FRANCAVILLA, FABIO
FRANCAVILLA, FABIO
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
Allosteric Modulators of Serotonin Receptors: A Medicinal Chemistry Survey
2024-01-01 Brunetti, Leonardo; Francavilla, Fabio; Leopoldo, Marcello; Lacivita, Enza
Conformational Restriction of Designer Drugs Reveals Subtype-Selective and Biased CB2Agonists with Neuroprotective Effects
2025-01-01 Gioé-Gallo, Claudia; Ortigueira, Sandra; Prieto-Díaz, Rubén; Contino, Marialessandra; Azuaje, Jhonny; Perrone, Maria Grazia; Riganti, Chiara; Alberga, Domenico; Felice Mangiatordi, Giuseppe; Andújar-Arias, Antonio; García-Rey, Aitor; Graziano, Giovanni; Stefanachi, Angela; Val, Cristina; Leandro Martínez, Antón; Biel Rebassa, Joan; Reza, David; Selas, Asier; Francavilla, Fabio; Rita Paleo, M.; García-Mera, Xerardo; Isabel Loza, M.; Navarro, Gemma; Brea, José; Sotelo, Eddy
Design, Synthesis, and Biological Evaluation of Novel Heteroaryl, Squaramide, and Indolcarboxamide Derivatives as Formyl Peptide Receptor 2 Agonists to Target Neuroinflammation
2025-01-01 Francavilla, Fabio; Vitone, Daniele; Schepetkin, Igor A; Kirpotina, Lilya N; Carrieri, Antonio; Brunetti, Leonardo; Ghafir El Idrissi, Imane; Perrone, Maria Grazia; Frydrych, Jakub Kosma; Trojan, Ewa; Quinn, Mark T; Basta-Kaim, Agnieszka; Lacivita, Enza; Leopoldo, Marcello
Development of potent isoflavone-based formyl peptide receptor 1 (FPR1) antagonists and their effects in gastric cancer cell models
2023-01-01 Francavilla, Fabio; Sarcina, Federica; Schepetkin, Igor A.; Kirpotina, Lilya N.; Contino, Marialessandra; Schirizzi, Annalisa; De Leonardis, Giampiero; Khlebnikov, Andrei I.; D'Alessandro, Rosalba; Quinn, Mark T.; Lacivita, Enza; Leopoldo, Marcello
FPR2 and brimstone: a novel approach for the treatment of neuroinflammation
2024-01-01 Brunetti, L.; Francavilla, F.; Schepetkin, I. A.; Kirpotina, L. N.; Quinn, M. T.; Leopoldo, M.; Lacivita, E.
Hydrogen Sulfide (H2S)-Donating Formyl Peptide Receptor 2 (FPR2) Agonists: Design, Synthesis, and Biological Evaluation in Primary Mouse Microglia Culture
2025-01-01 Brunetti, Leonardo; Francavilla, Fabio; Niso, Mauro; Frydrych, Jakub Kosma; Trojan, Ewa; Schepetkin, Igor A; Kirpotina, Liliya N; Grygier, Beata; Łukowicz, Krzysztof; Quinn, Mark T; Basta-Kaim, Agnieszka; Lacivita, Enza; Leopoldo, Marcello
Inflammaging and Immunosenescence in the Post‐COVID Era: Small Molecules, Big Challenges
2024-01-01 Francavilla, Fabio; Intranuovo, Francesca; La Spada, Gabriella; Lacivita, Enza; Catto, Marco; Graps, Elisabetta Anna; Altomare, Cosimo Damiano
Multiple approaches for developing novel FPR2 Agonists with Pro-Resolving, Anti-Inflammatory, and Antioxidant Properties: Bioisosteres of ureidopropanamide-based agonists, H2S-Releasing Moieties grafting, and Multicomponent Reaction strategies
2025-03-05 Francavilla, Fabio
Stimulation of Formyl Peptide Receptor-2 by the New Agonist CMC23 Protects against Endotoxin-Induced Neuroinflammatory Response: A Study in Organotypic Hippocampal Cultures
2023-01-01 Tylek, K.; Trojan, E.; Leskiewicz, M.; Francavilla, F.; Lacivita, E.; Leopoldo, M.; Basta-Kaim, A.
