LEOPOLDO, Marcello
LEOPOLDO, Marcello
DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO
1-(2-Methoxyphenyl)-4-alkylpiperazines: effect of the N-4 substituent on the affinity and selectivity for dopamine D4 receptor
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Aryl-4-[(1-tetralinyl)alkyl]piperazines: alkylamido and alkylamino derivatives. Synthesis, 5-HT1A receptor affinity, and selectivity. 3
1996-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V; Fornaretto, Mg; Caccia, C; Mcarthur, Ra
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors
2005-01-01 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
2-(Aryloxy)ethylamine derivatives: ring opened congeners of long chain 1-arylpiperazines with high 5-HT1A receptor affinity and selectivity versus D2 and a1 receptors
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
3-(1H-Indol-3-yl)-2-[3-(4-nitrophenyl)ureido]propanamide Derivatives are Agonists of Human Formyl Peptide Receptor 2
2011-01-01 Kirpotina, Ln; Schepetkin, Ia; Leopoldo, Marcello; Quinn, Mt
3-(1H-indol-3-yl)-2-[3-(4-nitrophenyl)ureido]propanamide enantiomers with human formyl-peptide receptor agonist activity: Molecular modeling of chiral recognition by FPR2.
2013-01-01 Schepetkin, Ia; Kirpotina, Ln; Khlebnikov, Ai; Leopoldo, Marcello; Lucente, E; Lacivita, Enza; De Giorgio, P; Quinn, M. T.
4-[omega-[4-arylpiperazin-1-yl]phenyl)imidazo[1,2-a]pyridine derivatives: fluorescent high-affinity dopamine D3 receptor ligands as potential probes for receptor visualization
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
4-[omega-Tetralin-1-yl]-1-benzylpiperazines and related compounds as 5-HT1A/D-2 ligands
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lograno, M.; Tortorella, V.
5 HT1A receptor, an old target for new therapeutic agents
2008-01-01 Lacivita, Enza; Leopoldo, Marcello; Berardi, Francesco; Perrone, R.
5-HT and DA receptor affinity of arylpiperazine derivatives with terminal benzamide fragment
1994-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V.; Lograno, Marcello Diego; Daniele, E.; Govoni, S.
5-HT1A and D-2 receptor affinity of o-methoxyphenyl derivatives with terminal benzamide fragment on N-4 alkyl chain. 2
1995-01-01 Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Tortorella, V; Lograno, Marcello Diego; Daniele, E; Govoni, S.
5-HT3 and 5-HT4 receptor affinities of naphtho[1,2-d]thiazole derivatives with various basic side chains
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
5-HT7 receptor activation: procognitive and antiamnesic effects
2015-01-01 Meneses, A; Perez Garcia, G; Liy Salmeron, G; Ponce López, T; Lacivita, Enza; Leopoldo, Marcello
5-HT7 receptor modulators: a medicinal chemistry survey of recent patent literature (2004 - 2009)
2010-01-01 Leopoldo, Marcello; Lacivita, Enza; Berardi, Francesco; Perrone, Roberto
5-HT7 Receptors Regulate Excitatory-Inhibitory Balance in Mouse Spinal Cord Dorsal Horn
2022-01-01 Comitato, Antonella; Lacivita, Enza; Leopoldo, Marcello; Bardoni, Rita
A Benzopyrane Derivative as a P-Glycoprotein Stimulator: A Potential Agent to Decrease β-Amyloid Accumulation in Alzheimer's Disease
2012-01-01 Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A.
A Benzopyrane derivative as P-glycoprotein stimulator: a potential agent to decrease beta-amyloid accumulation in Alzheimer’s disease
2012-01-01 Contino, M.; Cantore, M.; Capparelli, E.; Perrone, M. G.; Niso, M.; Inglese, C.; Berardi, F.; Leopoldo, M.; Perrone, R.; Colabufo, N. A.
A conformational rearrangement of the SARS-CoV-2 host protein sigma-1 is required for antiviral activity: insights from a combined in-silico/in-vitro approach
2023-01-01 Abatematteo, Francesca Serena; Delre, Pietro; Mercurio, Ivan; Rezelj, Veronica V; Siliqi, Dritan; Beaucourt, Stephanie; Lattanzi, Gianluca; Colabufo, Nicola Antonio; Leopoldo, Marcello; Saviano, Michele; Vignuzzi, Marco; Mangiatordi, Giuseppe Felice; Abate, Carmen