Sfoglia per Autore
Structure Activity Studies of a Novel Cytotoxic Benzodiazepine
2003-01-01 Boitano, A.; Emal, C. D.; Leonetti, Francesco; Blatt, N. B.; Dineen, T. A.; Ellman, J. A.; Roush, W. R.; Opipari, A. W.; Glick, G. D.
Structure-Based Design, Solid Phase Synthesis and SAFIR of New Dual Binding Site Acetylcholinesterase (AChE) Inhibitors.
2003-01-01 Leonetti, Francesco; Cappa, A; Catto, Marco; Carotti, A.
Insights into Diastereospecific Solvolysis of Peptidyl-β-Lactams: Combined Kinetic and Conformational Studies.
2003-01-01 Cellamare, Saverio; Coletti, A; Leonetti, Francesco; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A; Cellamare, S.
Synthesis of potential dual binding site acetylcholinesterase inhibitors through an efficient solid phase approach based on Mitsunobu reaction
2004-01-01 Leonetti, Francesco; Cappa, A.; Maccallini, C.; Carotti, Angelo
Sintesi su Fase Solida della Safinamide e di suoi Analoghi.
2004-01-01 Leonetti, Francesco; Salvati, P; Caccia, C; Ferappi, M; Carotti, A.
Design, Synthesis, and 3D QSAR of Novel Potent and Selective Aromatase Inhibitors
2004-01-01 Leonetti, Francesco; Favia, A.; Rao, A.; Aliano, R.; Paluszcak, A.; Hartmann, R. W.; Carotti, Angelo
olid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues.
2005-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, A; Carotti, A. S.
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies
2005-01-01 Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues
2005-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A.
Microwave-assisted solid phase synthesis of Imatinib, a blockbuster anticancer drug.
2006-01-01 Leonetti, Francesco; Capaldi, C; Carotti, A.
A novel function for non-deterministic scouting of optimal QSAR models out of a highly-structured physicochemical space.
2006-01-01 Nicolotti, Orazio; Miscioscia, T. F.; Leonetti, Francesco; Carotti, A.
Structural Insights into MAO Inhibitory Potency and Selectivity of 7-substituted Coumarins from Ligand- and Target-based Approaches
2006-01-01 Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Carotti, Angelo; Favia, Ad; SOTO OTERO, R; MENDEZ ALVAREZ, E; Carotti, A.
Substrate profiling of cysteine proteases using a combinatorial peptide library identifies functionally unique specificities
2006-01-01 Choe, Y; Leonetti, Francesco; Greenbaum, D. C.; Lecaille, F; Bogyo, M; Brmme, D; Ellman, J. A.; Craik, C. S.
Impact of species-dependent differences on screening, design, and development of MAO B inhibitors
2006-01-01 Novaroli, L; Daina, A; Favre, E; Bravo, J; Carotti, Angelo; Leonetti, Francesco; Catto, Marco; Carrupt, P. A.; Reist, M.
Screening of matrix metalloproteinases available from the protein data bank: Insights into biological functions, domain organization, and zinc binding groups
2007-01-01 Nicolotti, Orazio; Miscioscia, Tf; Leonetti, Francesco; Muncipinto, G; Carotti, A.
Microwave-assisted solid phase synthesis of Imatinib, a blockbuster anticancer drug
2007-01-01 Leonetti, Francesco; Capaldi, C; Carotti, Angelo
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors
2007-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo
Synthesis and Monoamine Oxidase Inhibitory Activity of new Pyridazine-, Pyrimidine and 1,2,4 Triazine containing Tryciclic derivatives
2007-01-01 Carotti, Angelo; Catto, Marco; Leonetti, Francesco; Campagna, F.; SOTO OTERO, R.; MENDEZ ALVAREZ, E.; Thull, U.; Testa, B.; Altomare, Cosimo Damiano
A new approach to combine ligand- and structure-based drug design.
2008-01-01 Nicolotti, Orazio; Miscioscia, Tf; Carotti, A; Leonetti, Francesco; Giangreco, I; Carotti, A.
