Sfoglia per Autore
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues
2005-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A.
Solid-phase and Microwave Assisted Synthesis of Focused libraries of Imatinib analogues
2005-01-01 Leonetti, F; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Stefanachi, Angela; Carotti, A.
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies
2005-01-01 Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio
Synthesis of heterocyclic compound libraries by automated sequential and parallel microwave synthesis.
2006-01-01 Pisani, L.; Prokopcová, H.; Kappe, C. O.
Application of Liebeskind-Srogl Thioester-Boronic Acid Couplings for the Scaffold Decoration of Dihydropyrimidines
2006-01-01 Pisani, L.; Prokopcová, H.; Kappe, C. O.
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors
2007-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo
Synthesis of 5-Aroyldihydropyrimidinones via Liebeskind–Srogl Thiol Ester– Boronic Acid Cross-Couplings
2007-01-01 Prokopcová, Hana; Pisani, Leonardo; Oliver Kappe, C.
5-aroyl-3,4-dihydropyrimidin-2-one library generation via automated sequential and parallel microwave-assisted synthesis techniques
2007-01-01 Pisani, Leonardo; Prokopcová, Hana; Kremsner, Jennifer M.; Oliver Kappe, C.
Structures of Human Monoamine Oxidase B Complexes with Selective Noncovalent Inhibitors: Safinamide and Coumarin Analogs
2007-01-01 Binda, C; Wang, J; Pisani, Leonardo; Caccia, C; Carotti, Angelo; Salvati, P; Edmondson, D. E.; Mattevi, A.
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors
2008-01-01 Leonetti, Francesco; Catto, Marco; Nicolotti, Orazio; Pisani, Leonardo; Cappa, A; Stefanachi, Angela; Carotti, Angelo
Discovery of a Novel Class of Potent Coumarin MAO-B inhibitors: Development and Biopharmacological Profiling of 7-[(3-Chlorobenzyl)oxy]-4-[(methylamino)methyl]-2H-chromen-2-one methanesulfonate (NW-1772) as a Highly Potent, Selective, Reversible and Orally Active MAO-B inhibitor
2009-01-01 Pisani, Leonardo; Muncipinto, G; Miscioscia, Tf; Nicolotti, Orazio; Leonetti, Francesco; Catto, Marco; Caccia, C; Salvati, P; SOTO OTERO, R; MENDEZ ALVAREZ, E; Passeleu, C; Carotti, A.
Solid phase synthesis of potential PKs inhibitors
2009-01-01 Pellegrino, G; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Stefanachi, Angela; Pisani, Leonardo; Carotti, A.
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity
2009-01-01 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
Solid phase synthesis of a molecular library of pyrimidines, pyrazoles and isoxazoles with biological potential
2010-01-01 Pellegrino, G; Leonetti, F; Carotti, Angelo; Nicolotti, Orazio; Pisani, Leonardo; Stefanachi, Angela; Catto, Marco
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor.
2010-01-01 Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A.
Ring closing metathesis mediated synthesis of d-, g- and e-N-HydroxylactaMS as potential coordinating molecular fragments of biologically relevant bivalent metals XX
2010-01-01 Leonetti, Francesco; Muncipinto, G; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Pisani, Leonardo; Carotti, A.
