PIEMONTESE, LUCA

PIEMONTESE, LUCA  

DIPARTIMENTO DI FARMACIA-SCIENZE DEL FARMACO  

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(2-Aminobenzothiazole)-Methyl-1,1-bisphosphonic acids: Targeting matrix metalloproteinase 13 inhibition to the bone 1-gen-2021 Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Loiodice, F.; Tortorella, P.
(contributo in convegno) MOLECULAR DETERMINANTS FOR NUCLEAR RECEPTORS SELECTIVITY; CHEMOMETRIC ANALYSIS, DOCKINGS AND SITE-DIRECTED MUTAGENESIS OF DUAL PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS α/γ AGONISTS 1-gen-2013 Carrieri, Antonio; Marco, Giudici; Mariagiovanna, Parente; Mario De, Rosas; Piemontese, Luca; Fracchiolla, Giuseppe; Laghezza, Antonio; Tortorella, Paolo; Carbonara, Giuseppe Gerardo; Antonio, Lavecchia; Federica, Gilardi; Maurizio, Crestani; Fulvio, Loiodice
1,3,5-triazine derivatives as dual inhibitors of 5-HT6R/FAAH in search of new therapy for Alzheimer's disease 1-gen-2022 Czarnota-Łydka, Kinga; Satała, Grzegorz; Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; DE CANDIA, Modesto; Purgatorio, Rosa; Gumułka, Magdalena; Kucwaj-Brysz, Katarzyna; Carrieri, Antonio; Handzlik, Jadwiga
A Chemoinformatics Search for Peroxisome Proliferator-Activated Receptors Ligands Revealed a New Pan-Agonist Able to Reduce Lipid Accumulation and Improve Insulin Sensitivity 1-gen-2022 Sblano, S.; Cerchia, C.; Laghezza, A.; Piemontese, L.; Brunetti, L.; Leuci, R.; Gilardi, F.; Thomas, A.; Genovese, M.; Santi, A.; Tortorella, P.; Paoli, P.; Lavecchia, A.; Loiodice, F.
A NEW ANTIDIABETIC AGENT SHOWING PPARα/γ DUAL AGONISM AND MITOCHONDRIAL PYRUVATE CARRIER INHIBITION 1-gen-2023 Cerchia, C.; Laghezza, A.; Genovese, M.; Leuci, R.; Pranzini, E.; Santi, A.; Brunetti, L.; Piemontese, L.; Tortorella, P.; Biswas, A.; Singh, R. P.; Tambe, S.; Ca, S.; Pattnaik, A. K.; Jayaprakash, V.; Paoli, P.; Loiodice, F.; Lavecchia, A.
A New Antidiabetic Agent Showing Short- and Long-Term Effects Due to Peroxisome Proliferator-Activated Receptor Alpha/Gamma Dual Agonism and Mitochondrial Pyruvate Carrier Inhibition 1-gen-2023 Laghezza, Antonio; Cerchia, Carmen; Genovese, Massimo; Leuci, Rosalba; Pranzini, Erica; Santi, Alice; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Biswas, Abanish; Pratap Singh, Ravi; Tambe, Suhas; Ca, Sudeep; Kumar Pattnaik, Ashok; Jayaprakash, Venkatesan; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio
A New Series of Aryloxyacetic Acids Endowed with Multi-Target Activity towards Peroxisome Proliferator-Activated Receptors (PPARs), Fatty Acid Amide Hydrolase (FAAH), and Acetylcholinesterase (AChE) 1-gen-2022 Leuci, R.; Brunetti, L.; Laghezza, A.; Piemontese, L.; Carrieri, A.; Pisani, L.; Tortorella, P.; Catto, M.; Loiodice, F.
A Review of Recent Patents (2016-2019) on Plant Food Supplements with Potential Application in the Treatment of Neurodegenerative and Metabolic Disorders 1-gen-2020 Leuci, Rosalba; Brunetti, Leonardo; Laghezza, Antonio; Tortorella, Paolo; Loiodice, Fulvio; Piemontese, Luca