An integrated methodology to interface structure- and ligand-based drug design
2008-01-01 Giangreco, I; Nicolotti, Orazio; Miscioscia, Tf; Tedeschi, P; Carotti, A; Leonetti, Francesco; Carotti, A.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Structure Activity Studies of a Novel Cytotoxic Benzodiazepine | 1-gen-2003 | Boitano, A.; Emal, C. D.; Leonetti, Francesco; Blatt, N. B.; Dineen, T. A.; Ellman, J. A.; Roush, W. R.; Opipari, A. W.; Glick, G. D. | |
Structure-Based Design, Solid Phase Synthesis and SAFIR of New Dual Binding Site Acetylcholinesterase (AChE) Inhibitors. | 1-gen-2003 | Leonetti, Francesco; Cappa, A; Catto, Marco; Carotti, A. | |
Insights into Diastereospecific Solvolysis of Peptidyl-β-Lactams: Combined Kinetic and Conformational Studies. | 1-gen-2003 | Cellamare, Saverio; Coletti, A; Leonetti, Francesco; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A; Cellamare, S. | |
Synthesis of potential dual binding site acetylcholinesterase inhibitors through an efficient solid phase approach based on Mitsunobu reaction | 1-gen-2004 | Leonetti, Francesco; Cappa, A.; Maccallini, C.; Carotti, Angelo | |
Sintesi su Fase Solida della Safinamide e di suoi Analoghi. | 1-gen-2004 | Leonetti, Francesco; Salvati, P; Caccia, C; Ferappi, M; Carotti, A. | |
Design, Synthesis, and 3D QSAR of Novel Potent and Selective Aromatase Inhibitors | 1-gen-2004 | Leonetti, Francesco; Favia, A.; Rao, A.; Aliano, R.; Paluszcak, A.; Hartmann, R. W.; Carotti, Angelo | |
olid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues. | 1-gen-2005 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, A; Carotti, A. S. | |
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies | 1-gen-2005 | Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio | |
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues | 1-gen-2005 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A. | |
Microwave-assisted solid phase synthesis of Imatinib, a blockbuster anticancer drug. | 1-gen-2006 | Leonetti, Francesco; Capaldi, C; Carotti, A. | |
A novel function for non-deterministic scouting of optimal QSAR models out of a highly-structured physicochemical space. | 1-gen-2006 | Nicolotti, Orazio; Miscioscia, T. F.; Leonetti, Francesco; Carotti, A. | |
Structural Insights into MAO Inhibitory Potency and Selectivity of 7-substituted Coumarins from Ligand- and Target-based Approaches | 1-gen-2006 | Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Carotti, Angelo; Favia, Ad; SOTO OTERO, R; MENDEZ ALVAREZ, E; Carotti, A. | |
Substrate profiling of cysteine proteases using a combinatorial peptide library identifies functionally unique specificities | 1-gen-2006 | Choe, Y; Leonetti, Francesco; Greenbaum, D. C.; Lecaille, F; Bogyo, M; Brmme, D; Ellman, J. A.; Craik, C. S. | |
Impact of species-dependent differences on screening, design, and development of MAO B inhibitors | 1-gen-2006 | Novaroli, L; Daina, A; Favre, E; Bravo, J; Carotti, Angelo; Leonetti, Francesco; Catto, Marco; Carrupt, P. A.; Reist, M. | |
Screening of matrix metalloproteinases available from the protein data bank: Insights into biological functions, domain organization, and zinc binding groups | 1-gen-2007 | Nicolotti, Orazio; Miscioscia, Tf; Leonetti, Francesco; Muncipinto, G; Carotti, A. | |
Microwave-assisted solid phase synthesis of Imatinib, a blockbuster anticancer drug | 1-gen-2007 | Leonetti, Francesco; Capaldi, C; Carotti, Angelo | |
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors | 1-gen-2007 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo | |
Synthesis and Monoamine Oxidase Inhibitory Activity of new Pyridazine-, Pyrimidine and 1,2,4 Triazine containing Tryciclic derivatives | 1-gen-2007 | Carotti, Angelo; Catto, Marco; Leonetti, Francesco; Campagna, F.; SOTO OTERO, R.; MENDEZ ALVAREZ, E.; Thull, U.; Testa, B.; Altomare, Cosimo Damiano | |
A new approach to combine ligand- and structure-based drug design. | 1-gen-2008 | Nicolotti, Orazio; Miscioscia, Tf; Carotti, A; Leonetti, Francesco; Giangreco, I; Carotti, A. | |
An integrated methodology to interface structure- and ligand-based drug design | 1-gen-2008 | Giangreco, I; Nicolotti, Orazio; Miscioscia, Tf; Tedeschi, P; Carotti, A; Leonetti, Francesco; Carotti, A. |
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