Sfoglia per Autore
Novel small molecules for PPARs modulation and their potential use for treatment of metabolic disorders
2019-01-01 Laghezza, Antonio; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio
Identification of Natural Scaffolds as New Multi-Functional Agents for the Treatment of Alzheimer’s Disease
2019-01-01 Laghezza, Antonio; Brunetti, Leonardo; Capriati, Vito; Catto, Marco; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca; Solfrizzo, Michele
Natural compounds as FAAH inhibitors: preliminary screening and potential developments
2019-01-01 Brunetti, L.; Laghezza, A.; Loiodice, F.; Piemontese, L.; Tortorella, P.
Peroxisome Proliferator Activated Receptor (PPAR) agonists as Fatty Acid Amide Hydrolase (FAAH) inhibitors: screening and preliminary structure-activity relationships
2019-01-01 Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio
New Approaches to Cancer Therapy: Combining Fatty Acid Amide Hydrolase (FAAH) Inhibition with Peroxisome Proliferator-Activated Receptors (PPARs) Activation
2019-01-01 Brunetti, Leonardo; Loiodice, Fulvio; Piemontese, Luca; Tortorella, Paolo; Laghezza, Antonio
Importance of Biometals as Targets in Medicinal Chemistry: An Overview about the Role of Zinc (II) Chelating Agents
2020-01-01 Leuci, Rosalba; Brunetti, Leonardo; Laghezza, Antonio; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca
Beyond the Canonical Endocannabinoid System. A Screening of PPAR Ligands as FAAH Inhibitors
2020-01-01 Brunetti, Leonardo; Carrieri, Antonio; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio; Laghezza, Antonio
Deep Eutectic Solvents as Effective Reaction Media for the Synthesis of 2‐Hydroxyphenylbenzimidazole-based Scaffolds en Route to Donepezil‐Like Compounds
2020-01-01 Piemontese, L.; Sergio, R.; Rinaldo, F.; Brunetti, L.; Perna, F. M.; Amelia Santos, M.; Capriati, V.
Bone-seeking matrix metalloproteinase inhibitors for the treatment of skeletal malignancy
2020-01-01 Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Di Pizio, A.; Pochetti, G.; Montanari, R.; Capelli, D.; Tauro, M.; Loiodice, F.; Tortorella, P.
Combining fatty acid amide hydrolase (FAAH) inhibition with peroxisome proliferator-activated receptor (PPAR) activation: a new potential multi-target therapeutic strategy for the treatment of Alzheimer’s disease
2020-01-01 Brunetti, Leonardo; Laghezza, Antonio; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca
A Review of Recent Patents (2016-2019) on Plant Food Supplements with Potential Application in the Treatment of Neurodegenerative and Metabolic Disorders
2020-01-01 Leuci, Rosalba; Brunetti, Leonardo; Laghezza, Antonio; Tortorella, Paolo; Loiodice, Fulvio; Piemontese, Luca
DEVELOPMENT OF PHENOXYALKYLPIPERIDINES AS HIGH-AFFINITY SIGMA-1 (s1) RECEPTOR LIGANDS WITH POTENT ANTI-AMNESIC ACTIVITY
2021-01-01 Laghezza, Antonio; Abatematteo, Francesca S.; Mosier, Philip D.; Niso, Mauro; Brunetti, Leonardo; Berardi, Francesco; Loiodice, Fulvio; Contino, Marialessandra; Delprat, Benjamin; Maurice, Tangui; Abate, Carmen
Derivatives of Tenuazonic Acid as Potential New Multi-Target Anti-Alzheimer’s Disease Agents
2021-01-01 Poliseno, Viviana; Chaves, Sílvia; Brunetti, Leonardo; Loiodice, Fulvio; Carrieri, Antonio; Laghezza, Antonio; Tortorella, Paolo; Magalhães, João D.; Cardoso, Sandra M.; Santos, M. Amélia; Piemontese, Luca
Natural Compounds for the Prevention and Treatment of Cardiovascular and Neurodegenerative Diseases
2021-01-01 Leuci, Rosalba; Brunetti, Leonardo; Poliseno, Viviana; Laghezza, Antonio; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca
(2-Aminobenzothiazole)-Methyl-1,1-bisphosphonic acids: Targeting matrix metalloproteinase 13 inhibition to the bone
2021-01-01 Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Loiodice, F.; Tortorella, P.
