Sfoglia per Autore
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent
2004-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines
2004-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands
2005-01-01 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Distribution of sigma receptors in EMT-6 cells: preliminary biological evaluation of PB167 and potential for in-vivo PET
2005-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto; Contino, Marialessandra; Fazio, Ferruccio; Matarrese, Mario; Moresco, Rosa Maria; Niso, Mauro; Tortorella, Vincenzo
The sigma-2 receptor agonist PB28 inhibits calcium release from the endoplasmic reticulum of SK-N-SH neuroblastoma cells
2006-01-01 Cassano, Giuseppe; Gasparre, Giuseppe; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio
Cyclohexylpiperazine derivative PB28, a σ2 agonist and σ1 antagonist receptor, inhibits cell growth, modulates P-glycoprotein, and synergizes with anthracyclines in breast cancer
2006-01-01 Azzariti, Amalia; Colabufo, Nicola Antonio; Berardi, Francesco; Porcelli, Letizia; Niso, Mauro; Simone, Grazia M.; Perrone, Roberto; Paradiso, Angelo
The potent sigma receptor ligand PB167, as a potential PET radiotracer for evaluating the mammary sarcoma in mice
2006-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Perrone, Roberto; Tortorella, Vincenzo
Recent advances in the field of 5-HT7 receptor agents with 1-arylpiperazine structure.
2006-01-01 Leopoldo, Marcello; Lacivita, Enza; De Giorgio, P; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Correlation between sigma2 receptor protein expression and histopathologic grade in human bladder cancer
2006-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Ferorelli, Savina; Niso, Mauro; Perrone, Roberto; Pagliarulo, Arcangelo; Saponaro, Pasquale; Pagliarulo, Vincenzo
Is the sigma-2 receptor a histone binding protein?
2006-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Abate, CARMEN rosa; Niso, Mauro; Perrone, Roberto; Contino, Marialessandra
Design synthesis, and binding affinity of potential positron emission tomography (PET) ligands for visualitation of brain dopamine D3 receptors
2006-01-01 Leopoldo, Marcello; Lacivita, Enza; DE GIORGIO, P; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Human epididymal and prostatic tracts of vas deferens: different contraction response to noradrenaline stimulation in isolated organ bath assay
2007-01-01 Colabufo, Nicola Antonio; Pagliarulo, Vincenzo; Berardi, Francesco; Contino, Marialessandra; Perrone, Roberto; Niso, Mauro; Albo, Giancarlo; de Rienzo, Gaetano; Pagliarulo, Arcangelo
Design and evaluation of naphthol- and carbazole- containing fluorescent sigma ligands as potential probes for receptor binding studies
2007-01-01 Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, An; Niso, Mauro; Inglese, C; Berardi, Francesco; Perrone, Roberto
Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: Synthesis and binding affinities for 5-HT7 and 5-HT1A receptors
2007-01-01 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Bicalutamide failure in prostate cancer treatment: involvement of Multi Drug Resistance proteins
2008-01-01 Colabufo, Nicola Antonio; Pagliarulo, Vincenzo; Berardi, Francesco; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Ancona, Patrizia; Albo, Giancarlo; Pagliarulo, Arcangelo; Perrone, Roberto
Small molecules and acridone derivatives as P-gp inhibitors
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, MARIA GRAZIA; Cantore, M; Niso, Mauro; Perrone, Roberto
PB183, a sigma receptor ligand, as a potential PET probe for the imaging of prostate adenocarcinoma
2008-01-01 Colabufo, Nicola Antonio; Abate, CARMEN rosa; Contino, Marialessandra; Inglese, C.; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Novel 4-(-4-Aryl)cyclohexyl-1-(2-pyridyl)piperazines as delta8-delta7 sterol isomerase ( Emopamil Binding Protein) selective ligands with antiprolifative activity
2008-01-01 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; DE ROBERTIS, A; Leopoldo, Marcello; Colabufo, An; Niso, Mauro; Perrone, Roberto
Effect of some P-glycoprotein modulators on Rhodamine-123 absorption in guinea-pig ileum
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators
2008-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent | 1-gen-2004 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V. | |
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines | 1-gen-2004 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V. | |
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands | 1-gen-2005 | Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V. | |
