Sfoglia per Autore
Structure-activity relationships of piperazine-2-one derivatives as novel human ClpP activators
2023-01-01 Armenise, D.; Baldelli, O. M.; Miciaccia, M.; Ferorelli, S.; Perrone, M. G.; Scilimati, A.
DIPG-27. Diffuse Intrinsic Pontine Glioma (DIPG) challenge: from gene expression profile to drug.
2023-01-01 Scilimati, Antonio; Armenise, Domenico; Baldelli, Olga; Centonze, Antonella; Derri, Davide; Ferorelli, Savina; Miciaccia, Morena; Solidoro, Roberta; Perrone, MARIA GRAZIA
Design and synthesis of new [4,5-b] and [4,5-c] imidazopyridines as potential fluorophores/inhibitors for Human Cyclooxygenase-1.
2023-01-01 Munzone, C.; Fortuna, C. G.; Bonaccorso, C.; Perrone, M. G.; Miciaccia, M.
Cyclooxygenase-1 Inhibition: A Promising Theragnostic Approach for Ovarian Cancer
2023-01-01 Miciaccia, Morena; Ferorelli, Savina; Centonze, Antonella; Solidoro, Roberta; Munzone, Cristina; Bonaccorso, Carmela; Gianluca Fortuna, Cosimo; Kleinmanns, Katrin; Bjørge, Line; Perrone, MARIA GRAZIA; Scilimati, Antonio
Human Caseinolytic Protease P (hClpP) Activity Modulating Agents For The Treatment Of DIPG/DMG
2023-01-01 Perrone, M. G.; Centonze, A.; Miciaccia, M.; Baldelli, O.; Cavallaro, G.; Ferorelli, S.; Fortuna, C.; Scilimati, A.
Harmaline-based scaffold as Human Caseinolytic Protease P (hClpP) inducers for Diffuse Intrinsic Pontine Glioma (DIPG) treatment
2023-01-01 Miciaccia, Morena; Centonze, Antonella; Baldelli, Olga; Solidoro, Roberta; Armenise, Domenico; Cavallaro, Gianfranco; Gianluca Fortuna, Cosimo; Ferorelli, Savina; Perrone, MARIA GRAZIA; Scilimati, Antonio
m-Terphenylamines, Acting as Selective COX-1 Inhibitors, Block Microglia Inflammatory Response and Exert Neuroprotective Activity
2023-01-01 Rocchi, Damiano; González, Juan F.; Martín-Cámara, Olmo; Perrone, MARIA GRAZIA; Miciaccia, Morena; Scilimati, Antonio; Decouty-Pérez, Celine; Parada, Esther; Egea, Javier; Carlos Menéndez, J.
A further pocket or conformational plasticity by mapping COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet behavior
2024-01-01 Solidoro, Roberta; Miciaccia, Morena; Bonaccorso, Carmela; Fortuna, Cosimo Gianluca; Armenise, Domenico; Centonze, Antonella; Ferorelli, Savina; Vitale, Paola; Rodrigues, Pryscila; Guimarães, Renilda; de Oliveira, Alana; da Paz, Mariana; Rangel, Luciana; Sathler, Plínio Cunha; Altomare, Angela; Perrone, Maria Grazia; Scilimati, Antonio
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment
2024-01-01 Miciaccia, Morena; Rizzo, Francesca; Centonze, Antonella; Cavallaro, Gianfranco; Contino, Marialessandra; Armenise, Domenico; Baldelli, OLGA MARIA; Solidoro, Roberta; Ferorelli, Savina; Scarcia, Pasquale; Agrimi, Gennaro; Zingales, Veronica; Cimetta, Elisa; Ronsisvalle, Simone; Maria Sipala, Federica; LOGUERCIO POLOSA, Paola Anna Maria; Gianluca Fortuna, Cosimo; Perrone, MARIA GRAZIA; Scilimati, Antonio
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment
2024-01-01 Miciaccia, M.; Rizzo, F.; Centonze, A.; Cavallaro, G.; Contino, M.; Armenise, D.; Baldelli, O. M.; Solidoro, R.; Ferorelli, S.; Scarcia, P.; Agrimi, G.; Zingales, V.; Cimetta, E.; Ronsisvalle, S.; Sipala, F. M.; Polosa, P. L.; Fortuna, C. G.; Perrone, M. G.; Scilimati, A.
