetrahydroindolizines and homologs: Design, kinetics, and mechanism of α-glucosidase inhibition
2017-01-01 Tavani, Cinzia; Bianchi, Lara; DE PALMA, Annalisa; Passeri, GIOVANNA ILARIA; Punzi, Giuseppe; Pierri, CIRO LEONARDO; Lovece, Angelo; Cavalluzzi, MARIA MADDALENA; Franchini, Carlo; Lentini, Giovanni; Petrillo, Giovanni
Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties
2017-01-01 Pisani, Leonardo; Catto, Marco; DE PALMA, Annalisa; Farina, Roberta; Cellamare, Saverio; Altomare, Cosimo Damiano
Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: a water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity
2017-01-01 Pisani, Leonardo; DE PALMA, Annalisa; Giangregorio, Nicola; Miniero, DANIELA VALERIA; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo Damiano; Catto, Marco
Fitocomplesso polifenolico standardizzato per la prevenzione delle patologie correlate all’esposizione da sostanze reattive dell’ossigeno e relativo metodo di produzione
2017-01-01 Cavalluzzi, MARIA MADDALENA; Mallamaci, Rosanna; Clodoveo, MARIA LISA; Moretti, Umberto; Lentini, Giovanni; Franchini, Carlo; Moretti, Pasquale; DE PALMA, Annalisa; Pisano, Isabella; Corbo, Filomena Faustina Rina; MASSARI CLAUDIO, Domenico
Insights into Structure-Activity Relationships of 3-Arylhydrazonoindolin-2-One Derivatives for Their Multitarget Activity on β-Amyloid Aggregation and Neurotoxicity
2018-01-01 Purgatorio, Rosa; de Candia, M; De Palma, A; DE SANTIS, Francesco; Pisani, L; Campagna, F; Cellamare, S; Altomare, Cd; Catto, M
Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease
2019-01-01 Purgatorio, R.; de Candia, M.; Catto, M.; Carrieri, A.; Pisani, L.; De Palma, A.; Toma, M.; Ivanova, O. A.; Voskressensky, L. G.; Altomare, C. D.
Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE Inhibitor
2020-01-01 Catto, Marco; Pisani, Leonardo; de la Mora, Eugenio; Belviso, Benny Danilo; Mangiatordi, Giuseppe Felice; Pinto, Andrea; Palma, Annalisa De; Denora, Nunzio; Caliandro, Rocco; Colletier, Jacques-Philippe; Silman, Israel; Nicolotti, Orazio; Altomare, Cosimo Damiano
Scouting around 1,2,3,4-Tetrahydrochromeno[3,2-c]pyridin-10-ones for Single- and Multitarget Ligands Directed towards Relevant Alzheimer's Targets
2020-01-01 Purgatorio, R.; Kulikova, L. N.; Pisani, L.; Catto, M.; de Candia, M.; Carrieri, A.; Cellamare, S.; De Palma, A.; Beloglazkin, A. A.; Reza Raesi, G.; Voskressensky, L. G.; Altomare, C. D.
The interaction of hemin, a porphyrin derivative, with the purified rat brain 2-oxoglutarate carrier
2021-01-01 Miniero, D. V.; Spagnoletta, A.; Gambacorta, N.; Scalera, V.; Pierri, C. L.; Nicolotti, O.; De Palma, A.
Synthesis and Evaluation of Voltage-Gated Sodium Channel Blocking Pyrroline Derivatives Endowed with Both Antiarrhythmic and Antioxidant Activities
2021-01-01 Carocci, Alessia; Roselli, Mariagrazia; Budriesi, Roberta; Micucci, Matteo; Desaphy, Jean-François; Altamura, Concetta; Cavalluzzi, Maria Maddalena; Toma, Maddalena; Passeri, Giovanna Ilaria; Milani, Gualtiero; Lovece, Angelo; Catalano, Alessia; Bruno, Claudio; De Palma, Annalisa; Corbo, Filomena; Franchini, Carlo; Habtemariam, Solomon; Lentini, Giovanni
Densely Functionalized 2-Methylideneazetidines: Evaluation as Antibacterials
2021-01-01 Petrillo, Giovanni; Tavani, Cinzia; Bianchi, Lara; Benzi, Alice; Cavalluzzi, MARIA MADDALENA; Salvagno, Lara; Quintieri, Laura; DE PALMA, Annalisa; Caputo, Leonardo; Rosato, Antonio; Lentini, Giovanni
New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction
2022-01-01 Miniero, DANIELA VALERIA; Gambacorta, Nicola; Spagnoletta, Anna; Tragni, Vincenzo; Loizzo, Stefano; Nicolotti, Orazio; Pierri, CIRO LEONARDO; DE PALMA, Annalisa
