Sfoglia per Autore
Theoretical evidence of a salt bridge disruption as the initiating process for the alpha1d-adrenergic receptor activation: a molecular dynamics and docking study
2001-01-01 Carrieri, Antonio; Centeno, N. B.; Rodrigo, J.; Sanz, F.; Carotti, Angelo
High Affinity Central Benzodiazepine Receptor Ligands. Part 2: Quantitative Structure-Activity Relationships and Comparative Molecular Field Analysis of Pyrazolo[4,3-c]quinolin-3-ones
2001-01-01 Savini, L.; Chiasserini, L.; Pellerano, C.; Biggio, G.; Maciocco, E.; Serra, M.; Cinone, N.; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, A.
Neuronal Nicotinic Agonists: a Multi-approach Development of the Pharmacophore
2001-01-01 Nicolotti, Orazio; PELLEGRINI CALACE, M. L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Centeno, N. B.; Sanz, F.; Carotti, Angelo
Binding Models of Reversible Inhibitors to Monoamine Oxidases
2002-01-01 Carotti, A.; Barreca, M. L.; PELLEGRINI CALACE, M.; Carrieri, Antonio; Altomare, Cosimo Damiano
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes
2002-01-01 Quaglia, W.; Pigini, M.; Piergentili, A.; Giannella, M.; Gentili, F.; Marucci, G.; Carrieri, Antonio; Carotti, Angelo; Poggesi, E.; Leonardi, A.; Melchiorre, C.
Distant collaboration in drug discovery: The LINK3D project
2002-01-01 Pastor, M.; Benedetti, P.; Carotti, Angelo; Carrieri, Antonio; Diaz, C.; Herriz, C.; Hltje, H. D.; Loza, M. I.; Oprea, T.; Padn, F.; Pubill, F.; Sanz, F.
New antagonists at serotonin 5-HT2A, 5-HT2B and 5-HT2C receptors, synthesis, pharmacology, 3D-QSAR and molecular modelling of (aminoalkyl)benzo and heterocycloalkanones
2002-01-01 Brea, J.; Rodrigo, J.; Carrieri, Antonio; Sanz, F.; Cadavid, M. I.; Enguix, M. J.; Villazon, M.; Mengod, G.; Caro, Y.; Masaguer, C. F.; Ravina, E.; Centeno, N. B.; Carotti, Angelo; Loza, M. I.
Structure-activity relationships in 1,4-benzodioxan-related Compounds. Role of the phenyl substituent at position 4 on the selectivity for alfa1–adrenoreceptor subtypes
2002-01-01 W., Quaglia; M., Pigini; A., Piergentili; M., Giannella; F., Gentili; G., Marucci; Carrieri, Antonio; A., Carotti; E., Poggesi; A., Leonardi; C., Melchiorre
alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(Biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole
2002-01-01 F., Gentili; P., Bousquet; L., Brasili; M., Caretto; Carrieri, Antonio; M., Dontenwill; M., Giannella; G., Marucci; M., Perfumi; A., Piergentili; W., Quaglia; C., Rascente; M., Pigini
Natural and synthetic geiparvarins are strong and selective MAO-B inhibitors. Synthesis and SAR studies.
2002-01-01 Carotti, Angelo; Carrieri, Antonio; S., Chimichi; M., Boccalini; B., Cosimelli; C., Gnerre; A., Carotti
Ligands of neuronal nicotinic acetylcholine receptor (nAChR): inferences from the Hansch and 3-D Quantitative Structure-Activity Relationship (QSAR) models
2002-01-01 Nicolotti, Orazio; Pellegrini Calace, M; Altomare, Cosimo Damiano; Carotti, Angelo; Carrieri, Antonio; Sanz, F.
