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Synthesis and binding profile of constrained analogs of N-4-(4-ARYLPIPERAZIN-1-YL)BUTYL 3-METHOXYBENZAMIDES, a class of potential dopamine D3 receptor ligands
2006-01-01 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto
Synthesis and Biological Evaluation of (Hetero)Arylmethyloxy- and Arylmethylamine-phenyl Derivatives as Potent P-gp Modulating Agents
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A.
Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT 1A receptor agonists for CNS disorders and neuropathic pain
2018-01-01 Franchini, S.; Bencheva, L. I.; Battisti, U. M.; Tait, A.; Sorbi, C.; Fossa, P.; Cichero, E.; Ronsisvalle, S.; Arico, G.; Denora, N.; Iacobazzi, R. M.; Cilia, A.; Pirona, L.; Brasili, L.
Synthesis and biological evaluation of 2-heteroarylthioalkanoic acid analogues of clofibric acid as peroxisome proliferator-activated receptor alpha agonists
2009-01-01 Giampietro, L; Ammazzalorso, A; Giancristofaro, A; Lannutti, F; Bettoni, G; DE FILIPPIS, B; Fantacuzzi, M; Maccallini, C; Petruzzelli, M; Morgano, A; Moschetta, Antonio; Amoroso, R.
Synthesis and Biological Evaluation of 2-Mercapto-1,3-benzothiazole Derivatives with Potential Antimicrobial Activity
2009-01-01 Franchini, Carlo; Muraglia, M; Corbo, Filomena Faustina Rina; Florio, M. A.; DI MOLA, A; Rosato, Antonio; Matucci, R; Nesi, M; VAN BAMBEKE, F; Vitali, C.
Synthesis and biological evaluation of 3,5-diaryl-pyrazole derivatives as potential antiprostate cancer agents
2021-01-01 Anil, D.; Caykoylu, E. U.; Sanli, F.; Gambacorta, N.; Karatas, O. F.; Nicolotti, O.; Algul, O.; Burmaoglu, S.
Synthesis and biological evaluation of 3-alkyloxazolidin-2-ones as reversible MAO inhibitors
2004-01-01 Lamanna, C; Sinicropi, M. S.; Pietrangeli, P; Corbo, Filomena Faustina Rina; Franchini, Carlo; Mondovi', B; Perrone, MARIA GRAZIA; Scilimati, Antonio
Synthesis and Biological Evaluation of a Valinomycin Analog Bearing a Pentafluorophenyl Active Ester Moiety
2015-01-01 D'Accolti, Lucia; Denora, Nunzio; LA PIANA, Gianluigi; Marzulli, Domenico; Siwy, Zuzanna S.; Fusco, Caterina; Annese, Cosimo
Synthesis and biological evaluation of chiral alfa-aminoanilides with central antinociceptive activity
2007-01-01 Corbo, Filomena Faustina Rina; Franchini, Carlo; Lentini, Giovanni; Muraglia, M; Ghelardini, C; Matucci, R; Galeotti, ; N., VIVOLI E; Tortorella, V.
Synthesis and Biological Evaluation of Chiral α-Aminoanilides with Central Antinociceptive Activity
2007-01-01 Corbo, Filomena; Franchini, Carlo; Lentini, Giovanni; Muraglia, Marilena; Ghelardini, Carla; Matucci, Rosanna; Galeotti, Nicoletta; Vivoli, Elisa; Tortorella, Vincenzo
Synthesis and Biological Evaluation of Dantrolene-Like Hydrazide and Hydrazone Analogues as Multitarget Agents for Neurodegenerative Diseases
2021-01-01 Bolognino, I.; Giangregorio, N.; Tonazzi, A.; Martinez, A. L.; Altomare, C. D.; Loza, M. I.; Sablone, S.; Cellamare, S.; Catto, M.
Synthesis and Biological Evaluation of Direct Thrombin Inhibitors Bearing 4-(Piperidin-1-yl)pyridine at the P1 Position with Potent Anticoagulant Activity
2013-01-01 DE CANDIA, Modesto; Fiorella, F.; Lopopolo, G.; Carotti, Angelo; Romano, M. R.; Logramo, M. D.; Martel, S.; Carrupt, P. A.; Belviso, B. D.; Caliandro, R.; Altomare, Cosimo Damiano
Synthesis and Biological Evaluation of Enantiomerically Pure (R)- and (S)-[18F]OF-NB1 for Imaging the GluN2B Subunit-Containing NMDA Receptors
2023-01-01 Korff, Marvin; Chaudhary, Ahmad; Li, Yinlong; Zhou, Xin; Zhao, Chunyu; Rong, Jian; Chen, Jiahui; Xiao, Zhiwei; Elghazawy, Nehal H.; Sippl, Wolfgang; Davenport, April T.; Daunais, James B.; Wang, Lu; Abate, Carmen; Ahmed, Hazem; Crowe, Ron; Schmidt, Thomas J.; Liang, Steven H.; Ametamey, Simon M.; Wünsch, Bernhard; Haider, Ahmed
Synthesis and biological evaluation of N-biphenyl-nicotinic based moiety compounds: A new class of antimitotic agents for the treatment of Hodgkin Lymphoma
2019-01-01 Porcelli, L.; Stolfa, D.; Stefanachi, A.; Di Fonte, R.; Garofoli, M.; Iacobazzi, R. M.; Silvestris, N.; Guarini, A.; Cellamare, S.; Azzariti, A.