Design, Synthesis and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors
2010-01-01 Pisani, Leonardo; Catto, Marco; Giangreco, I; Leonetti, Francesco; Nicolotti, Orazio; Stefanachi, Angela; Cellamare, Saverio; Carotti, Angelo
Screening of benzamidine-based thrombin inhibitors via a linear interaction energy in continuum electrostatics model
2010-01-01 Nicolotti, Orazio; Giangreco, I; Miscioscia, Tf; Convertino, M; Leonetti, Francesco; Pisani, Leonardo; Carotti, Angelo
Discovery of a potent and selective hetero-bivalent AChE inhibitor via bioisosteric replacement
2011-01-01 Nicolotti, Orazio; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Giangreco, I.; Stefanachi, Angela; Carotti, Angelo
Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity
2011-01-01 CONEJO GARCÍA, A; Pisani, Leonardo; DEL CARMEN NÚÑEZ, M; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Campos, J; Gallo, M; Espinosa, A; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues | 1-gen-2005 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A. | |
Solid-phase and Microwave Assisted Synthesis of Focused libraries of Imatinib analogues | 1-gen-2005 | Leonetti, F; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Stefanachi, Angela; Carotti, A. | |
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies | 1-gen-2005 | Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio | |
Synthesis of heterocyclic compound libraries by automated sequential and parallel microwave synthesis. | 1-gen-2006 | Pisani, L.; Prokopcová, H.; Kappe, C. O. | |
Application of Liebeskind-Srogl Thioester-Boronic Acid Couplings for the Scaffold Decoration of Dihydropyrimidines | 1-gen-2006 | Pisani, L.; Prokopcová, H.; Kappe, C. O. | |
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors | 1-gen-2007 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo | |
Synthesis of 5-Aroyldihydropyrimidinones via Liebeskind–Srogl Thiol Ester– Boronic Acid Cross-Couplings | 1-gen-2007 | Prokopcová, Hana; Pisani, Leonardo; Oliver Kappe, C. | |
5-aroyl-3,4-dihydropyrimidin-2-one library generation via automated sequential and parallel microwave-assisted synthesis techniques | 1-gen-2007 | Pisani, Leonardo; Prokopcová, Hana; Kremsner, Jennifer M.; Oliver Kappe, C. | |
Structures of Human Monoamine Oxidase B Complexes with Selective Noncovalent Inhibitors: Safinamide and Coumarin Analogs | 1-gen-2007 | Binda, C; Wang, J; Pisani, Leonardo; Caccia, C; Carotti, Angelo; Salvati, P; Edmondson, D. E.; Mattevi, A. | |
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors | 1-gen-2008 | Leonetti, Francesco; Catto, Marco; Nicolotti, Orazio; Pisani, Leonardo; Cappa, A; Stefanachi, Angela; Carotti, Angelo | |
Discovery of a Novel Class of Potent Coumarin MAO-B inhibitors: Development and Biopharmacological Profiling of 7-[(3-Chlorobenzyl)oxy]-4-[(methylamino)methyl]-2H-chromen-2-one methanesulfonate (NW-1772) as a Highly Potent, Selective, Reversible and Orally Active MAO-B inhibitor | 1-gen-2009 | Pisani, Leonardo; Muncipinto, G; Miscioscia, Tf; Nicolotti, Orazio; Leonetti, Francesco; Catto, Marco; Caccia, C; Salvati, P; SOTO OTERO, R; MENDEZ ALVAREZ, E; Passeleu, C; Carotti, A. | |
Solid phase synthesis of potential PKs inhibitors | 1-gen-2009 | Pellegrino, G; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Stefanachi, Angela; Pisani, Leonardo; Carotti, A. | |
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity | 1-gen-2009 | Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A. | |
Solid phase synthesis of a molecular library of pyrimidines, pyrazoles and isoxazoles with biological potential | 1-gen-2010 | Pellegrino, G; Leonetti, F; Carotti, Angelo; Nicolotti, Orazio; Pisani, Leonardo; Stefanachi, Angela; Catto, Marco | |
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor. | 1-gen-2010 | Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A. | |
Ring closing metathesis mediated synthesis of d-, g- and e-N-HydroxylactaMS as potential coordinating molecular fragments of biologically relevant bivalent metals XX | 1-gen-2010 | Leonetti, Francesco; Muncipinto, G; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Pisani, Leonardo; Carotti, A. | |
Design, Synthesis and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors | 1-gen-2010 | Pisani, Leonardo; Catto, Marco; Giangreco, I; Leonetti, Francesco; Nicolotti, Orazio; Stefanachi, Angela; Cellamare, Saverio; Carotti, Angelo | |
Screening of benzamidine-based thrombin inhibitors via a linear interaction energy in continuum electrostatics model | 1-gen-2010 | Nicolotti, Orazio; Giangreco, I; Miscioscia, Tf; Convertino, M; Leonetti, Francesco; Pisani, Leonardo; Carotti, Angelo | |
Discovery of a potent and selective hetero-bivalent AChE inhibitor via bioisosteric replacement | 1-gen-2011 | Nicolotti, Orazio; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Giangreco, I.; Stefanachi, Angela; Carotti, Angelo | |
Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity | 1-gen-2011 | CONEJO GARCÍA, A; Pisani, Leonardo; DEL CARMEN NÚÑEZ, M; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Campos, J; Gallo, M; Espinosa, A; Carotti, Angelo |
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