Distribution of sigma receptors in EMT-6 cells: preliminary biological evaluation of PB167 and potential for in-vivo PET | 1-gen-2005 | Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto; Contino, Marialessandra; Fazio, Ferruccio; Matarrese, Mario; Moresco, Rosa Maria; Niso, Mauro; Tortorella, Vincenzo | |
The sigma-2 receptor agonist PB28 inhibits calcium release from the endoplasmic reticulum of SK-N-SH neuroblastoma cells | 1-gen-2006 | Cassano, Giuseppe; Gasparre, Giuseppe; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio | |
Cyclohexylpiperazine derivative PB28, a σ2 agonist and σ1 antagonist receptor, inhibits cell growth, modulates P-glycoprotein, and synergizes with anthracyclines in breast cancer | 1-gen-2006 | Azzariti, Amalia; Colabufo, Nicola Antonio; Berardi, Francesco; Porcelli, Letizia; Niso, Mauro; Simone, Grazia M.; Perrone, Roberto; Paradiso, Angelo | |
The potent sigma receptor ligand PB167, as a potential PET radiotracer for evaluating the mammary sarcoma in mice | 1-gen-2006 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Perrone, Roberto; Tortorella, Vincenzo | |
Recent advances in the field of 5-HT7 receptor agents with 1-arylpiperazine structure. | 1-gen-2006 | Leopoldo, Marcello; Lacivita, Enza; De Giorgio, P; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
Correlation between sigma2 receptor protein expression and histopathologic grade in human bladder cancer | 1-gen-2006 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Ferorelli, Savina; Niso, Mauro; Perrone, Roberto; Pagliarulo, Arcangelo; Saponaro, Pasquale; Pagliarulo, Vincenzo | |
Is the sigma-2 receptor a histone binding protein? | 1-gen-2006 | Colabufo, Nicola Antonio; Berardi, Francesco; Abate, CARMEN rosa; Niso, Mauro; Perrone, Roberto; Contino, Marialessandra | |
Design synthesis, and binding affinity of potential positron emission tomography (PET) ligands for visualitation of brain dopamine D3 receptors | 1-gen-2006 | Leopoldo, Marcello; Lacivita, Enza; DE GIORGIO, P; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
Human epididymal and prostatic tracts of vas deferens: different contraction response to noradrenaline stimulation in isolated organ bath assay | 1-gen-2007 | Colabufo, Nicola Antonio; Pagliarulo, Vincenzo; Berardi, Francesco; Contino, Marialessandra; Perrone, Roberto; Niso, Mauro; Albo, Giancarlo; de Rienzo, Gaetano; Pagliarulo, Arcangelo | |
Design and evaluation of naphthol- and carbazole- containing fluorescent sigma ligands as potential probes for receptor binding studies | 1-gen-2007 | Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, An; Niso, Mauro; Inglese, C; Berardi, Francesco; Perrone, Roberto | |
Bivalent ligand approach on 4-[2-(3-methoxyphenyl)ethyl]-1-(2-methoxyphenyl)piperazine: Synthesis and binding affinities for 5-HT7 and 5-HT1A receptors | 1-gen-2007 | Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
Bicalutamide failure in prostate cancer treatment: involvement of Multi Drug Resistance proteins | 1-gen-2008 | Colabufo, Nicola Antonio; Pagliarulo, Vincenzo; Berardi, Francesco; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Ancona, Patrizia; Albo, Giancarlo; Pagliarulo, Arcangelo; Perrone, Roberto | |
Small molecules and acridone derivatives as P-gp inhibitors | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, MARIA GRAZIA; Cantore, M; Niso, Mauro; Perrone, Roberto | |
PB183, a sigma receptor ligand, as a potential PET probe for the imaging of prostate adenocarcinoma | 1-gen-2008 | Colabufo, Nicola Antonio; Abate, CARMEN rosa; Contino, Marialessandra; Inglese, C.; Niso, Mauro; Berardi, Francesco; Perrone, Roberto | |
Novel 4-(-4-Aryl)cyclohexyl-1-(2-pyridyl)piperazines as delta8-delta7 sterol isomerase ( Emopamil Binding Protein) selective ligands with antiprolifative activity | 1-gen-2008 | Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; DE ROBERTIS, A; Leopoldo, Marcello; Colabufo, An; Niso, Mauro; Perrone, Roberto | |
Effect of some P-glycoprotein modulators on Rhodamine-123 absorption in guinea-pig ileum | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto | |
4-Biphenyl and 2-naphthyl substituted 6,7-dimethoxytetrahydroisoquinoline derivatives as potent P-gp modulators | 1-gen-2008 | Colabufo, Nicola Antonio; Berardi, Francesco; Cantore, Mariangela; Perrone, MARIA GRAZIA; Contino, Marialessandra; Inglese, Carmela; Niso, Mauro; Perrone, Roberto; Azzariti, Amalia; Simone, Grazia Maria; Paradiso, Angelo |
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