CONTINO, MARIALESSANDRA
CONTINO, MARIALESSANDRA
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Delta8─Delta7 sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activity
2011-01-01 Abate, CARMEN rosa; Niso, Mauro; Contino, Marialessandra; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto; Berardi, Francesco
4-(Tetralin-1-yl)- and 4-(Naphthalen-1-yl)alkyl Derivatives of 1-Cycloheylpiperazine as sigma receptor Ligands with Agonist sigma 2 Activity
2004-01-01 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, N. C.; Contino, Marialessandra; Perrone, Roberto; Tortorella, V.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes
2015-01-01 Schininà, B; Martorana, A; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Perrone, MARIA GRAZIA; de Guidi, G; Catalfo, A; Rappazzo, G; Zuccarello, E; Prezzavento, O; Amata, E; Rescifina, A; Marrazzo, A.
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers
2020-01-01 Braconi, Laura; Bartolucci, Gianluca; Contino, Marialessandra; Chiaramonte, Niccolò; Giampietro, Roberta; Manetti, Dina; Perrone, Maria Grazia; Romanelli, Maria Novella; Colabufo, Nicola Antonio; Riganti, Chiara; Dei, Silvia; Teodori, Elisabetta
A Benzopyrane Derivative as a P-Glycoprotein Stimulator: A Potential Agent to Decrease β-Amyloid Accumulation in Alzheimer's Disease
2012-01-01 Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A.
A Benzopyrane derivative as P-glycoprotein stimulator: a potential agent to decrease beta-amyloid accumulation in Alzheimer’s disease
2012-01-01 Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A.
A new generation of MDR modulating agents with dual activity: P-gp inhibitor and iNOS inducer agents
2011-01-01 Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto; Panaro, Maria Antonietta; Cianciulli, Antonia; Mitolo, V.; Azzariti, A.; Quatrale, A.; Paradiso, A.
A new method for evaluating sigma(2) ligand activity in the isolated guinea-pig bladder
2003-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Perrone, Roberto; Tortorella, Vincenzo
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression
2016-01-01 Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, MARIA GRAZIA; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio
ABC pumps and their role in active drug transport
2009-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Niso, M; Perrone, Roberto; Contino, Marialessandra
ABC transporters in CSCs membranes as a novel target for treating tumor relapse
2014-01-01 Zinzi, Laura; Contino, Marialessandra; Cantore, Mariangela; Capparelli, Elena; Leopoldo, Marcello; Colabufo, Nicola Antonio
Activity-lipophilicity relationship studies on P-gp ligands designed as simplified tariquidar bulky fragments
2013-01-01 Contino, Marialessandra; Zinzi, Laura; Cantore, Mariangela; Perrone, Maria Grazia; Leopoldo, Marcello; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio
ALPACA: A machine Learning Platform for Affinity and selectivity profiling of CAnnabinoids receptors modulators
2023-01-01 Delre, Pietro; Contino, Marialessandra; Alberga, Domenico; Saviano, Michele; Corriero, Nicola; Mangiatordi, Giuseppe Felice
An innovative small molecule for promoting neuroreparative strategies
2018-01-01 Colabufo, Nicola Antonio; Contino, Marialessandra; Cantore, Mariangela; Berardi, Francesco; Perrone, Roberto; Tonazzi, Annamaria; Console, Lara; Panaro, Maria Antonietta; Savolainen, Heli; Luurtsema, Gert
An updated patent review on P-glycoprotein inhibitors (2011-2018)
2019-01-01 Leopoldo, M; Nardulli, P; Contino, M; Leonetti, F; Gert, Luurtsema; Colabufo, Na
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines
2004-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V.
