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Design of multiple-target anticancer agents: a daunting challenge for the medicinal chemist
2009-01-01 Carotti, A; Leonetti, Francesco; Catto, Marco; Stefanachi, Angela; Nicolotti, Orazio
Dihydroquinazolinebenzylamides as Acetylcholinesterase and Butyrylcholinesterase inhibitors.
2016-01-01 Onnis, V.; Balboni, G.; Deplano, A.; Demurtas, M.; Buyn, J. S.; Sohn, J. M.; Jae Yeol Lee, J. Y.; Catto, Marco; Pisani, Leonardo; Carotti, A.
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity
2009-01-01 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
Hybrid inhibitors of Monoamine Oxidase B and Cholinesterases from a “designing in” chemical decoration of coumarin-based hit compounds
2015-01-01 Pisani, L.; Farina, R.; Catto, M.; Nicolotti, O.; Soto-Otero, R.; Denora, N.; Altomare, C. D.; Carotti, A.
Improved Fluorimetric Method for a Medium-Throughput Screening of Inhibitors of Beta-amyloid Aggregation: Application to Glycopeptide antibiotics and Quinone Derivatives
2006-01-01 Catto, Marco; Cellamare, Saverio; Chiti, F; Carotti, A.
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications
2007-01-01 Campagna, F; Cellamare, Saverio; Stefanachi, Angela; Stolfa, Ad; Basile, T; Ferappi, M; Catto, Marco; Carotti, A.
New small molecules and scaffolds inhibiting the β-amyloid aggregation
2007-01-01 Convertino, M; Pellarin, R; Catto, Marco; Carotti, A; Caflisch, A.
olid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues.
2005-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, A; Carotti, A. S.
Quinolizidinyl derivatives as potent inhibitors of acetyl- and butyryl-cholinesterase (AChE and BChE) of potential interest for the treatment of Alzheimer’s disease
2010-01-01 Tasso, B; Novelli, F; Catto, Marco; Tonelli, M; Sparatore, A; Nicolotti, Orazio; Boido, V; Sparatore, F; Carotti, A.
Quinolizidinyl derivatives of bi- and tricyclic systems as AChE/BChE and beta-amyloid aggregation inhibitors
2011-01-01 Tasso, B; Novelli, F; Catto, Marco; Nicolotti, Orazio; Tonelli, M; Vettoretti, G; Boido, V; Sparatore, F; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design of multiple-target anticancer agents: a daunting challenge for the medicinal chemist | 1-gen-2009 | Carotti, A; Leonetti, Francesco; Catto, Marco; Stefanachi, Angela; Nicolotti, Orazio | |
Dihydroquinazolinebenzylamides as Acetylcholinesterase and Butyrylcholinesterase inhibitors. | 1-gen-2016 | Onnis, V.; Balboni, G.; Deplano, A.; Demurtas, M.; Buyn, J. S.; Sohn, J. M.; Jae Yeol Lee, J. Y.; Catto, Marco; Pisani, Leonardo; Carotti, A. | |
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity | 1-gen-2009 | Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A. | |
Hybrid inhibitors of Monoamine Oxidase B and Cholinesterases from a “designing in” chemical decoration of coumarin-based hit compounds | 1-gen-2015 | Pisani, L.; Farina, R.; Catto, M.; Nicolotti, O.; Soto-Otero, R.; Denora, N.; Altomare, C. D.; Carotti, A. | |
Improved Fluorimetric Method for a Medium-Throughput Screening of Inhibitors of Beta-amyloid Aggregation: Application to Glycopeptide antibiotics and Quinone Derivatives | 1-gen-2006 | Catto, Marco; Cellamare, Saverio; Chiti, F; Carotti, A. | |
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications | 1-gen-2007 | Campagna, F; Cellamare, Saverio; Stefanachi, Angela; Stolfa, Ad; Basile, T; Ferappi, M; Catto, Marco; Carotti, A. | |
New small molecules and scaffolds inhibiting the β-amyloid aggregation | 1-gen-2007 | Convertino, M; Pellarin, R; Catto, Marco; Carotti, A; Caflisch, A. | |
olid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues. | 1-gen-2005 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, A; Carotti, A. S. | |
Quinolizidinyl derivatives as potent inhibitors of acetyl- and butyryl-cholinesterase (AChE and BChE) of potential interest for the treatment of Alzheimer’s disease | 1-gen-2010 | Tasso, B; Novelli, F; Catto, Marco; Tonelli, M; Sparatore, A; Nicolotti, Orazio; Boido, V; Sparatore, F; Carotti, A. | |
Quinolizidinyl derivatives of bi- and tricyclic systems as AChE/BChE and beta-amyloid aggregation inhibitors | 1-gen-2011 | Tasso, B; Novelli, F; Catto, Marco; Nicolotti, Orazio; Tonelli, M; Vettoretti, G; Boido, V; Sparatore, F; Carotti, Angelo |
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Opzioni
Scopri
Tipologia
- 4 Contributo in Atti di Convegno ... 31
- 4 Contributo in Atti di Convegno ... 31
Data di pubblicazione
- 2010 - 2019 14
- 2000 - 2009 16
- 1997 - 1999 1
Keyword
- beta Amyloid 2
- NON PREVISTO 2
- acetylcholinesterases 1
- Alzheimer's disease 1
- Arylhydrazones 1
- beta-amyloid 1
- Dantrolene 1
- fibrill 1
- Indoles 1
- inhibitor 1
Lingua
- eng 4
Accesso al fulltext
- no fulltext 30
- reserved 1