Sfoglia per Autore
A multitarget approach in cancer research
2009-01-01 Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A.
Solid phase synthesis of potential PKs inhibitors
2009-01-01 Pellegrino, G; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Stefanachi, Angela; Pisani, Leonardo; Carotti, A.
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity
2009-01-01 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
An improved method for the biological evaluation of polyphenol derivatives as potential inhibitors of aβ(1–40) aggregation
2009-01-01 Stolfa, A; Cellamare, Saverio; Stefanachi, Angela; Catto, Marco; Leonetti, Francesco; Nicolotti, Orazio; Carotti, A.
Design of multiple-target anticancer agents: a daunting challenge for the medicinal chemist
2009-01-01 Carotti, A; Leonetti, Francesco; Catto, Marco; Stefanachi, Angela; Nicolotti, Orazio
A multitarget approach in cancer research. Joint Meeting on Medicinal Chemistry
2009-01-01 Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A.
A Multi-Objective Optimization Algorithm for Molecular Design
2009-01-01 Giangreco, I; Nicolotti, Orazio; Miscioscia, T. F.; Convertino, M; Mangiatordi, G. F.; Siragusa, L; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships
2009-01-01 Fernandez, F; Caamano, O; Nieto, Mi; Lopez, C; Garcia Mera, X; Stefanachi, Angela; Nicolotti, Orazio; Loza, Mi; Brea, J; Esteve, C; Segarra, V; Vidal, B; Carotti, Angelo
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity
2009-01-01 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
Ring closing metathesis mediated synthesis of d-, g- and e-N-HydroxylactaMS as potential coordinating molecular fragments of biologically relevant bivalent metals XX
2010-01-01 Leonetti, Francesco; Muncipinto, G; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Pisani, Leonardo; Carotti, A.
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor.
2010-01-01 Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A.
DESIGN SYNTHESIS AND BIOLOGYCAL ACTIVITY OF NEW POTENT GALLOYL-BASED MRP1 INHIBITORS FOR REVERSING MDR
2010-01-01 Pellicani, R. Z.; Niso, Mauro; Stefanachi, Angela; Berardi, Francesco; Carotti, A; Cellamare, Saverio; Colabufo, Nicola Antonio; Perrone, R.
Solid phase synthesis of a molecular library of pyrimidines, pyrazoles and isoxazoles with biological potential
2010-01-01 Pellegrino, G; Leonetti, F; Carotti, Angelo; Nicolotti, Orazio; Pisani, Leonardo; Stefanachi, Angela; Catto, Marco
Design, Synthesis and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors
2010-01-01 Pisani, Leonardo; Catto, Marco; Giangreco, I; Leonetti, Francesco; Nicolotti, Orazio; Stefanachi, Angela; Cellamare, Saverio; Carotti, Angelo
Coumarin as a versatile scaffold to selectively target biologically relevant cytochrome P450 enzymes: aromatase, steroid 11β-hydroxylase and aldosterone synthase
2011-01-01 Stefanachi, Angela; Favia, Ad; Nicolotti, Orazio; Leonetti, Francesco; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, Rw; Cellamare, Saverio; Carotti, Angelo
Insights into the complex formed by Matrix Metalloproteinase-2 and alloxan inhibitors: molecular dynamics simulations and free energy calculations
2011-01-01 Giangreco, I; Lattanzi, Gianluca; Nicolotti, Orazio; Catto, Marco; Laghezza, Antonio; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo
Discovery of a potent and selective hetero-bivalent AChE inhibitor via bioisosteric replacement
2011-01-01 Nicolotti, Orazio; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Giangreco, I.; Stefanachi, Angela; Carotti, Angelo
BCR-ABL inhibitors in chronic myeloid leukemia: process chemistry and biochemical profile
2011-01-01 Leonetti, Francesco; Stefanachi, Angela; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Cellamare, Saverio; Carotti, Angelo
Strategies of multi-objective optimization in drug discovery and development
2011-01-01 Nicolotti, Orazio; Giangreco, I; Introcaso, A; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo
Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Selective Aromatase Inhibitors
2011-01-01 Stefanachi, Angela; Favia, A. D.; Nicolotti, Orazio; Leonetti, F; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, R. W.; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A multitarget approach in cancer research | 1-gen-2009 | Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A. | |