Fluorescent imaging probes for in vivo ovarian cancer targeted detection and surgery
2024-01-01 Solidoro, Roberta; Centonze, Antonella; Miciaccia, Morena; Baldelli, Olga Maria; Armenise, Domenico; Ferorelli, Savina; Perrone, Maria Grazia; Scilimati, Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Structure-activity relationships of piperazine-2-one derivatives as novel human ClpP activators | 1-gen-2023 | Armenise, D.; Baldelli, O. M.; Miciaccia, M.; Ferorelli, S.; Perrone, M. G.; Scilimati, A. | |
DIPG-27. Diffuse Intrinsic Pontine Glioma (DIPG) challenge: from gene expression profile to drug. | 1-gen-2023 | Scilimati, Antonio; Armenise, Domenico; Baldelli, Olga; Centonze, Antonella; Derri, Davide; Ferorelli, Savina; Miciaccia, Morena; Solidoro, Roberta; Perrone, MARIA GRAZIA | |
Design and synthesis of new [4,5-b] and [4,5-c] imidazopyridines as potential fluorophores/inhibitors for Human Cyclooxygenase-1. | 1-gen-2023 | Munzone, C.; Fortuna, C. G.; Bonaccorso, C.; Perrone, M. G.; Miciaccia, M. | |
Cyclooxygenase-1 Inhibition: A Promising Theragnostic Approach for Ovarian Cancer | 1-gen-2023 | Miciaccia, Morena; Ferorelli, Savina; Centonze, Antonella; Solidoro, Roberta; Munzone, Cristina; Bonaccorso, Carmela; Gianluca Fortuna, Cosimo; Kleinmanns, Katrin; Bjørge, Line; Perrone, MARIA GRAZIA; Scilimati, Antonio | |
Human Caseinolytic Protease P (hClpP) Activity Modulating Agents For The Treatment Of DIPG/DMG | 1-gen-2023 | Perrone, M. G.; Centonze, A.; Miciaccia, M.; Baldelli, O.; Cavallaro, G.; Ferorelli, S.; Fortuna, C.; Scilimati, A. | |
Harmaline-based scaffold as Human Caseinolytic Protease P (hClpP) inducers for Diffuse Intrinsic Pontine Glioma (DIPG) treatment | 1-gen-2023 | Miciaccia, Morena; Centonze, Antonella; Baldelli, Olga; Solidoro, Roberta; Armenise, Domenico; Cavallaro, Gianfranco; Gianluca Fortuna, Cosimo; Ferorelli, Savina; Perrone, MARIA GRAZIA; Scilimati, Antonio | |
m-Terphenylamines, Acting as Selective COX-1 Inhibitors, Block Microglia Inflammatory Response and Exert Neuroprotective Activity | 1-gen-2023 | Rocchi, Damiano; González, Juan F.; Martín-Cámara, Olmo; Perrone, MARIA GRAZIA; Miciaccia, Morena; Scilimati, Antonio; Decouty-Pérez, Celine; Parada, Esther; Egea, Javier; Carlos Menéndez, J. | |
A further pocket or conformational plasticity by mapping COX-1 catalytic site through modified-mofezolac structure-inhibitory activity relationships and their antiplatelet behavior | 1-gen-2024 | Solidoro, Roberta; Miciaccia, Morena; Bonaccorso, Carmela; Fortuna, Cosimo Gianluca; Armenise, Domenico; Centonze, Antonella; Ferorelli, Savina; Vitale, Paola; Rodrigues, Pryscila; Guimarães, Renilda; de Oliveira, Alana; da Paz, Mariana; Rangel, Luciana; Sathler, Plínio Cunha; Altomare, Angela; Perrone, Maria Grazia; Scilimati, Antonio | |
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment | 1-gen-2024 | Miciaccia, Morena; Rizzo, Francesca; Centonze, Antonella; Cavallaro, Gianfranco; Contino, Marialessandra; Armenise, Domenico; Baldelli, OLGA MARIA; Solidoro, Roberta; Ferorelli, Savina; Scarcia, Pasquale; Agrimi, Gennaro; Zingales, Veronica; Cimetta, Elisa; Ronsisvalle, Simone; Maria Sipala, Federica; LOGUERCIO POLOSA, Paola Anna Maria; Gianluca Fortuna, Cosimo; Perrone, MARIA GRAZIA; Scilimati, Antonio | |
Harmaline to Human Mitochondrial Caseinolytic Serine Protease Activation for Pediatric Diffuse Intrinsic Pontine Glioma Treatment | 1-gen-2024 | Miciaccia, M.; Rizzo, F.; Centonze, A.; Cavallaro, G.; Contino, M.; Armenise, D.; Baldelli, O. M.; Solidoro, R.; Ferorelli, S.; Scarcia, P.; Agrimi, G.; Zingales, V.; Cimetta, E.; Ronsisvalle, S.; Sipala, F. M.; Polosa, P. L.; Fortuna, C. G.; Perrone, M. G.; Scilimati, A. | |
Fluorescent imaging probes for in vivo ovarian cancer targeted detection and surgery | 1-gen-2024 | Solidoro, Roberta; Centonze, Antonella; Miciaccia, Morena; Baldelli, Olga Maria; Armenise, Domenico; Ferorelli, Savina; Perrone, Maria Grazia; Scilimati, Antonio |
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