Sfoglia per Autore LACIVITA, ENZA
trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogs of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines
2001-01-01 Perrone, R; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, Enza; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R.
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands
2002-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands
2002-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; DE GIORGIO, P.; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
Synthesis and Structure-affinity relationship of 1-[omega-(4-Aryl-1-piperazinyl)alkyl]-1-arylketones as 5-HT7 Receptor Ligands
2003-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Leopoldo, Marcello; Tortorella, V.
Studies on 1-arylpiperazine derivatives with affinity for rat 5-HT7 and 5-HT1A receptors
2004-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent
2004-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides as 5-HT7 receptor agents
2005-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter(SERT)and 5-HT1A receptors
2005-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Larizza, C.; Leopoldo, Marcello; Tortorella, V.
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors
2005-01-01 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
First structure–activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure
2005-01-01 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto
Synthesis and Biological Evaluation of Potential Positron Emission Tomography (PET) Ligands for Brain Visualization of Dopamine D3 Receptors.
2005-01-01 Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands
2005-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Synthesis and binding profile of constrained analogs of N-4-(4-ARYLPIPERAZIN-1-YL)BUTYL 3-METHOXYBENZAMIDES, a class of potential dopamine D3 receptor ligands
2006-01-01 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto
Design synthesis, and binding affinity of potential positron emission tomography (PET) ligands for visualitation of brain dopamine D3 receptors
2006-01-01 Leopoldo, Marcello; Lacivita, Enza; DE GIORGIO, P; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Selective Agents for Serotonin2C (5-HT2C) Receptor
2006-01-01 Lacivita, Enza; Leopoldo, Marcello
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands
2006-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Recent advances in the field of 5-HT7 receptor agents with 1-arylpiperazine structure.
2006-01-01 Leopoldo, Marcello; Lacivita, Enza; De Giorgio, P; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors
2006-01-01 Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
Design and synthesis of arylpiperazine-based fluorescent ligands for serotonin 5-HT1A and dopamine D3 receptors.
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogs of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines | 1-gen-2001 | Perrone, R; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, Enza; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R. | |
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands | 1-gen-2002 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V. | |
Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands | 1-gen-2002 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; DE GIORGIO, P.; Lacivita, Enza; Perrone, Roberto; Tortorella, V. | |
Synthesis and Structure-affinity relationship of 1-[omega-(4-Aryl-1-piperazinyl)alkyl]-1-arylketones as 5-HT7 Receptor Ligands | 1-gen-2003 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Leopoldo, Marcello; Tortorella, V. | |
Studies on 1-arylpiperazine derivatives with affinity for rat 5-HT7 and 5-HT1A receptors | 1-gen-2004 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Perrone, Roberto; Tortorella, V. | |
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent | 1-gen-2004 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V. | |
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides as 5-HT7 receptor agents | 1-gen-2005 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V. | |
Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter(SERT)and 5-HT1A receptors | 1-gen-2005 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Larizza, C.; Leopoldo, Marcello; Tortorella, V. | |
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors | 1-gen-2005 | Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto | |
First structure–activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure | 1-gen-2005 | Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto | |
Synthesis and Biological Evaluation of Potential Positron Emission Tomography (PET) Ligands for Brain Visualization of Dopamine D3 Receptors. | 1-gen-2005 | Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V. | |
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands | 1-gen-2005 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V. | |
Synthesis and binding profile of constrained analogs of N-4-(4-ARYLPIPERAZIN-1-YL)BUTYL 3-METHOXYBENZAMIDES, a class of potential dopamine D3 receptor ligands | 1-gen-2006 | Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto | |
Design synthesis, and binding affinity of potential positron emission tomography (PET) ligands for visualitation of brain dopamine D3 receptors | 1-gen-2006 | Leopoldo, Marcello; Lacivita, Enza; DE GIORGIO, P; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
Selective Agents for Serotonin2C (5-HT2C) Receptor | 1-gen-2006 | Lacivita, Enza; Leopoldo, Marcello | |
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands | 1-gen-2006 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V. | |
Recent advances in the field of 5-HT7 receptor agents with 1-arylpiperazine structure. | 1-gen-2006 | Leopoldo, Marcello; Lacivita, Enza; De Giorgio, P; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors | 1-gen-2006 | Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V. | |
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization | 1-gen-2007 | Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R. | |
Design and synthesis of arylpiperazine-based fluorescent ligands for serotonin 5-HT1A and dopamine D3 receptors. | 1-gen-2007 | Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R. |
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