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Mostrati risultati da 21 a 40 di 81
Titolo Data di pubblicazione Autore(i) File
A multitarget approach in cancer research 1-gen-2009 Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A.
Solid phase synthesis of potential PKs inhibitors 1-gen-2009 Pellegrino, G; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Stefanachi, Angela; Pisani, Leonardo; Carotti, A.
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity 1-gen-2009 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
An improved method for the biological evaluation of polyphenol derivatives as potential inhibitors of aβ(1–40) aggregation 1-gen-2009 Stolfa, A; Cellamare, Saverio; Stefanachi, Angela; Catto, Marco; Leonetti, Francesco; Nicolotti, Orazio; Carotti, A.
Design of multiple-target anticancer agents: a daunting challenge for the medicinal chemist 1-gen-2009 Carotti, A; Leonetti, Francesco; Catto, Marco; Stefanachi, Angela; Nicolotti, Orazio
A multitarget approach in cancer research. Joint Meeting on Medicinal Chemistry 1-gen-2009 Leonetti, Francesco; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Muncipinto, G; Carotti, A.
A Multi-Objective Optimization Algorithm for Molecular Design 1-gen-2009 Giangreco, I; Nicolotti, Orazio; Miscioscia, T. F.; Convertino, M; Mangiatordi, G. F.; Siragusa, L; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
1,3-Dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships 1-gen-2009 Fernandez, F; Caamano, O; Nieto, Mi; Lopez, C; Garcia Mera, X; Stefanachi, Angela; Nicolotti, Orazio; Loza, Mi; Brea, J; Esteve, C; Segarra, V; Vidal, B; Carotti, Angelo
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity 1-gen-2009 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
Ring closing metathesis mediated synthesis of d-, g- and e-N-HydroxylactaMS as potential coordinating molecular fragments of biologically relevant bivalent metals XX 1-gen-2010 Leonetti, Francesco; Muncipinto, G; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Pisani, Leonardo; Carotti, A.
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor. 1-gen-2010 Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A.
DESIGN SYNTHESIS AND BIOLOGYCAL ACTIVITY OF NEW POTENT GALLOYL-BASED MRP1 INHIBITORS FOR REVERSING MDR 1-gen-2010 Pellicani, R. Z.; Niso, Mauro; Stefanachi, Angela; Berardi, Francesco; Carotti, A; Cellamare, Saverio; Colabufo, Nicola Antonio; Perrone, R.
Solid phase synthesis of a molecular library of pyrimidines, pyrazoles and isoxazoles with biological potential 1-gen-2010 Pellegrino, G; Leonetti, F; Carotti, Angelo; Nicolotti, Orazio; Pisani, Leonardo; Stefanachi, Angela; Catto, Marco
Design, Synthesis and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors 1-gen-2010 Pisani, Leonardo; Catto, Marco; Giangreco, I; Leonetti, Francesco; Nicolotti, Orazio; Stefanachi, Angela; Cellamare, Saverio; Carotti, Angelo
Coumarin as a versatile scaffold to selectively target biologically relevant cytochrome P450 enzymes: aromatase, steroid 11β-hydroxylase and aldosterone synthase 1-gen-2011 Stefanachi, Angela; Favia, Ad; Nicolotti, Orazio; Leonetti, Francesco; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, Rw; Cellamare, Saverio; Carotti, Angelo
Insights into the complex formed by Matrix Metalloproteinase-2 and alloxan inhibitors: molecular dynamics simulations and free energy calculations 1-gen-2011 Giangreco, I; Lattanzi, Gianluca; Nicolotti, Orazio; Catto, Marco; Laghezza, Antonio; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo
Discovery of a potent and selective hetero-bivalent AChE inhibitor via bioisosteric replacement 1-gen-2011 Nicolotti, Orazio; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Giangreco, I.; Stefanachi, Angela; Carotti, Angelo
BCR-ABL inhibitors in chronic myeloid leukemia: process chemistry and biochemical profile 1-gen-2011 Leonetti, Francesco; Stefanachi, Angela; Nicolotti, Orazio; Catto, Marco; Pisani, Leonardo; Cellamare, Saverio; Carotti, Angelo
Strategies of multi-objective optimization in drug discovery and development 1-gen-2011 Nicolotti, Orazio; Giangreco, I; Introcaso, A; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo
Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Selective Aromatase Inhibitors 1-gen-2011 Stefanachi, Angela; Favia, A. D.; Nicolotti, Orazio; Leonetti, F; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, R. W.; Carotti, Angelo
Mostrati risultati da 21 a 40 di 81
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