LEONETTI, Francesco

LEONETTI, Francesco  

DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO  

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Titolo Data di pubblicazione Autore(i) File
(EN) GALLOYL BENZAMIDE-BASED COMPOUNDS AS JNK MODULATORS (FR) COMPOSES A BASE DE GALLOYL BENZAMIDE UTILISES EN TANT QUE MODULATEURS DE JNK 1-gen-2014 Cellamare, Saverio; Carotti, Angelo; Stefanachi, Angela; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Tardia, Piero; Introcaso, Antonellina; Valentina, Leo; Addabbo, Francesco; Montagnani, Monica; Nacci, Carmela
1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships 1-gen-2008 Stefanachi, Angela; Nicolotti, Orazio; Leonetti, Francesco; Cellamare, Saverio; Campagna, Francesco; Loza, Mi; Brea, Jm; Mazza, F; Gavuzzo, E; Carotti, Angelo
2-D and 3-D modeling of imadazoline receptor ligands: insights into pharmacophore 1-gen-1997 Carrieri, Antonio; L., Brasili; Leonetti, Francesco; M., Pigini; M., Giannella; P., Bousquet; Carotti, Angelo
4-(Alkylamino)methyl-substituted coumarins as potent and selective AChE and MAO-B dual inhibitors with a therapeutic potential in neurodegenerative disorders 1-gen-2013 Pisani, L.; Catto, M.; Stefanachi, A.; Leonetti, F.; Campagna, F.; Nicolotti, O.; Soto-Otero, R.; Carotti, A.
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor. 1-gen-2010 Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A.
A Multi-Objective Optimization Algorithm for Molecular Design 1-gen-2009 Giangreco, I; Nicolotti, Orazio; Miscioscia, T. F.; Convertino, M; Mangiatordi, G. F.; Siragusa, L; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
A multitarget approach in cancer research 1-gen-2009 Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A.
A multitarget approach in cancer research. Joint Meeting on Medicinal Chemistry 1-gen-2009 Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A.
A New Approach for Drug Target and Bioactivity Prediction: The Multifingerprint Similarity Search Algorithm (MuSSeL) 1-gen-2019 Alberga, Domenico; Trisciuzzi, Daniela; Montaruli, Michele; Leonetti, Francesco; Mangiatordi, Giuseppe Felice; Nicolotti, Orazio
A new approach to combine ligand- and structure-based drug design. 1-gen-2008 Nicolotti, Orazio; Miscioscia, Tf; Carotti, A; Leonetti, Francesco; Giangreco, I; Carotti, A.
A novel function for non-deterministic scouting of optimal QSAR models out of a highly-structured physicochemical space. 1-gen-2006 Nicolotti, Orazio; Miscioscia, T. F.; Leonetti, Francesco; Carotti, A.
A twenty-year journey exploring coumarin-based derivatives as bioactive molecules 1-gen-2022 Pisani, Leonardo; Catto, Marco; Muncipinto, Giovanni; Nicolotti, Orazio; Carrieri, Antonio; Rullo, Mariagrazia; Stefanachi, Angela; Leonetti, Francesco; Altomare, Cosimo
An improved method for the biological evaluation of polyphenol derivatives as potential inhibitors of aβ(1–40) aggregation 1-gen-2009 Stolfa, A; Cellamare, Saverio; Stefanachi, Angela; Catto, Marco; Leonetti, Francesco; Nicolotti, Orazio; Carotti, A.
An integrated approach to ligand- and structure-based drug design: development and application to a series of serine protease inhibitors 1-gen-2008 Nicolotti, Orazio; Miscioscia, Tf; Carotti, Angelo; Leonetti, Francesco; Carotti, A.
An integrated methodology to interface structure- and ligand-based drug design 1-gen-2008 Giangreco, I; Nicolotti, Orazio; Miscioscia, Tf; Tedeschi, P; Carotti, A; Leonetti, Francesco; Carotti, A.
An updated patent review on P-glycoprotein inhibitors (2011-2018) 1-gen-2019 Leopoldo, M; Nardulli, P; Contino, M; Leonetti, F; Gert, Luurtsema; Colabufo, Na
Attenuation of autoimmune disease in fas-deficient mice by treatment with a cytotoxic benzodiazepine 1-gen-2003 Bednarski, J. J.; Warner, R. E.; Rao, T.; Leonetti, Francesco; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A.; OPIPARI JR, A. W.; Glick, G. D.
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitors 1-gen-2018 Mangiatordi, G. F.; Trisciuzzi, D.; Iacobazzi, R.; Denora, N.; Pisani, L.; Catto, M.; Leonetti, F.; Alberga, D.; Nicolotti, O.
BCR-ABL inhibitors in chronic myeloid leukemia: process chemistry and biochemical profile 1-gen-2011 Leonetti, Francesco; Stefanachi, Angela; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Cellamare, Saverio; Carotti, Angelo
Bcr-abl tyrosine kinase inhibitors in the treatment of pediatric cml 1-gen-2020 Carofiglio, F.; Lopalco, A.; Lopedota, A.; Cutrignelli, A.; Nicolotti, O.; Denora, N.; Stefanachi, A.; Leonetti, F.