Binding models of reversible inhibitors to type-B monoamine oxidase
2002-01-01 Carrieri, Antonio; Carotti, Angelo; Barreca, Ml; Altomare, Cosimo Damiano
stant collaboration in drug discovery: The LINK3D project
2002-01-01 M., Pastor; P., Benedetti; A., Carotti; Carrieri, Antonio; C., Daz; C., Herriz; H. D., Hltje; M. I., Loza; T., Oprea; F., Padn; F., Pubill; F., Sanz; F., STOLL AND THE LINKD CONSORTIUM
Alpidem analogues containinig a GABA or glycine moiety as new anticonvulsant agents
2003-01-01 Trapani, Giuseppe; A., Latrofa; Franco, Massimo; Carrieri, Antonio; Cellamare, Saverio; M., Serra; E., Sanna; G., Biggio; G., Liso
Coumarin, chromone, and 4(3H)-pyrimidinone novel bicyclic and tricyclic derivatives as antiplatelet agents: synthesis, biological evaluation, and comparative molecular field analysis
2003-01-01 Roma, G.; DI BRACCIO, M.; Carrieri, Antonio; Grossi, G.; Leoncini, G.; Signorello, M. G.; Carotti, Angelo
Investigation on platelet aggregation inhibitory activity by phenyl amides and esters of piperidinecarboxylic acids
2003-01-01 DE CANDIA, Modesto; Summo, L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Nardecchia, A.; Cellamare, Saverio; Carotti, Angelo
Synthesis.and biological evaluation of pyridazino[4,3-b]indoles and indeno[1,2-c]pyridazines as new ligands of central and peripheral benzodiazepine receptors
2003-01-01 Campagna, Francesco; Palluotto, Fausta; Mascia, M. P.; Maciocco, E.; Marra, C.; Carotti, Angelo; Carrieri, Antonio
alfa2-adrenoreceptors profile modulation. 2.1 Biphenyline analogues as tools for selective activation of alfa2C-subtype
2004-01-01 F., Gentili; F., Ghelfi; M., Giannella; A., Piergentili; M., Pigini; W., Quaglia; C., Vesprini; P. A., Crassous; H., Paris; Carrieri, Antonio
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands
2004-01-01 Nicolotti, Orazio; Carotti, Angelo; Carrieri, Antonio; Pigini, M; Gentili, F; Brasili, L; Giannella, M; Quaglia, W; Piergentili, A; Bousquet, P; Dontenwill, M.
Rational design of the new antihypertensive I1-receptor ligand 2-(2-biphenyl-2-yl-1-methyl-ethyl-)4,5-dihydro-1H-imidazole
2005-01-01 F., Gentili; P., Bousquet; Carrieri, Antonio; J., Feldman; F., Ghelfi; M., Giannella; A., Piergentili; W., Quaglia; C., Vesprini; M., Pigin
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Theoretical evidence of a salt bridge disruption as the initiating process for the alpha1d-adrenergic receptor activation: a molecular dynamics and docking study | 1-gen-2001 | Carrieri, Antonio; Centeno, N. B.; Rodrigo, J.; Sanz, F.; Carotti, Angelo | |
High Affinity Central Benzodiazepine Receptor Ligands. Part 2: Quantitative Structure-Activity Relationships and Comparative Molecular Field Analysis of Pyrazolo[4,3-c]quinolin-3-ones | 1-gen-2001 | Savini, L.; Chiasserini, L.; Pellerano, C.; Biggio, G.; Maciocco, E.; Serra, M.; Cinone, N.; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, A. | |
Neuronal Nicotinic Agonists: a Multi-approach Development of the Pharmacophore | 1-gen-2001 | Nicolotti, Orazio; PELLEGRINI CALACE, M. L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Centeno, N. B.; Sanz, F.; Carotti, Angelo | |
Binding Models of Reversible Inhibitors to Monoamine Oxidases | 1-gen-2002 | Carotti, A.; Barreca, M. L.; PELLEGRINI CALACE, M.; Carrieri, Antonio; Altomare, Cosimo Damiano | |
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes | 1-gen-2002 | Quaglia, W.; Pigini, M.; Piergentili, A.; Giannella, M.; Gentili, F.; Marucci, G.; Carrieri, Antonio; Carotti, Angelo; Poggesi, E.; Leonardi, A.; Melchiorre, C. | |
Distant collaboration in drug discovery: The LINK3D project | 1-gen-2002 | Pastor, M.; Benedetti, P.; Carotti, Angelo; Carrieri, Antonio; Diaz, C.; Herriz, C.; Hltje, H. D.; Loza, M. I.; Oprea, T.; Padn, F.; Pubill, F.; Sanz, F. | |