Multiple causes, multiple targets: FAAH as a centerpiece for therapy of multifactorial pathologies.
2021-01-01 Brunetti, Leonardo; Leuci, Rosalba; Carrieri, Antonio; Laghezza, Antonio; Catto, Marco; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio
Multi-Target Approach for the Design of New Compounds Potentially Useful for the Prevention and Treatment of Cardiovascular and/or Neurodegenerative Diseases
2021-01-01 Leuci, R.; Brunetti, L.; Carocci, A.; Carrieri, A.; Catto, M.; Laghezza, A.; Tortorella, P.; Piemontese, L.; Loiodice, F.
Novel Rivastigmine-Based Multitarget Hybrids For Potential Treatment of Alzheimer’s Disease: Cu(II) And Fe(III) Chelation Studies
2022-01-01 Vicente-Zurdo, David; Brunetti, Leonardo; Piemontese, Luca; Madrid, Yolanda; Chaves, Sílvia; Amélia Santos., M.
Novel rivastigmine structure-based hybrids for the potential treatment of Alzheimer’s disease
2022-01-01 Leuci, R.; Brunetti, L.; Carrieri, A.; Catto, M.; Laghezza, A.; Tortorella, P.; Loiodice, F.; Piemontese, L.
1,3,5-triazine derivatives as dual inhibitors of 5-HT6R/FAAH in search of new therapy for Alzheimer's disease
2022-01-01 Czarnota-Łydka, Kinga; Satała, Grzegorz; Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; DE CANDIA, Modesto; Purgatorio, Rosa; Gumułka, Magdalena; Kucwaj-Brysz, Katarzyna; Carrieri, Antonio; Handzlik, Jadwiga
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel small molecules for PPARs modulation and their potential use for treatment of metabolic disorders | 1-gen-2019 | Laghezza, Antonio; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio | |
Identification of Natural Scaffolds as New Multi-Functional Agents for the Treatment of Alzheimer’s Disease | 1-gen-2019 | Laghezza, Antonio; Brunetti, Leonardo; Capriati, Vito; Catto, Marco; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca; Solfrizzo, Michele | |
Natural compounds as FAAH inhibitors: preliminary screening and potential developments | 1-gen-2019 | Brunetti, L.; Laghezza, A.; Loiodice, F.; Piemontese, L.; Tortorella, P. | |
Peroxisome Proliferator Activated Receptor (PPAR) agonists as Fatty Acid Amide Hydrolase (FAAH) inhibitors: screening and preliminary structure-activity relationships | 1-gen-2019 | Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio | |
New Approaches to Cancer Therapy: Combining Fatty Acid Amide Hydrolase (FAAH) Inhibition with Peroxisome Proliferator-Activated Receptors (PPARs) Activation | 1-gen-2019 | Brunetti, Leonardo; Loiodice, Fulvio; Piemontese, Luca; Tortorella, Paolo; Laghezza, Antonio | |
Importance of Biometals as Targets in Medicinal Chemistry: An Overview about the Role of Zinc (II) Chelating Agents | 1-gen-2020 | Leuci, Rosalba; Brunetti, Leonardo; Laghezza, Antonio; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca | |
Beyond the Canonical Endocannabinoid System. A Screening of PPAR Ligands as FAAH Inhibitors | 1-gen-2020 | Brunetti, Leonardo; Carrieri, Antonio; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio; Laghezza, Antonio | |
Deep Eutectic Solvents as Effective Reaction Media for the Synthesis of 2‐Hydroxyphenylbenzimidazole-based Scaffolds en Route to Donepezil‐Like Compounds | 1-gen-2020 | Piemontese, L.; Sergio, R.; Rinaldo, F.; Brunetti, L.; Perna, F. M.; Amelia Santos, M.; Capriati, V. | |