Synthesis and Biological Evaluation of New Clofibrate Analogues as Potential PPARa Agonists
2005-01-01 Perrone, MARIA GRAZIA; Santandrea, E; Delluomo, N; Giannessi, F; Milazzo, F. M.; Sciarroni, A. F.; Scilimati, Antonio; Tortorella, V.
Synthesis and Biological Evaluation of Novel Hybrid Molecules Containing Purine, Coumarin and Isoxazoline or Isoxazole Moieties
2017-01-01 Kallitsakis, Michael G.; Carotti, Angelo; Catto, Marco; Peperidou, Aikaterini; Hadjipavlou-Litina, Dimitra J.; Litinas, Konstantinos E.
Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors
2006-01-01 Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V.
Synthesis and biological evaluation of pyrazoles and pyrazole-containing polycyclic derivatives as new ligands of central and peripheral benzodiazepine receptors
2004-01-01 Campagna, Francesco; Palluotto, F.; Carotti, Angelo; Maciocco, E.
Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents
2020-01-01 Tilekar, Kalpana; Upadhyay, Neha; Meyer‐almes, Franz‐josef; Loiodice, Fulvio; Anisimova, Natalia Y.; Spirina, Tatiana S.; Sokolova, Darina V.; Smirnova, Galina B.; Choe, Jun‐yong; Pokrovsky, Vadim S.; Lavecchia, Antonio; Ramaa, C. S.
Synthesis and Biological Properties of Coumarin Derivatives. A Review
2021-01-01 Bouhaoui, Abderrazzak; Eddahmi, Mohammed; Dib, Mustapha; Khouili, Mostafa; Aires, Alfredo; Catto, Marco; Bouissane, Latifa
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Synthesis and binding profile of constrained analogs of N-4-(4-ARYLPIPERAZIN-1-YL)BUTYL 3-METHOXYBENZAMIDES, a class of potential dopamine D3 receptor ligands | 1-gen-2006 | Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto | |
| Synthesis and Biological Evaluation of (Hetero)Arylmethyloxy- and Arylmethylamine-phenyl Derivatives as Potent P-gp Modulating Agents | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R; Rapposelli, S; Digiacomo, M; Vanni, M; Balsamo, A. | |
| Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT 1A receptor agonists for CNS disorders and neuropathic pain | 1-gen-2018 | Franchini, S.; Bencheva, L. I.; Battisti, U. M.; Tait, A.; Sorbi, C.; Fossa, P.; Cichero, E.; Ronsisvalle, S.; Arico, G.; Denora, N.; Iacobazzi, R. M.; Cilia, A.; Pirona, L.; Brasili, L. | |
| Synthesis and biological evaluation of 2-heteroarylthioalkanoic acid analogues of clofibric acid as peroxisome proliferator-activated receptor alpha agonists | 1-gen-2009 | Giampietro, L; Ammazzalorso, A; Giancristofaro, A; Lannutti, F; Bettoni, G; DE FILIPPIS, B; Fantacuzzi, M; Maccallini, C; Petruzzelli, M; Morgano, A; Moschetta, Antonio; Amoroso, R. | |
| Synthesis and Biological Evaluation of 2-Mercapto-1,3-benzothiazole Derivatives with Potential Antimicrobial Activity | 1-gen-2009 | Franchini, Carlo; Muraglia, M; Corbo, Filomena Faustina Rina; Florio, M. A.; DI MOLA, A; Rosato, Antonio; Matucci, R; Nesi, M; VAN BAMBEKE, F; Vitali, C. | |
| Synthesis and biological evaluation of 3,5-diaryl-pyrazole derivatives as potential antiprostate cancer agents | 1-gen-2021 | Anil, D.; Caykoylu, E. U.; Sanli, F.; Gambacorta, N.; Karatas, O. F.; Nicolotti, O.; Algul, O.; Burmaoglu, S. | |
| Synthesis and biological evaluation of 3-alkyloxazolidin-2-ones as reversible MAO inhibitors | 1-gen-2004 | Lamanna, C; Sinicropi, M. S.; Pietrangeli, P; Corbo, Filomena Faustina Rina; Franchini, Carlo; Mondovi', B; Perrone, MARIA GRAZIA; Scilimati, Antonio | |
| Synthesis and Biological Evaluation of a Valinomycin Analog Bearing a Pentafluorophenyl Active Ester Moiety | 1-gen-2015 | D'Accolti, Lucia; Denora, Nunzio; LA PIANA, Gianluigi; Marzulli, Domenico; Siwy, Zuzanna S.; Fusco, Caterina; Annese, Cosimo | |
