Sfoglia per Autore
5-HT3 and 5-HT4 receptor affinities of naphtho[1,2-d]thiazole derivatives with various basic side chains
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
N-omega-(Tetralin-1-yl)alkyl Derivatives of 3,3-Dimethylpiperidine Are Highly Potent and Selective sigma-1 or sigma-2 Ligands
1998-01-01 Berardi, Francesco; Santoro, S.; Perrone, Roberto; Tortorella, V.; Govoni, S.; Lucchi, L.
N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: a potent and selective dopamine D4 ligand
1998-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella,
2-(Aryloxy)ethylamine derivatives: ring opened congeners of long chain 1-arylpiperazines with high 5-HT1A receptor affinity and selectivity versus D2 and a1 receptors
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
Preparation of Carbon-11 labelled N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a radioligand with picomolar affinity for dopamine D4 receptors.
1999-01-01 Langer, O; Halldin, C; Chou, Y; Sandell, J; Swahn, C; Nagren, K; Perrone, R; Berardi, Francesco; Leopoldo, Marcello; Farde, L.
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
Le applicazioni della chimica farmaceutica
2000-01-01 Altomare, Cosimo Damiano; Berardi, Francesco; Carotti, Angelo; Casini, G; Catalano, Alessia; Ferappi, M; Franchini, C; Lentini, Giovanni; Liso, G; Loiodice, Fulvio; Perrone, R; Tangari, N; Tortorella, Paolo; Trapani, G; revisore TORTORELLA, V.
N-aryl- or N-alkylpiperazine derivatives: the role of N-substituent on sigma-1, sigma-2, 5-HT1A and D2 receptor affinity
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Abate, CARMEN rosa; Tortorella, V.
Affinity of new chiral aryloxyalkylpiperidines towards sigma receptors
2000-01-01 Fracchiolla, Giuseppe; Berardi, Francesco; Colabufo, Nicola Antonio; Loiodice, F.; Perrone, R.; Tortorella, V.
AFFINITY OF NEW CHIRAL ARYLOXYALKYLPIPERIDINES TOWARDS σ RECEPTOR SUBTYPES.
2000-01-01 Berardi, F.; Colabufo, N. A.; Fracchiolla, G.; Loiodice, Fulvio; Perrone, R.; Tortorella, V.
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
Carbon-11 PB-12: an attempt to visualize the dopamine D4 receptor in the primate brain with positron emission tomography
2000-01-01 Langer, O.; Halldin, C.; Chou, Y. H.; Sandell, J.; Swahn, C. G.; Nagren, K; Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Farde, L.
A structure-affinity relationship study on derivatives of N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a high-affinity and selective D4 receptor ligand
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
The practice of medicinal chemistry
2001-01-01 Altomare, C; Berardi, Francesco; Carotti, Angelo; Casini, G; Catalano, Alessia; Ferappi, M; Franchini, Carlo; Lentini, Giovanni; Liso, G; Loiodice, F; Perrone, R; Tangari, N; Tortorella, Paolo; Trapani, G; Tortorella, V.
trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogs of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines
2001-01-01 Perrone, R; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, Enza; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R.
Determination of dopamine D4 receptor density in rat striatum using PB12 as a probe
2001-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Calo', R.; Leopoldo, Marcello; Perrone, Roberto; Tortorella, V.
Le applicazioni della Chimica Farmaceutica di Camille G. Wermuth
2001-01-01 Altomare, Cosimo Damiano; Berardi, Francesco; Carotti, Angelo; Casini, Giovanni; Catalano, Alessia; Ferappi, Marcello; Franchini, Carlo; Lentini, Giovanni; Liso, Gaetano; Loiodice, Fulvio; Perrone, Roberto; Tangari, Nicola; Tortorella, Paolo; Trapani, Giuseppe; Tortorella, Vincenzo
A multireceptorial binding reinvestigation on an extended class of sigma ligands: N-[omega-(indan-1-yl and tetralin-1-yl)alkyl] derivatives of 3,3-dimethylpiperidine reveal high affinities towards sigma1 and EBP sites
2001-01-01 Berardi, Francesco; Ferorelli, Savina; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, Roberto; Tortorella, V.
trans-4,4methoxyphenyl cycloehyl piperazines: A new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogues of aryl piperazines
2001-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, E; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R.