Solid phase synthesis of potential PKs inhibitors | 1-gen-2009 | Pellegrino, G; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Stefanachi, Angela; Pisani, Leonardo; Carotti, A. | |
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity | 1-gen-2009 | Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A. | |
An improved method for the biological evaluation of polyphenol derivatives as potential inhibitors of aβ(1–40) aggregation | 1-gen-2009 | Stolfa, A; Cellamare, Saverio; Stefanachi, Angela; Catto, Marco; Leonetti, Francesco; Nicolotti, Orazio; Carotti, A. | |
Design of multiple-target anticancer agents: a daunting challenge for the medicinal chemist | 1-gen-2009 | Carotti, A; Leonetti, Francesco; Catto, Marco; Stefanachi, Angela; Nicolotti, Orazio | |
A multitarget approach in cancer research. Joint Meeting on Medicinal Chemistry | 1-gen-2009 | Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A. | |
A Multi-Objective Optimization Algorithm for Molecular Design | 1-gen-2009 | Giangreco, I; Nicolotti, Orazio; Miscioscia, T. F.; Convertino, M; Mangiatordi, G. F.; Siragusa, L; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Carotti, A. | |
1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships | 1-gen-2009 | Fernandez, F; Caamano, O; Nieto, Mi; Lopez, C; Garcia Mera, X; Stefanachi, Angela; Nicolotti, Orazio; Loza, Mi; Brea, J; Esteve, C; Segarra, V; Vidal, B; Carotti, Angelo | |
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity | 1-gen-2009 | Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A. | |
Ring closing metathesis mediated synthesis of d-, g- and e-N-HydroxylactaMS as potential coordinating molecular fragments of biologically relevant bivalent metals XX | 1-gen-2010 | Leonetti, Francesco; Muncipinto, G; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Pisani, Leonardo; Carotti, A. | |
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor. | 1-gen-2010 | Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A. | |
DESIGN SYNTHESIS AND BIOLOGYCAL ACTIVITY OF NEW POTENT GALLOYL-BASED MRP1 INHIBITORS FOR REVERSING MDR | 1-gen-2010 | Pellicani, R. Z.; Niso, Mauro; Stefanachi, Angela; Berardi, Francesco; Carotti, A; Cellamare, Saverio; Colabufo, Nicola Antonio; Perrone, R. | |
Solid phase synthesis of a molecular library of pyrimidines, pyrazoles and isoxazoles with biological potential | 1-gen-2010 | Pellegrino, G; Leonetti, F; Carotti, Angelo; Nicolotti, Orazio; Pisani, Leonardo; Stefanachi, Angela; Catto, Marco | |
Design, Synthesis and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors | 1-gen-2010 | Pisani, Leonardo; Catto, Marco; Giangreco, I; Leonetti, Francesco; Nicolotti, Orazio; Stefanachi, Angela; Cellamare, Saverio; Carotti, Angelo | |
Coumarin as a versatile scaffold to selectively target biologically relevant cytochrome P450 enzymes: aromatase, steroid 11β-hydroxylase and aldosterone synthase | 1-gen-2011 | Stefanachi, Angela; Favia, Ad; Nicolotti, Orazio; Leonetti, Francesco; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, Rw; Cellamare, Saverio; Carotti, Angelo | |
Insights into the complex formed by Matrix Metalloproteinase-2 and alloxan inhibitors: molecular dynamics simulations and free energy calculations | 1-gen-2011 | Giangreco, I; Lattanzi, Gianluca; Nicolotti, Orazio; Catto, Marco; Laghezza, Antonio; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo | |
Discovery of a potent and selective hetero-bivalent AChE inhibitor via bioisosteric replacement | 1-gen-2011 | Nicolotti, Orazio; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Giangreco, I.; Stefanachi, Angela; Carotti, Angelo | |
BCR-ABL inhibitors in chronic myeloid leukemia: process chemistry and biochemical profile | 1-gen-2011 | Leonetti, Francesco; Stefanachi, Angela; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Cellamare, Saverio; Carotti, Angelo | |
Strategies of multi-objective optimization in drug discovery and development | 1-gen-2011 | Nicolotti, Orazio; Giangreco, I; Introcaso, A; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo | |
Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Selective Aromatase Inhibitors | 1-gen-2011 | Stefanachi, Angela; Favia, A. D.; Nicolotti, Orazio; Leonetti, F; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, R. W.; Carotti, Angelo |
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