Tackling neuroinflammation with H2S releasing FPR2 agonists
2024-01-01 Brunetti, Leonardo; Francavilla, Fabio; Schepetkin, Igor A.; Kirpotina, Liliya N.; Trojan, Ewa; Quinn, Mark T.; Basta-Kaim, Agnieszka; Leopoldo, Marcello; Lacivita, Enza
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Allosteric Modulators of Serotonin Receptors: A Medicinal Chemistry Survey | 1-gen-2024 | Brunetti, Leonardo; Francavilla, Fabio; Leopoldo, Marcello; Lacivita, Enza | |
| Conformational Restriction of Designer Drugs Reveals Subtype-Selective and Biased CB2Agonists with Neuroprotective Effects | 1-gen-2025 | Gioé-Gallo, Claudia; Ortigueira, Sandra; Prieto-Díaz, Rubén; Contino, Marialessandra; Azuaje, Jhonny; Perrone, Maria Grazia; Riganti, Chiara; Alberga, Domenico; Felice Mangiatordi, Giuseppe; Andújar-Arias, Antonio; García-Rey, Aitor; Graziano, Giovanni; Stefanachi, Angela; Val, Cristina; Leandro Martínez, Antón; Biel Rebassa, Joan; Reza, David; Selas, Asier; Francavilla, Fabio; Rita Paleo, M.; García-Mera, Xerardo; Isabel Loza, M.; Navarro, Gemma; Brea, José; Sotelo, Eddy | |
| Design, Synthesis, and Biological Evaluation of Novel Heteroaryl, Squaramide, and Indolcarboxamide Derivatives as Formyl Peptide Receptor 2 Agonists to Target Neuroinflammation | 1-gen-2025 | Francavilla, Fabio; Vitone, Daniele; Schepetkin, Igor A; Kirpotina, Lilya N; Carrieri, Antonio; Brunetti, Leonardo; Ghafir El Idrissi, Imane; Perrone, Maria Grazia; Frydrych, Jakub Kosma; Trojan, Ewa; Quinn, Mark T; Basta-Kaim, Agnieszka; Lacivita, Enza; Leopoldo, Marcello | |
| Development of potent isoflavone-based formyl peptide receptor 1 (FPR1) antagonists and their effects in gastric cancer cell models | 1-gen-2023 | Francavilla, Fabio; Sarcina, Federica; Schepetkin, Igor A.; Kirpotina, Lilya N.; Contino, Marialessandra; Schirizzi, Annalisa; De Leonardis, Giampiero; Khlebnikov, Andrei I.; D'Alessandro, Rosalba; Quinn, Mark T.; Lacivita, Enza; Leopoldo, Marcello | |
| FPR2 and brimstone: a novel approach for the treatment of neuroinflammation | 1-gen-2024 | Brunetti, L.; Francavilla, F.; Schepetkin, I. A.; Kirpotina, L. N.; Quinn, M. T.; Leopoldo, M.; Lacivita, E. | |
| Hydrogen Sulfide (H2S)-Donating Formyl Peptide Receptor 2 (FPR2) Agonists: Design, Synthesis, and Biological Evaluation in Primary Mouse Microglia Culture | 1-gen-2025 | Brunetti, Leonardo; Francavilla, Fabio; Niso, Mauro; Frydrych, Jakub Kosma; Trojan, Ewa; Schepetkin, Igor A; Kirpotina, Liliya N; Grygier, Beata; Łukowicz, Krzysztof; Quinn, Mark T; Basta-Kaim, Agnieszka; Lacivita, Enza; Leopoldo, Marcello | |
| Inflammaging and Immunosenescence in the Post‐COVID Era: Small Molecules, Big Challenges | 1-gen-2024 | Francavilla, Fabio; Intranuovo, Francesca; La Spada, Gabriella; Lacivita, Enza; Catto, Marco; Graps, Elisabetta Anna; Altomare, Cosimo Damiano | |
| Multiple approaches for developing novel FPR2 Agonists with Pro-Resolving, Anti-Inflammatory, and Antioxidant Properties: Bioisosteres of ureidopropanamide-based agonists, H2S-Releasing Moieties grafting, and Multicomponent Reaction strategies | 5-mar-2025 | Francavilla, Fabio | |
| Stimulation of Formyl Peptide Receptor-2 by the New Agonist CMC23 Protects against Endotoxin-Induced Neuroinflammatory Response: A Study in Organotypic Hippocampal Cultures | 1-gen-2023 | Tylek, K.; Trojan, E.; Leskiewicz, M.; Francavilla, F.; Lacivita, E.; Leopoldo, M.; Basta-Kaim, A. | |
| Tackling neuroinflammation with H2S releasing FPR2 agonists | 1-gen-2024 | Brunetti, Leonardo; Francavilla, Fabio; Schepetkin, Igor A.; Kirpotina, Liliya N.; Trojan, Ewa; Quinn, Mark T.; Basta-Kaim, Agnieszka; Leopoldo, Marcello; Lacivita, Enza |