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands
2002-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
5-HT3 and 5-HT4 receptor affinities of naphtho[1,2-d]thiazole derivatives with various basic side chains | 1-gen-1997 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V. | |
N-omega-(Tetralin-1-yl)alkyl Derivatives of 3,3-Dimethylpiperidine Are Highly Potent and Selective sigma-1 or sigma-2 Ligands | 1-gen-1998 | Berardi, Francesco; Santoro, S.; Perrone, Roberto; Tortorella, V.; Govoni, S.; Lucchi, L. | |
N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: a potent and selective dopamine D4 ligand | 1-gen-1998 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, | |
2-(Aryloxy)ethylamine derivatives: ring opened congeners of long chain 1-arylpiperazines with high 5-HT1A receptor affinity and selectivity versus D2 and a1 receptors | 1-gen-1999 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V. | |
Preparation of Carbon-11 labelled N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a radioligand with picomolar affinity for dopamine D4 receptors. | 1-gen-1999 | Langer, O; Halldin, C; Chou, Y; Sandell, J; Swahn, C; Nagren, K; Perrone, R; Berardi, Francesco; Leopoldo, Marcello; Farde, L. | |
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5 | 1-gen-1999 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V. | |
Le applicazioni della chimica farmaceutica | 1-gen-2000 | Altomare, Cosimo Damiano; Berardi, Francesco; Carotti, Angelo; Casini, G; Catalano, Alessia; Ferappi, M; Franchini, C; Lentini, Giovanni; Liso, G; Loiodice, Fulvio; Perrone, R; Tangari, N; Tortorella, Paolo; Trapani, G; revisore TORTORELLA, V. | |
N-aryl- or N-alkylpiperazine derivatives: the role of N-substituent on sigma-1, sigma-2, 5-HT1A and D2 receptor affinity | 1-gen-2000 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Abate, CARMEN rosa; Tortorella, V. | |
Affinity of new chiral aryloxyalkylpiperidines towards sigma receptors | 1-gen-2000 | Fracchiolla, Giuseppe; Berardi, Francesco; Colabufo, Nicola Antonio; Loiodice, F.; Perrone, R.; Tortorella, V. | |
AFFINITY OF NEW CHIRAL ARYLOXYALKYLPIPERIDINES TOWARDS σ RECEPTOR SUBTYPES. | 1-gen-2000 | Berardi, F.; Colabufo, N. A.; Fracchiolla, G.; Loiodice, Fulvio; Perrone, R.; Tortorella, V. | |
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6 | 1-gen-2000 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V. | |
Carbon-11 PB-12: an attempt to visualize the dopamine D4 receptor in the primate brain with positron emission tomography | 1-gen-2000 | Langer, O.; Halldin, C.; Chou, Y. H.; Sandell, J.; Swahn, C. G.; Nagren, K; Perrone, Roberto; Berardi, Francesco; Leopoldo, Marcello; Farde, L. | |
A structure-affinity relationship study on derivatives of N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a high-affinity and selective D4 receptor ligand | 1-gen-2000 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V. | |
The practice of medicinal chemistry | 1-gen-2001 | Altomare, C; Berardi, Francesco; Carotti, Angelo; Casini, G; Catalano, Alessia; Ferappi, M; Franchini, Carlo; Lentini, Giovanni; Liso, G; Loiodice, F; Perrone, R; Tangari, N; Tortorella, Paolo; Trapani, G; Tortorella, V. | |
trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogs of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines | 1-gen-2001 | Perrone, R; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, Enza; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R. | |
Determination of dopamine D4 receptor density in rat striatum using PB12 as a probe | 1-gen-2001 | Colabufo, Nicola Antonio; Berardi, Francesco; Calo', R.; Leopoldo, Marcello; Perrone, Roberto; Tortorella, V. | |
Le applicazioni della Chimica Farmaceutica di Camille G. Wermuth | 1-gen-2001 | Altomare, Cosimo Damiano; Berardi, Francesco; Carotti, Angelo; Casini, Giovanni; Catalano, Alessia; Ferappi, Marcello; Franchini, Carlo; Lentini, Giovanni; Liso, Gaetano; Loiodice, Fulvio; Perrone, Roberto; Tangari, Nicola; Tortorella, Paolo; Trapani, Giuseppe; Tortorella, Vincenzo | |
A multireceptorial binding reinvestigation on an extended class of sigma ligands: N-[omega-(indan-1-yl and tetralin-1-yl)alkyl] derivatives of 3,3-dimethylpiperidine reveal high affinities towards sigma1 and EBP sites | 1-gen-2001 | Berardi, Francesco; Ferorelli, Savina; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, Roberto; Tortorella, V. | |
trans-4,4methoxyphenyl cycloehyl piperazines: A new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogues of aryl piperazines | 1-gen-2001 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, E; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R. | |
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands | 1-gen-2002 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V. |
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