Arylamides hybrids of two high-affinity sigma-2 receptor ligands as tools for the development of PET radiotracers
2011-01-01 Abate, CARMEN rosa; Ferorelli, Savina; Contino, Marialessandra; Marottoli, R; Colabufo, Nicola Antonio; Perrone, Roberto; Berardi, Francesco
Arylamino Esters As P-Glycoprotein Modulators: SAR Studies to Establish Requirements for Potency and Selectivity
2015-01-01 Teodori, Elisabetta; Dei, Silvia; Floriddia, Elisa; Perrone, MARIA GRAZIA; Manetti, Dina; Romanelli, Maria Novella; Contino, Marialessandra; Colabufo, Nicola Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and human Delta8─Delta7 sterol isomerase ligands with antiproliferative and P-glycoprotein inhibitory activity | 1-gen-2011 | Abate, CARMEN rosa; Niso, Mauro; Contino, Marialessandra; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto; Berardi, Francesco | |
4-(Tetralin-1-yl)- and 4-(Naphthalen-1-yl)alkyl Derivatives of 1-Cycloheylpiperazine as sigma receptor Ligands with Agonist sigma 2 Activity | 1-gen-2004 | Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, N. C.; Contino, Marialessandra; Perrone, Roberto; Tortorella, V. | |
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization | 1-gen-2007 | Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R. | |
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo | |
4-Nitro-2,1,3-benzoxadiazole derivatives as potential fluorescent sigma receptor probes | 1-gen-2015 | Schininà, B; Martorana, A; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Perrone, MARIA GRAZIA; de Guidi, G; Catalfo, A; Rappazzo, G; Zuccarello, E; Prezzavento, O; Amata, E; Rescifina, A; Marrazzo, A. | |
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers | 1-gen-2020 | Braconi, Laura; Bartolucci, Gianluca; Contino, Marialessandra; Chiaramonte, Niccolò; Giampietro, Roberta; Manetti, Dina; Perrone, Maria Grazia; Romanelli, Maria Novella; Colabufo, Nicola Antonio; Riganti, Chiara; Dei, Silvia; Teodori, Elisabetta | |
A Benzopyrane Derivative as a P-Glycoprotein Stimulator: A Potential Agent to Decrease β-Amyloid Accumulation in Alzheimer's Disease | 1-gen-2012 | Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A. | |
A Benzopyrane derivative as P-glycoprotein stimulator: a potential agent to decrease beta-amyloid accumulation in Alzheimer’s disease | 1-gen-2012 | Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A. | |
A new generation of MDR modulating agents with dual activity: P-gp inhibitor and iNOS inducer agents | 1-gen-2011 | Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto; Panaro, Maria Antonietta; Cianciulli, Antonia; Mitolo, V.; Azzariti, A.; Quatrale, A.; Paradiso, A. | |
A new method for evaluating sigma(2) ligand activity in the isolated guinea-pig bladder | 1-gen-2003 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Perrone, Roberto; Tortorella, Vincenzo | |
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression | 1-gen-2016 | Guglielmo, Stefano; Contino, Marialessandra; Lazzarato, Loretta; Perrone, MARIA GRAZIA; Blangetti, Marco; Fruttero, Roberta; Colabufo, Nicola Antonio | |
ABC pumps and their role in active drug transport | 1-gen-2009 | Colabufo, Nicola Antonio; Berardi, Francesco; Niso, M; Perrone, Roberto; Contino, Marialessandra | |
ABC transporters in CSCs membranes as a novel target for treating tumor relapse | 1-gen-2014 | Zinzi, Laura; Contino, Marialessandra; Cantore, Mariangela; Capparelli, Elena; Leopoldo, Marcello; Colabufo, Nicola Antonio | |
Activity-lipophilicity relationship studies on P-gp ligands designed as simplified tariquidar bulky fragments | 1-gen-2013 | Contino, Marialessandra; Zinzi, Laura; Cantore, Mariangela; Perrone, Maria Grazia; Leopoldo, Marcello; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio | |
ALPACA: A machine Learning Platform for Affinity and selectivity profiling of CAnnabinoids receptors modulators | 1-gen-2023 | Delre, Pietro; Contino, Marialessandra; Alberga, Domenico; Saviano, Michele; Corriero, Nicola; Mangiatordi, Giuseppe Felice | |
An innovative small molecule for promoting neuroreparative strategies | 1-gen-2018 | Colabufo, Nicola Antonio; Contino, Marialessandra; Cantore, Mariangela; Berardi, Francesco; Perrone, Roberto; Tonazzi, Annamaria; Console, Lara; Panaro, Maria Antonietta; Savolainen, Heli; Luurtsema, Gert | |
An updated patent review on P-glycoprotein inhibitors (2011-2018) | 1-gen-2019 | Leopoldo, M; Nardulli, P; Contino, M; Leonetti, F; Gert, Luurtsema; Colabufo, Na | |
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines | 1-gen-2004 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V. | |
Arylamides hybrids of two high-affinity sigma-2 receptor ligands as tools for the development of PET radiotracers | 1-gen-2011 | Abate, CARMEN rosa; Ferorelli, Savina; Contino, Marialessandra; Marottoli, R; Colabufo, Nicola Antonio; Perrone, Roberto; Berardi, Francesco | |
Arylamino Esters As P-Glycoprotein Modulators: SAR Studies to Establish Requirements for Potency and Selectivity | 1-gen-2015 | Teodori, Elisabetta; Dei, Silvia; Floriddia, Elisa; Perrone, MARIA GRAZIA; Manetti, Dina; Romanelli, Maria Novella; Contino, Marialessandra; Colabufo, Nicola Antonio |