Sfoglia per Autore
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands
2002-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands
2002-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; DE GIORGIO, P.; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
A new method for evaluating sigma(2) ligand activity in the isolated guinea-pig bladder
2003-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Perrone, Roberto; Tortorella, Vincenzo
A new method to evaluate sigma-2 ligands activity in isolated guinea-pig bladder
2003-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, M.; Perrone, Roberto; Tortorella, V.
Synthesis and Structure-affinity relationship of 1-[omega-(4-Aryl-1-piperazinyl)alkyl]-1-arylketones as 5-HT7 Receptor Ligands
2003-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Leopoldo, Marcello; Tortorella, V.
Synthesis of chiral 1-[w-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at s1, s2 and sterol D8-D7 isomerase sites
2003-01-01 Berardi, Francesco; Loiodice, Fulvio; Fracchiolla, Giuseppe; Colabufo, Nicola Antonio; Perrone, R; Tortorella, V.
Synthesis of chiral 1-[omega-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at sigma1, sigma2 and Sterol delta 8-delta 7 isomerase sites
2003-01-01 Berardi, Francesco; Loiodice, F.; Fracchiolla, Giuseppe; Colabufo, Nicola Antonio; Perrone, Roberto; Tortorella, V.
Exploring the binding at sigma-1 receptor subtype: newly prepared heterocyclic omega-(1-alkyl)-derivatives of 3,3-dimethylpiperidine
2003-01-01 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Pedone, M. P.; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, R; Tortorella, V.
Studies on 1-arylpiperazine derivatives with affinity for rat 5-HT7 and 5-HT1A receptors
2004-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent
2004-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines
2004-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides as 5-HT7 receptor agents
2005-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands
2005-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Evaluation of sigma2 receptor expression in human invasive bladder cancer
2005-01-01 Pagliarulo, Vincenzo; Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Saponaro, P; Pagliarulo, A; Perrone, Roberto
First structure–activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure
2005-01-01 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto
Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter(SERT)and 5-HT1A receptors
2005-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Larizza, C.; Leopoldo, Marcello; Tortorella, V.
Synthesis and Biological Evaluation of Potential Positron Emission Tomography (PET) Ligands for Brain Visualization of Dopamine D3 Receptors.
2005-01-01 Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V.
A cyclohexylpiperazine derivate (PB28), displaying sigma-2 agonist and sigma-1 antagonist receptor activity, as a possible Glycoprotein P modulator and revertant of anthracycline resistance
2005-01-01 Azzariti, A; Colabufo, Nicola Antonio; Berardi, Francesco; Porcelli, L; Niso, M; Simone, Gm; Perrone, Roberto; Paradiso, A.
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors
2005-01-01 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma1 receptor
2005-01-01 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; M. P., Pedone; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, Roberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands | 1-gen-2002 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V. | |
Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands | 1-gen-2002 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; DE GIORGIO, P.; Lacivita, Enza; Perrone, Roberto; Tortorella, V. | |
A new method for evaluating sigma(2) ligand activity in the isolated guinea-pig bladder | 1-gen-2003 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Perrone, Roberto; Tortorella, Vincenzo | |
A new method to evaluate sigma-2 ligands activity in isolated guinea-pig bladder | 1-gen-2003 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, M.; Perrone, Roberto; Tortorella, V. | |
Synthesis and Structure-affinity relationship of 1-[omega-(4-Aryl-1-piperazinyl)alkyl]-1-arylketones as 5-HT7 Receptor Ligands | 1-gen-2003 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Leopoldo, Marcello; Tortorella, V. | |
Synthesis of chiral 1-[w-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at s1, s2 and sterol D8-D7 isomerase sites | 1-gen-2003 | Berardi, Francesco; Loiodice, Fulvio; Fracchiolla, Giuseppe; Colabufo, Nicola Antonio; Perrone, R; Tortorella, V. | |
Synthesis of chiral 1-[omega-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at sigma1, sigma2 and Sterol delta 8-delta 7 isomerase sites | 1-gen-2003 | Berardi, Francesco; Loiodice, F.; Fracchiolla, Giuseppe; Colabufo, Nicola Antonio; Perrone, Roberto; Tortorella, V. | |
Exploring the binding at sigma-1 receptor subtype: newly prepared heterocyclic omega-(1-alkyl)-derivatives of 3,3-dimethylpiperidine | 1-gen-2003 | Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Pedone, M. P.; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, R; Tortorella, V. | |
Studies on 1-arylpiperazine derivatives with affinity for rat 5-HT7 and 5-HT1A receptors | 1-gen-2004 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Perrone, Roberto; Tortorella, V. | |
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent | 1-gen-2004 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V. | |
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines | 1-gen-2004 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V. | |
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides as 5-HT7 receptor agents | 1-gen-2005 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V. | |
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands | 1-gen-2005 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V. | |
Evaluation of sigma2 receptor expression in human invasive bladder cancer | 1-gen-2005 | Pagliarulo, Vincenzo; Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Saponaro, P; Pagliarulo, A; Perrone, Roberto | |
First structure–activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure | 1-gen-2005 | Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto | |
Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter(SERT)and 5-HT1A receptors | 1-gen-2005 | Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Larizza, C.; Leopoldo, Marcello; Tortorella, V. | |
Synthesis and Biological Evaluation of Potential Positron Emission Tomography (PET) Ligands for Brain Visualization of Dopamine D3 Receptors. | 1-gen-2005 | Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V. | |
A cyclohexylpiperazine derivate (PB28), displaying sigma-2 agonist and sigma-1 antagonist receptor activity, as a possible Glycoprotein P modulator and revertant of anthracycline resistance | 1-gen-2005 | Azzariti, A; Colabufo, Nicola Antonio; Berardi, Francesco; Porcelli, L; Niso, M; Simone, Gm; Perrone, Roberto; Paradiso, A. | |
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors | 1-gen-2005 | Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto | |
Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma1 receptor | 1-gen-2005 | Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; M. P., Pedone; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, Roberto |
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