Sfoglia per Autore
REAZIONE DI ALOGENOBENZONITRILI CON LDA: UN CASO DI MECCANISMO BENZINICO DOVUTO ALL’INGOMBRO STERICO DEL NUCLEOFILO
2008-01-01 Vitale, Paola; LEONARDO DI, Nunno; Davide, Nardi; Scilimati, Antonio
Functionalized diarylisoxazoles inhibitors of cyclooxygenase
2008-01-01 Scilimati, Antonio; Vitale, Paola; DI NUNNO, L; Patrignani, P; Tacconelli, S; Capone, M. L.
Stereospecific synthesis and bio-activity of novel beta3-adrenoceptor agonists and inverse agonists
2008-01-01 Perrone, MARIA GRAZIA; Santandrea, E; Bleve, L; Vitale, Paola; Colabufo, Nicola Antonio; Jockers, R; Milazzo, F. M.; Sciarroni, A. F.; Scilimati, Antonio
Effect of the aryl group substituent in the dimerization of 3-arylisoxazoles to syn 2,6-diaryl-3,7-diazatricyclo[4.2.0.02,5]octan-4,8-diones induced by LDA
2008-01-01 DI NUNNO, L; Vitale, Paola; Scilimati, Antonio
3-Substituted-5-phenylthio-2-isoxazolines: synthesis and reactions with bases
2009-01-01 Vitale, Paola; DI NUNNO, L.; Scilimati, Antonio
Highly selective COX-1 inhibitors as novel cardioprotective anti-thrombotic agents
2009-01-01 Perrone, MARIA GRAZIA; Simone, L; Vitale, Paola; DI NUNNO, L; Scilimati, Antonio; Lavecchia, A; Novellino, E; Capone, M. L.; Tacconelli, S; Patrignani, P.
The tertiary amine nitrogen atom of piperazine sulfonamides as a novel determinant of potent and selective beta3-adrenoceptor agonists
2009-01-01 Perrone, MARIA GRAZIA; Bleve, L; Santandrea, E; Vitale, Paola; Niso, Mauro; Scilimati, Antonio
Use of isoxazole derivatives as cyclooxygenase inhibitors
2010-01-01 Scilimati, Antonio; DI NUNNO, L; Vitale, Paola; Patrignani, P; Tacconelli, S; Porreca, E; Stuppia, L.
A Novel Synthesis of N-Unsubstituted beta-Enamino Thioesters from 3-Arylisoxazoles and 3-Aryl-5-phenylthio-2-isoxazolines
2010-01-01 Vitale, Paola; DI NUNNO, L; Scilimati, Antonio
Selective COX-1 inhibition: a therapeutic target to be reconsidered
2010-01-01 Perrone, MARIA GRAZIA; Scilimati, Antonio; Simone, L.; Vitale, Paola
Synthesis of N,N-dialkylaminobenzonitriles and halo-(N,N-dialkyl) benzamidines by reaction of halobenzonitriles with lithium amides
2011-01-01 Vitale, Paola; DI NUNNO, L; Scilimati, Antonio
Enantioselective bio-reduction of prochiral ketones by the non-conventional yeast Kluyveromyces marxianus
2011-01-01 Vitale, Paola; Perna, Filippo; Perrone, Mg; Scilimati, Antonio
Selective inhibition of cyclooxygenase (COX) isoenzymes and neuroinflammation
2011-01-01 Malerba, P.; Perrone, MARIA GRAZIA; Vitale, Paola; Scilimati, Antonio
Isoxazole and pyrazole core in COX-1 inhibitors
2011-01-01 Vitale, Paola; P., Malerba; M. G., Perrone; Scilimati, Antonio
Screening on the use of Kluyveromyces marxianus CBS 6556 growing cells as enantioselective biocatalyst for ketones reduction
2011-01-01 Vitale, Paola; Perna, Filippo; Perrone, M. G.; Scilimati, Antonio
Synthesis of N,N-dialkylaminobenzonitriles and halo-(N,N-dialkyl)benzamidines by reaction of halobenzonitriles with lithium amides
2011-01-01 Vitale, Paola; DI NUNNO, L; Scilimati, Antonio
Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition
2012-01-01 Perrone, M. G.; Vitale, P.; Malerba, P.; Altomare, A.; Rizzi, R.; Lavecchia, A.; Digiovanni, C.; Novellino, E.; Scilimati, A.