Bone-seeking matrix metalloproteinase inhibitors for the treatment of skeletal malignancy | 1-gen-2020 | Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Di Pizio, A.; Pochetti, G.; Montanari, R.; Capelli, D.; Tauro, M.; Loiodice, F.; Tortorella, P. | |
Combining fatty acid amide hydrolase (FAAH) inhibition with peroxisome proliferator-activated receptor (PPAR) activation: a new potential multi-target therapeutic strategy for the treatment of Alzheimer’s disease | 1-gen-2020 | Brunetti, Leonardo; Laghezza, Antonio; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca | |
A Review of Recent Patents (2016-2019) on Plant Food Supplements with Potential Application in the Treatment of Neurodegenerative and Metabolic Disorders | 1-gen-2020 | Leuci, Rosalba; Brunetti, Leonardo; Laghezza, Antonio; Tortorella, Paolo; Loiodice, Fulvio; Piemontese, Luca | |
DEVELOPMENT OF PHENOXYALKYLPIPERIDINES AS HIGH-AFFINITY SIGMA-1 (s1) RECEPTOR LIGANDS WITH POTENT ANTI-AMNESIC ACTIVITY | 1-gen-2021 | Laghezza, Antonio; Abatematteo, Francesca S.; Mosier, Philip D.; Niso, Mauro; Brunetti, Leonardo; Berardi, Francesco; Loiodice, Fulvio; Contino, Marialessandra; Delprat, Benjamin; Maurice, Tangui; Abate, Carmen | |
Derivatives of Tenuazonic Acid as Potential New Multi-Target Anti-Alzheimer’s Disease Agents | 1-gen-2021 | Poliseno, Viviana; Chaves, Sílvia; Brunetti, Leonardo; Loiodice, Fulvio; Carrieri, Antonio; Laghezza, Antonio; Tortorella, Paolo; Magalhães, João D.; Cardoso, Sandra M.; Santos, M. Amélia; Piemontese, Luca | |
Natural Compounds for the Prevention and Treatment of Cardiovascular and Neurodegenerative Diseases | 1-gen-2021 | Leuci, Rosalba; Brunetti, Leonardo; Poliseno, Viviana; Laghezza, Antonio; Loiodice, Fulvio; Tortorella, Paolo; Piemontese, Luca | |
(2-Aminobenzothiazole)-Methyl-1,1-bisphosphonic acids: Targeting matrix metalloproteinase 13 inhibition to the bone | 1-gen-2021 | Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Loiodice, F.; Tortorella, P. | |
Multiple causes, multiple targets: FAAH as a centerpiece for therapy of multifactorial pathologies. | 1-gen-2021 | Brunetti, Leonardo; Leuci, Rosalba; Carrieri, Antonio; Laghezza, Antonio; Catto, Marco; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio | |
Multi-Target Approach for the Design of New Compounds Potentially Useful for the Prevention and Treatment of Cardiovascular and/or Neurodegenerative Diseases | 1-gen-2021 | Leuci, R.; Brunetti, L.; Carocci, A.; Carrieri, A.; Catto, M.; Laghezza, A.; Tortorella, P.; Piemontese, L.; Loiodice, F. | |
Novel Rivastigmine-Based Multitarget Hybrids For Potential Treatment of Alzheimer’s Disease: Cu(II) And Fe(III) Chelation Studies | 1-gen-2022 | Vicente-Zurdo, David; Brunetti, Leonardo; Piemontese, Luca; Madrid, Yolanda; Chaves, Sílvia; Amélia Santos., M. | |
Novel rivastigmine structure-based hybrids for the potential treatment of Alzheimer’s disease | 1-gen-2022 | Leuci, R.; Brunetti, L.; Carrieri, A.; Catto, M.; Laghezza, A.; Tortorella, P.; Loiodice, F.; Piemontese, L. | |
1,3,5-triazine derivatives as dual inhibitors of 5-HT6R/FAAH in search of new therapy for Alzheimer's disease | 1-gen-2022 | Czarnota-Łydka, Kinga; Satała, Grzegorz; Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; DE CANDIA, Modesto; Purgatorio, Rosa; Gumułka, Magdalena; Kucwaj-Brysz, Katarzyna; Carrieri, Antonio; Handzlik, Jadwiga |
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