New antagonists at serotonin 5-HT2A, 5-HT2B and 5-HT2C receptors, synthesis, pharmacology, 3D-QSAR and molecular modelling of (aminoalkyl)benzo and heterocycloalkanones | 1-gen-2002 | Brea, J.; Rodrigo, J.; Carrieri, Antonio; Sanz, F.; Cadavid, M. I.; Enguix, M. J.; Villazon, M.; Mengod, G.; Caro, Y.; Masaguer, C. F.; Ravina, E.; Centeno, N. B.; Carotti, Angelo; Loza, M. I. | |
Structure-activity relationships in 1,4-benzodioxan-related Compounds. Role of the phenyl substituent at position 4 on the selectivity for alfa1–adrenoreceptor subtypes | 1-gen-2002 | W., Quaglia; M., Pigini; A., Piergentili; M., Giannella; F., Gentili; G., Marucci; Carrieri, Antonio; A., Carotti; E., Poggesi; A., Leonardi; C., Melchiorre | |
alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(Biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole | 1-gen-2002 | F., Gentili; P., Bousquet; L., Brasili; M., Caretto; Carrieri, Antonio; M., Dontenwill; M., Giannella; G., Marucci; M., Perfumi; A., Piergentili; W., Quaglia; C., Rascente; M., Pigini | |
Natural and synthetic geiparvarins are strong and selective MAO-B inhibitors. Synthesis and SAR studies. | 1-gen-2002 | Carotti, Angelo; Carrieri, Antonio; S., Chimichi; M., Boccalini; B., Cosimelli; C., Gnerre; A., Carotti | |
Ligands of neuronal nicotinic acetylcholine receptor (nAChR): inferences from the Hansch and 3-D Quantitative Structure-Activity Relationship (QSAR) models | 1-gen-2002 | Nicolotti, Orazio; Pellegrini Calace, M; Altomare, Cosimo Damiano; Carotti, Angelo; Carrieri, Antonio; Sanz, F. | |
Binding models of reversible inhibitors to type-B monoamine oxidase | 1-gen-2002 | Carrieri, Antonio; Carotti, Angelo; Barreca, Ml; Altomare, Cosimo Damiano | |
stant collaboration in drug discovery: The LINK3D project | 1-gen-2002 | M., Pastor; P., Benedetti; A., Carotti; Carrieri, Antonio; C., Daz; C., Herriz; H. D., Hltje; M. I., Loza; T., Oprea; F., Padn; F., Pubill; F., Sanz; F., STOLL AND THE LINKD CONSORTIUM | |
Alpidem analogues containinig a GABA or glycine moiety as new anticonvulsant agents | 1-gen-2003 | Trapani, Giuseppe; A., Latrofa; Franco, Massimo; Carrieri, Antonio; Cellamare, Saverio; M., Serra; E., Sanna; G., Biggio; G., Liso | |
Coumarin, chromone, and 4(3H)-pyrimidinone novel bicyclic and tricyclic derivatives as antiplatelet agents: synthesis, biological evaluation, and comparative molecular field analysis | 1-gen-2003 | Roma, G.; DI BRACCIO, M.; Carrieri, Antonio; Grossi, G.; Leoncini, G.; Signorello, M. G.; Carotti, Angelo | |
Investigation on platelet aggregation inhibitory activity by phenyl amides and esters of piperidinecarboxylic acids | 1-gen-2003 | DE CANDIA, Modesto; Summo, L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Nardecchia, A.; Cellamare, Saverio; Carotti, Angelo | |
Synthesis.and biological evaluation of pyridazino[4,3-b]indoles and indeno[1,2-c]pyridazines as new ligands of central and peripheral benzodiazepine receptors | 1-gen-2003 | Campagna, Francesco; Palluotto, Fausta; Mascia, M. P.; Maciocco, E.; Marra, C.; Carotti, Angelo; Carrieri, Antonio | |
alfa2-adrenoreceptors profile modulation. 2.1 Biphenyline analogues as tools for selective activation of alfa2C-subtype | 1-gen-2004 | F., Gentili; F., Ghelfi; M., Giannella; A., Piergentili; M., Pigini; W., Quaglia; C., Vesprini; P. A., Crassous; H., Paris; Carrieri, Antonio | |
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands | 1-gen-2004 | Nicolotti, Orazio; Carotti, Angelo; Carrieri, Antonio; Pigini, M; Gentili, F; Brasili, L; Giannella, M; Quaglia, W; Piergentili, A; Bousquet, P; Dontenwill, M. | |
Rational design of the new antihypertensive I1-receptor ligand 2-(2-biphenyl-2-yl-1-methyl-ethyl-)4,5-dihydro-1H-imidazole | 1-gen-2005 | F., Gentili; P., Bousquet; Carrieri, Antonio; J., Feldman; F., Ghelfi; M., Giannella; A., Piergentili; W., Quaglia; C., Vesprini; M., Pigin |
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