AGONISTI DEI RECETTORI NUCLEARI PPARs COME POTENZIALI NUOVI AGENTI TERAPEUTICI PER IL TRATTAMENTO DELLA SINDROME METABOLICA. 1-gen-2010 Piemontese, Luca; Mariagiovanna, Parente; Fracchiolla, Giuseppe; Laghezza, Antonio; Carbonara, Giuseppe Gerardo; Tortorella, Paolo; Loiodice, Fulvio
An efficient synthesis of the optically active isomers of 2H-1,4-benzoxazine derivatives, novel KATP channel modulators 1-gen-2013 Piemontese, Luca; Laghezza, Antonio; Fracchiolla, Giuseppe; Carbonara, Giuseppe Gerardo; Tortorella, Paolo; Loiodice, Fulvio
An innovative approach for the treatment of Alzheimer’s disease: the role of peroxisome proliferator-activated receptors and their ligands in development of alternative therapeutic interventions 1-gen-2019 Piemontese, Luca
An update about the crucial role of stereochemistry on the effects of Peroxisome Proliferator-Activated Receptor ligands 1-gen-2019 Laghezza, Antonio; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio
Aspergillus carbonarius proteases and their possible activity in Ochratoxin A degradation 1-gen-2017 Gallo, Antonia; Ferrara, Massimo; Bleve, Gianluca; Cervini, Carla; Piemontese, Luca; Epifani, Filomena; Logrieco, Antonio F; Solfrizzo, Michele; Perrone, Giancarlo
Beyond the Canonical Endocannabinoid System. A Screening of PPAR Ligands as FAAH Inhibitors 1-gen-2020 Brunetti, Leonardo; Carrieri, Antonio; Piemontese, Luca; Tortorella, Paolo; Loiodice, Fulvio; Laghezza, Antonio
Bone-seeking matrix metalloproteinase inhibitors for the treatment of skeletal malignancy 1-gen-2020 Laghezza, A.; Piemontese, L.; Brunetti, L.; Caradonna, A.; Agamennone, M.; Di Pizio, A.; Pochetti, G.; Montanari, R.; Capelli, D.; Tauro, M.; Loiodice, F.; Tortorella, P.
Can foods influence the onset and progress of neurodegenerative diseases? 1-gen-2022 Piemontese, Luca; Brunetti, Leonardo; Leuci, Rosalba
Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity 1-gen-2016 Tauro, Marilena; Laghezza, Antonio; Loiodice, Fulvio; Piemontese, Luca; Caradonna, Alessia; Capelli, Davide; Montanari, Roberta; Pochetti, Giorgio; Di Pizio, Antonella; Agamennone, Mariangela; Campestre, Cristina; Tortorella, Paolo
ChemInform Abstract: Convenient Synthesis of Some 3-Phenyl-1-benzofuran-2-carboxylic Acid Derivatives as New Potential Inhibitors of CLC-Kb Channels. 1-gen-2011 Piemontese, Luca; Carbonara, Giuseppe Gerardo; Fracchiolla, Giuseppe; Laghezza, Antonio; Paolo Tortorella andFulvio Loiodice,
Chiral phenoxyacetic acid analogues inhibit colon cancer cell proliferation acting as PPARγ partial agonists 1-gen-2019 Sabatino, Lina; Ziccardi, Pamela; Cerchia, Carmen; Muccillo, Livio; Piemontese, Luca; Loiodice, Fulvio; Colantuoni, Vittorio; Lupo, Angelo; Lavecchia, Antonio
Climate change effect on ochratoxin A production and gene expression in Aspergillus carbonarius 1-gen-2018 Perrone, G; Gallo, A; Piemontese, L; Magistà, D; Solfrizzo, M; Cervini, C