| Synthesis and biological evaluation of chiral alfa-aminoanilides with central antinociceptive activity | 1-gen-2007 | Corbo, Filomena Faustina Rina; Franchini, Carlo; Lentini, Giovanni; Muraglia, M; Ghelardini, C; Matucci, R; Galeotti, ; N., VIVOLI E; Tortorella, V. | |
| Synthesis and Biological Evaluation of Chiral α-Aminoanilides with Central Antinociceptive Activity | 1-gen-2007 | Corbo, Filomena; Franchini, Carlo; Lentini, Giovanni; Muraglia, Marilena; Ghelardini, Carla; Matucci, Rosanna; Galeotti, Nicoletta; Vivoli, Elisa; Tortorella, Vincenzo | |
| Synthesis and Biological Evaluation of Dantrolene-Like Hydrazide and Hydrazone Analogues as Multitarget Agents for Neurodegenerative Diseases | 1-gen-2021 | Bolognino, I.; Giangregorio, N.; Tonazzi, A.; Martinez, A. L.; Altomare, C. D.; Loza, M. I.; Sablone, S.; Cellamare, S.; Catto, M. | |
| Synthesis and Biological Evaluation of Direct Thrombin Inhibitors Bearing 4-(Piperidin-1-yl)pyridine at the P1 Position with Potent Anticoagulant Activity | 1-gen-2013 | DE CANDIA, Modesto; Fiorella, F.; Lopopolo, G.; Carotti, Angelo; Romano, M. R.; Logramo, M. D.; Martel, S.; Carrupt, P. A.; Belviso, B. D.; Caliandro, R.; Altomare, Cosimo Damiano | |
| Synthesis and Biological Evaluation of Enantiomerically Pure (R)- and (S)-[18F]OF-NB1 for Imaging the GluN2B Subunit-Containing NMDA Receptors | 1-gen-2023 | Korff, Marvin; Chaudhary, Ahmad; Li, Yinlong; Zhou, Xin; Zhao, Chunyu; Rong, Jian; Chen, Jiahui; Xiao, Zhiwei; Elghazawy, Nehal H.; Sippl, Wolfgang; Davenport, April T.; Daunais, James B.; Wang, Lu; Abate, Carmen; Ahmed, Hazem; Crowe, Ron; Schmidt, Thomas J.; Liang, Steven H.; Ametamey, Simon M.; Wünsch, Bernhard; Haider, Ahmed | |
| Synthesis and biological evaluation of N-biphenyl-nicotinic based moiety compounds: A new class of antimitotic agents for the treatment of Hodgkin Lymphoma | 1-gen-2019 | Porcelli, L.; Stolfa, D.; Stefanachi, A.; Di Fonte, R.; Garofoli, M.; Iacobazzi, R. M.; Silvestris, N.; Guarini, A.; Cellamare, S.; Azzariti, A. | |
| Synthesis and Biological Evaluation of New Clofibrate Analogues as Potential PPARa Agonists | 1-gen-2005 | Perrone, MARIA GRAZIA; Santandrea, E; Delluomo, N; Giannessi, F; Milazzo, F. M.; Sciarroni, A. F.; Scilimati, Antonio; Tortorella, V. | |
| Synthesis and Biological Evaluation of Novel Hybrid Molecules Containing Purine, Coumarin and Isoxazoline or Isoxazole Moieties | 1-gen-2017 | Kallitsakis, Michael G.; Carotti, Angelo; Catto, Marco; Peperidou, Aikaterini; Hadjipavlou-Litina, Dimitra J.; Litinas, Konstantinos E. | |
| Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors | 1-gen-2006 | Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V. | |
| Synthesis and biological evaluation of pyrazoles and pyrazole-containing polycyclic derivatives as new ligands of central and peripheral benzodiazepine receptors | 1-gen-2004 | Campagna, Francesco; Palluotto, F.; Carotti, Angelo; Maciocco, E. | |
| Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents | 1-gen-2020 | Tilekar, Kalpana; Upadhyay, Neha; Meyer‐almes, Franz‐josef; Loiodice, Fulvio; Anisimova, Natalia Y.; Spirina, Tatiana S.; Sokolova, Darina V.; Smirnova, Galina B.; Choe, Jun‐yong; Pokrovsky, Vadim S.; Lavecchia, Antonio; Ramaa, C. S. | |
| Synthesis and Biological Properties of Coumarin Derivatives. A Review | 1-gen-2021 | Bouhaoui, Abderrazzak; Eddahmi, Mohammed; Dib, Mustapha; Khouili, Mostafa; Aires, Alfredo; Catto, Marco; Bouissane, Latifa |
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