Novel selective COX-1 inhibitors suppress neuroinflammatory mediators in LPS-stimulated N13 microglial cells
2012-01-01 Calvello, Rosa; Panaro, Maria Antonietta; Carbone, M. L.; Cianciulli, Antonia; Perrone, MARIA GRAZIA; Vitale, Paola; Malerba, P.; Scilimati, Antonio
Novel pyrazoles and their radiolabeled derivatives useful as COX-1 selective inhibitors
2013-01-01 Scilimati, Antonio; Perrone, MARIA GRAZIA; Vitale, Paola
Synthesis, Pharmacological Characterization, and Docking Analysis of a Novel Family of Diarylisoxazoles as Highly Selective Cyclooxygenase‑1 (COX-1) Inhibitors
2013-01-01 Vitale, Paola; Tacconelli, Stefania; Perrone, MARIA GRAZIA; Malerba, Paola; Simone, Laura; Scilimati, Antonio; Lavecchia, Antonio; Dovizio, Melania; Marcantoni, Emanuela; Bruno, Annalisa; Patrignani, Paola
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
REAZIONE DI ALOGENOBENZONITRILI CON LDA: UN CASO DI MECCANISMO BENZINICO DOVUTO ALL’INGOMBRO STERICO DEL NUCLEOFILO | 1-gen-2008 | Vitale, Paola; LEONARDO DI, Nunno; Davide, Nardi; Scilimati, Antonio | |
Functionalized diarylisoxazoles inhibitors of cyclooxygenase | 1-gen-2008 | Scilimati, Antonio; Vitale, Paola; DI NUNNO, L; Patrignani, P; Tacconelli, S; Capone, M. L. | |
Stereospecific synthesis and bio-activity of novel beta3-adrenoceptor agonists and inverse agonists | 1-gen-2008 | Perrone, MARIA GRAZIA; Santandrea, E; Bleve, L; Vitale, Paola; Colabufo, Nicola Antonio; Jockers, R; Milazzo, F. M.; Sciarroni, A. F.; Scilimati, Antonio | |
Effect of the aryl group substituent in the dimerization of 3-arylisoxazoles to syn 2,6-diaryl-3,7-diazatricyclo[4.2.0.02,5]octan-4,8-diones induced by LDA | 1-gen-2008 | DI NUNNO, L; Vitale, Paola; Scilimati, Antonio | |
3-Substituted-5-phenylthio-2-isoxazolines: synthesis and reactions with bases | 1-gen-2009 | Vitale, Paola; DI NUNNO, L.; Scilimati, Antonio | |
Highly selective COX-1 inhibitors as novel cardioprotective anti-thrombotic agents | 1-gen-2009 | Perrone, MARIA GRAZIA; Simone, L; Vitale, Paola; DI NUNNO, L; Scilimati, Antonio; Lavecchia, A; Novellino, E; Capone, M. L.; Tacconelli, S; Patrignani, P. | |
The tertiary amine nitrogen atom of piperazine sulfonamides as a novel determinant of potent and selective beta3-adrenoceptor agonists | 1-gen-2009 | Perrone, MARIA GRAZIA; Bleve, L; Santandrea, E; Vitale, Paola; Niso, Mauro; Scilimati, Antonio | |
Use of isoxazole derivatives as cyclooxygenase inhibitors | 1-gen-2010 | Scilimati, Antonio; DI NUNNO, L; Vitale, Paola; Patrignani, P; Tacconelli, S; Porreca, E; Stuppia, L. | |
A Novel Synthesis of N-Unsubstituted beta-Enamino Thioesters from 3-Arylisoxazoles and 3-Aryl-5-phenylthio-2-isoxazolines | 1-gen-2010 | Vitale, Paola; DI NUNNO, L; Scilimati, Antonio | |
Selective COX-1 inhibition: a therapeutic target to be reconsidered | 1-gen-2010 | Perrone, MARIA GRAZIA; Scilimati, Antonio; Simone, L.; Vitale, Paola | |
Synthesis of N,N-dialkylaminobenzonitriles and halo-(N,N-dialkyl) benzamidines by reaction of halobenzonitriles with lithium amides | 1-gen-2011 | Vitale, Paola; DI NUNNO, L; Scilimati, Antonio | |
Enantioselective bio-reduction of prochiral ketones by the non-conventional yeast Kluyveromyces marxianus | 1-gen-2011 | Vitale, Paola; Perna, Filippo; Perrone, Mg; Scilimati, Antonio | |
Selective inhibition of cyclooxygenase (COX) isoenzymes and neuroinflammation | 1-gen-2011 | Malerba, P.; Perrone, MARIA GRAZIA; Vitale, Paola; Scilimati, Antonio | |
Isoxazole and pyrazole core in COX-1 inhibitors | 1-gen-2011 | Vitale, Paola; P., Malerba; M. G., Perrone; Scilimati, Antonio | |
Screening on the use of Kluyveromyces marxianus CBS 6556 growing cells as enantioselective biocatalyst for ketones reduction | 1-gen-2011 | Vitale, Paola; Perna, Filippo; Perrone, M. G.; Scilimati, Antonio | |
Synthesis of N,N-dialkylaminobenzonitriles and halo-(N,N-dialkyl)benzamidines by reaction of halobenzonitriles with lithium amides | 1-gen-2011 | Vitale, Paola; DI NUNNO, L; Scilimati, Antonio | |
Diarylheterocycle Core Ring Features Effect in Selective COX-1 Inhibition | 1-gen-2012 | Perrone, M. G.; Vitale, P.; Malerba, P.; Altomare, A.; Rizzi, R.; Lavecchia, A.; Digiovanni, C.; Novellino, E.; Scilimati, A. | |
Novel selective COX-1 inhibitors suppress neuroinflammatory mediators in LPS-stimulated N13 microglial cells | 1-gen-2012 | Calvello, Rosa; Panaro, Maria Antonietta; Carbone, M. L.; Cianciulli, Antonia; Perrone, MARIA GRAZIA; Vitale, Paola; Malerba, P.; Scilimati, Antonio | |
Novel pyrazoles and their radiolabeled derivatives useful as COX-1 selective inhibitors | 1-gen-2013 | Scilimati, Antonio; Perrone, MARIA GRAZIA; Vitale, Paola | |
Synthesis, Pharmacological Characterization, and Docking Analysis of a Novel Family of Diarylisoxazoles as Highly Selective Cyclooxygenase‑1 (COX-1) Inhibitors | 1-gen-2013 | Vitale, Paola; Tacconelli, Stefania; Perrone, MARIA GRAZIA; Malerba, Paola; Simone, Laura; Scilimati, Antonio; Lavecchia, Antonio; Dovizio, Melania; Marcantoni, Emanuela; Bruno, Annalisa; Patrignani, Paola |
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