Microwave-Assisted Extraction of Bioactive Compounds from Lentil Wastes: Antioxidant Activity Evaluation and Metabolomic Characterization
2022-01-01 Cavalluzzi, Maria Maddalena; Lamonaca, Antonella; Rotondo, Natalie Paola; Miniero, Daniela Valeria; Muraglia, Marilena; Gabriele, Paola; Corbo, Filomena; De Palma, Annalisa; Budriesi, Roberta; De Angelis, Elisabetta; Monaci, Linda; Lentini, Giovanni
hERG stereoselective modulation by mexiletine‐derived ureas: Molecular docking study, synthesis, and biological evaluation
2023-01-01 Milani, Gualtiero; Budriesi, Roberta; Tavazzani, Elisa; Cavalluzzi, MARIA MADDALENA; Beatrice Mattioli, Laura; Miniero, DANIELA VALERIA; Delre, Pietro; Belviso, BENNY DANILO; Denegri, Marco; Cuocci, Corrado; Rotondo, NATALIE PAOLA; DE PALMA, Annalisa; Gualdani, Roberta; Caliandro, Rocco; Mangiatordi, Giuseppe Felice; Kumawat, Amit; Camilloni, Carlo; Priori, Silvia; Lentini, Giovanni
Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults
2024-01-01 Samarelli, Francesco; Purgatorio, Rosa; Lopopolo, Gianfranco; Deruvo, Caterina; Catto, Marco; Andresini, Michael; Carrieri, Antonio; Nicolotti, Orazio; DE PALMA, Annalisa; Miniero, DANIELA VALERIA; DE CANDIA, Modesto; Altomare, Cosimo D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis, antiarrhythmic activity, and toxicological evaluation of mexiletine analogues | 1-gen-2016 | Roselli, Mariagrazia; Carocci, Alessia; Budriesi, Roberta; Micucci, Matteo; Toma, Maddalena; Di Cesare Mannelli, Lorenzo; Lovece, Angelo; Catalano, Alessia; Cavalluzzi, MARIA MADDALENA; Bruno, Claudio; DE PALMA, Annalisa; Contino, Marialessandra; Perrone, MARIA GRAZIA; Colabufo, Nicola Antonio; Chiarini, Alberto; Franchini, Carlo; Ghelardini, Carla; Habtemariam, Solomon; Lentini, Giovanni | |
The mitochondrial carnitine/acylcarnitine carrier is regulated by hydrogen sulfide via interaction with C136 and C155 | 1-gen-2016 | Giangregorio, Nicola; Tonazzi, Annamaria; Console, Lara; Lorusso, Imma; DE PALMA, Annalisa; Indiveri, Cesare | |
Nitric oxide inhibits the mitochondrial carnitine/acylcarnitine carrier through reversible S-nitrosylation of cysteine 136 | 1-gen-2017 | Tonazzi, Annamaria; Giangregorio, Nicola; Console, Lara; DE PALMA, Annalisa; Indiveri, Cesare | |
Nitro-substituted tetrahydroindolizines and homologs: Design, kinetics, and mechanism of α-glucosidase inhibition | 1-gen-2017 | Tavani, Cinzia; Bianchi, Lara; DE PALMA, Annalisa; Passeri, GIOVANNA ILARIA; Punzi, Giuseppe; Pierri, CIRO LEONARDO; Lovece, Angelo; Cavalluzzi, MARIA MADDALENA; Franchini, Carlo; Lentini, Giovanni; Petrillo, Giovanni | |
Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties | 1-gen-2017 | Pisani, Leonardo; Catto, Marco; DE PALMA, Annalisa; Farina, Roberta; Cellamare, Saverio; Altomare, Cosimo Damiano | |
Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: a water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity | 1-gen-2017 | Pisani, Leonardo; DE PALMA, Annalisa; Giangregorio, Nicola; Miniero, DANIELA VALERIA; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo Damiano; Catto, Marco | |
Fitocomplesso polifenolico standardizzato per la prevenzione delle patologie correlate all’esposizione da sostanze reattive dell’ossigeno e relativo metodo di produzione | 1-gen-2017 | Cavalluzzi, MARIA MADDALENA; Mallamaci, Rosanna; Clodoveo, MARIA LISA; Moretti, Umberto; Lentini, Giovanni; Franchini, Carlo; Moretti, Pasquale; DE PALMA, Annalisa; Pisano, Isabella; Corbo, Filomena Faustina Rina; MASSARI CLAUDIO, Domenico | |
Insights into Structure-Activity Relationships of 3-Arylhydrazonoindolin-2-One Derivatives for Their Multitarget Activity on β-Amyloid Aggregation and Neurotoxicity | 1-gen-2018 | Purgatorio, Rosa; de Candia, M; De Palma, A; DE SANTIS, Francesco; Pisani, L; Campagna, F; Cellamare, S; Altomare, Cd; Catto, M | |
Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease | 1-gen-2019 | Purgatorio, R.; de Candia, M.; Catto, M.; Carrieri, A.; Pisani, L.; De Palma, A.; Toma, M.; Ivanova, O. A.; Voskressensky, L. G.; Altomare, C. D. | |
Chiral Separation, X-ray Structure, and Biological Evaluation of a Potent and Reversible Dual Binding Site AChE Inhibitor | 1-gen-2020 | Catto, Marco; Pisani, Leonardo; de la Mora, Eugenio; Belviso, Benny Danilo; Mangiatordi, Giuseppe Felice; Pinto, Andrea; Palma, Annalisa De; Denora, Nunzio; Caliandro, Rocco; Colletier, Jacques-Philippe; Silman, Israel; Nicolotti, Orazio; Altomare, Cosimo Damiano | |
Scouting around 1,2,3,4-Tetrahydrochromeno[3,2-c]pyridin-10-ones for Single- and Multitarget Ligands Directed towards Relevant Alzheimer's Targets | 1-gen-2020 | Purgatorio, R.; Kulikova, L. N.; Pisani, L.; Catto, M.; de Candia, M.; Carrieri, A.; Cellamare, S.; De Palma, A.; Beloglazkin, A. A.; Reza Raesi, G.; Voskressensky, L. G.; Altomare, C. D. | |
The interaction of hemin, a porphyrin derivative, with the purified rat brain 2-oxoglutarate carrier | 1-gen-2021 | Miniero, D. V.; Spagnoletta, A.; Gambacorta, N.; Scalera, V.; Pierri, C. L.; Nicolotti, O.; De Palma, A. | |
Synthesis and Evaluation of Voltage-Gated Sodium Channel Blocking Pyrroline Derivatives Endowed with Both Antiarrhythmic and Antioxidant Activities | 1-gen-2021 | Carocci, Alessia; Roselli, Mariagrazia; Budriesi, Roberta; Micucci, Matteo; Desaphy, Jean-François; Altamura, Concetta; Cavalluzzi, Maria Maddalena; Toma, Maddalena; Passeri, Giovanna Ilaria; Milani, Gualtiero; Lovece, Angelo; Catalano, Alessia; Bruno, Claudio; De Palma, Annalisa; Corbo, Filomena; Franchini, Carlo; Habtemariam, Solomon; Lentini, Giovanni | |
Densely Functionalized 2-Methylideneazetidines: Evaluation as Antibacterials | 1-gen-2021 | Petrillo, Giovanni; Tavani, Cinzia; Bianchi, Lara; Benzi, Alice; Cavalluzzi, MARIA MADDALENA; Salvagno, Lara; Quintieri, Laura; DE PALMA, Annalisa; Caputo, Leonardo; Rosato, Antonio; Lentini, Giovanni | |
New Insights Regarding Hemin Inhibition of the Purified Rat Brain 2-Oxoglutarate Carrier and Relationships with Mitochondrial Dysfunction | 1-gen-2022 | Miniero, DANIELA VALERIA; Gambacorta, Nicola; Spagnoletta, Anna; Tragni, Vincenzo; Loizzo, Stefano; Nicolotti, Orazio; Pierri, CIRO LEONARDO; DE PALMA, Annalisa | |
Microwave-Assisted Extraction of Bioactive Compounds from Lentil Wastes: Antioxidant Activity Evaluation and Metabolomic Characterization | 1-gen-2022 | Cavalluzzi, Maria Maddalena; Lamonaca, Antonella; Rotondo, Natalie Paola; Miniero, Daniela Valeria; Muraglia, Marilena; Gabriele, Paola; Corbo, Filomena; De Palma, Annalisa; Budriesi, Roberta; De Angelis, Elisabetta; Monaci, Linda; Lentini, Giovanni | |
hERG stereoselective modulation by mexiletine‐derived ureas: Molecular docking study, synthesis, and biological evaluation | 1-gen-2023 | Milani, Gualtiero; Budriesi, Roberta; Tavazzani, Elisa; Cavalluzzi, MARIA MADDALENA; Beatrice Mattioli, Laura; Miniero, DANIELA VALERIA; Delre, Pietro; Belviso, BENNY DANILO; Denegri, Marco; Cuocci, Corrado; Rotondo, NATALIE PAOLA; DE PALMA, Annalisa; Gualdani, Roberta; Caliandro, Rocco; Mangiatordi, Giuseppe Felice; Kumawat, Amit; Camilloni, Carlo; Priori, Silvia; Lentini, Giovanni | |
Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults | 1-gen-2024 | Samarelli, Francesco; Purgatorio, Rosa; Lopopolo, Gianfranco; Deruvo, Caterina; Catto, Marco; Andresini, Michael; Carrieri, Antonio; Nicolotti, Orazio; DE PALMA, Annalisa; Miniero, DANIELA VALERIA; DE CANDIA, Modesto; Altomare, Cosimo D. |
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