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NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
Structure-Activity Relationship Studies on 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline Derivatives as Multidrug Resistance Reversers.
2017-01-01 Teodori, E; Dei, S; Bartolucci, G; Perrone, MARIA GRAZIA; Manetti, D; Romanelli, Mn; Contino, Marialessandra; Colabufo, Nicola Antonio
Structure-Activity Relationship Studies on Tetrahydroisoquinoline Derivatives: [4′-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl)biphenyl-4-ol] (MC70) Conjugated through Flexible Alkyl Chains with Furazan Moieties Gives Rise to Potent and Selective Ligands of P-glycoprotein
2016-01-01 Guglielmo, Stefano; Lazzarato, Loretta; Contino, Marialessandra; Perrone, MARIA GRAZIA; Chegaev, Konstantin; Carrieri, Antonio; Fruttero, Roberta; Colabufo, Nicola Antonio; Gasco, Alberto
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent
2004-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. 2
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto
Structure-activity relationship study towards non-peptidic positron emission tomography (PET) radiotracer for gastrin releasing peptide receptors: Development of [18F] (S)-3-(1H-indol-3-yl)-N-[1-[5-(2-fluoroethoxy)pyridin-2-yl]cyclohexylmethyl]-2-methyl-2-[3-(4-nitrophenyl)ureido]propionamide.
2017-01-01 Lacivita, Enza; Lucente, Ermelinda; Kwizera, C; Antunes, If; Niso, Mauro; DE GIORGIO, Paola; Perrone, Roberto; Colabufo, Nicola Antonio; Elsinga, Ph; Leopoldo, Marcello
Structure-activity relationships and effects on neuroactive steroid synthesis in a series of 2-phenylimidazo[1,2-alpha]pyridineacetamide peripheral benzodiazepine receptors ligands
2005-01-01 Trapani, Giuseppe; Laquintana, Valentino; Denora, Nunzio; Trapani, Adriana; Lopedota, Angela Assunta; Latrofa, A.; Franco, Massimo; Serra, M.; Pisu, M. G.; Floris, I.; Sanna, E.; Biggio, G.; Liso, G.
Structure-activity relationships and effects on neuroactive steroids in a series of 2-phenylimidazo[1,2-a]pyridineacetamide peripheral benzodiazepine receptors ligands
2005-01-01 Trapani, G.; Laquintana, V.; Denora, N.; Trapani, A.; Lopedota, A.; Latrofa, A.; Franco, M.; Serra, M.; Pisu, M. G.; Floris, I.; Sanna, E.; Biggio, G.; Liso, G.
Structure-Activity Relationships and Therapeutic Potential of Purinergic P2X7 Receptor Antagonists
2024-01-01 GHAFIR EL IDRISSI, Imane; Podlewska, Sabina; Abate, Carmen; J Bojarski, Andrzej; Lacivita, Enza; Leopoldo, Marcello
Structure-Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update
2018-01-01 Modica, Maria N; Lacivita, Enza; Intagliata, Sebastiano; Salerno, Loredana; Romeo, Giuseppe; Pittalà, Valeria; Leopoldo, Marcello
Structure-activity relationships in 1,4-benzodioxan-related compounds. 10. Novel α1-adrenoreceptor antagonists related to openphendioxan: synthesis, biological evaluation, and α1d computational study
2010-01-01 Carrieri, Antonio; Piergentili, A; DEL BELLO, F; Giannella, M; Pigini, M; Leonardi, A; Fanelli, F; Quaglia, W.
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes
2002-01-01 Quaglia, W.; Pigini, M.; Piergentili, A.; Giannella, M.; Gentili, F.; Marucci, G.; Carrieri, Antonio; Carotti, Angelo; Poggesi, E.; Leonardi, A.; Melchiorre, C.
Structure-activity relationships in 1,4-benzodioxan-related compounds. 9. From 1,4-benzodioxane to 1,4-dioxane ring as a promising template of novel alpha1D-adrenoreceptor antagonists, 5-HT1A full agonists, and cytotoxic agents
2008-01-01 Quaglia, W; Piergentili, A; DEL BELLO, F; Farande, Y; Giannella, M; Pigini, M; Rafaiani, G; Carrieri, Antonio; Amantini, C; Lucciarini, R; Santoni, G; Poggesi, E; Leonardi, A.
Structure-activity relationships in 1,4-benzodioxan-related Compounds. Role of the phenyl substituent at position 4 on the selectivity for alfa1–adrenoreceptor subtypes
2002-01-01 W., Quaglia; M., Pigini; A., Piergentili; M., Giannella; F., Gentili; G., Marucci; Carrieri, Antonio; A., Carotti; E., Poggesi; A., Leonardi; C., Melchiorre
Structure-activity relationships in tocainide analogues
2003-01-01 Muraglia, M; Catalano, Alessia; Corbo, Filomena Faustina Rina; Franchini, C; Scilimati, Antonio; Tortorella, V; DE LUCA, A; CONTE CAMERINO, D.
Structure-activity relationships of 2-aryl-2,5-dihydropyridazino [4,3-b]indol-3(3H)-ones at the benzodiazepine receptor.
1996-01-01 Palluotto, F; Carotti, Angelo; Casini, G; Campagna, F; Genchi, G; Rizzo, M; De Sarro, Gb
Structure-activity relationships of antitumor thiazolo[3,4-a]benzimidazole derivatives
1994-01-01 Chimirri, A; Grasso, S; Monforte, A. M.; Monforte, P; Zappala', M; Carotti, Angelo
Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands
2002-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; DE GIORGIO, P.; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
Structure-affinity relationships of some alkoxycarbonyl-2H- or -4H-pyrimido[2,1-b]benzothiazol-2- or 4-one benzodiazepine receptor ligands
1993-01-01 Trapani, Giuseppe; Carotti, Angelo; Franco, Massimo; Latrofa, A.; Genchi, G.; Liso, G.
Structure-Antimicrobial Activity Relationships of Quaternary Ammonium Derivatives of Perhydropyrrolo[3,4-c] pyridine
1992-01-01 Altomare, Cosimo Damiano; Carotti, Angelo; Casini, G; Cellamare, Saverio; Ferappi, M; Vitali, C.
Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases
2015-01-01 Farina, Roberta; Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Gadaleta, Domenico; Denora, Nunzio; Soto Otero, R; Mendez Alvarez, E; Passos, Cs; Muncipinto, Giovanni; Altomare, Cosimo Damiano; Nurisso, A; Carrupt, Pa; Carotti, Angelo
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- 1 Contributo su Rivista 82162
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