IRIS

Sfoglia per Autore  

Opzioni
Mostrati risultati da 1 a 20 di 89
Titolo Data di pubblicazione Autore(i) File
Solid-phase and Microwave Assisted Synthesis of Focused libraries of Imatinib analogues 1-gen-2005 Leonetti, F; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Stefanachi, Angela; Carotti, A.
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies 1-gen-2005 Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues 1-gen-2005 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A.
Application of Liebeskind-Srogl Thioester-Boronic Acid Couplings for the Scaffold Decoration of Dihydropyrimidines 1-gen-2006 Pisani, L.; Prokopcová, H.; Kappe, C. O.
Synthesis of heterocyclic compound libraries by automated sequential and parallel microwave synthesis. 1-gen-2006 Pisani, L.; Prokopcová, H.; Kappe, C. O.
Synthesis of 5-Aroyldihydropyrimidinones via Liebeskind–Srogl Thiol Ester– Boronic Acid Cross-Couplings 1-gen-2007 Prokopcová, Hana; Pisani, Leonardo; Oliver Kappe, C.
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors 1-gen-2007 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo
Structures of Human Monoamine Oxidase B Complexes with Selective Noncovalent Inhibitors: Safinamide and Coumarin Analogs 1-gen-2007 Binda, C; Wang, J; Pisani, Leonardo; Caccia, C; Carotti, Angelo; Salvati, P; Edmondson, D. E.; Mattevi, A.
5-aroyl-3,4-dihydropyrimidin-2-one library generation via automated sequential and parallel microwave-assisted synthesis techniques 1-gen-2007 Pisani, Leonardo; Prokopcová, Hana; Kremsner, Jennifer M.; Oliver Kappe, C.
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors 1-gen-2008 Leonetti, Francesco; Catto, Marco; Nicolotti, Orazio; Pisani, Leonardo; Cappa, A; Stefanachi, Angela; Carotti, Angelo
Solid phase synthesis of potential PKs inhibitors 1-gen-2009 Pellegrino, G; Leonetti, Francesco; Nicolotti, Orazio; Catto, Marco; Stefanachi, Angela; Pisani, Leonardo; Carotti, A.
Heterodimeric dual binding site cholinesterase inhibitors: surfing on the sub-nanomolar affinity 1-gen-2009 Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Leonetti, Francesco; Stefanachi, Angela; Carotti, A.
Discovery of a Novel Class of Potent Coumarin MAO-B inhibitors: Development and Biopharmacological Profiling of 7-[(3-Chlorobenzyl)oxy]-4-[(methylamino)methyl]-2H-chromen-2-one methanesulfonate (NW-1772) as a Highly Potent, Selective, Reversible and Orally Active MAO-B inhibitor 1-gen-2009 Pisani, Leonardo; Muncipinto, G; Miscioscia, Tf; Nicolotti, Orazio; Leonetti, Francesco; Catto, Marco; Caccia, C; Salvati, P; SOTO OTERO, R; MENDEZ ALVAREZ, E; Passeleu, C; Carotti, A.
Ring closing metathesis mediated synthesis of d-, g- and e-N-HydroxylactaMS as potential coordinating molecular fragments of biologically relevant bivalent metals XX 1-gen-2010 Leonetti, Francesco; Muncipinto, G; Stefanachi, Angela; Pellegrino, G; Nicolotti, Orazio; Catto, Marco; Cellamare, Saverio; Pisani, Leonardo; Carotti, A.
A molecular dynamics study of a sub-nanomolar dual binding site heterodimeric AChE inhibitor. 1-gen-2010 Nicolotti, Orazio; Giangreco, I; Pisani, Leonardo; Catto, Marco; Leonetti, Francesco; Stefanachi, Angela; Cellamare, Saverio; Carotti, A.
Solid phase synthesis of a molecular library of pyrimidines, pyrazoles and isoxazoles with biological potential 1-gen-2010 Pellegrino, G; Leonetti, F; Carotti, Angelo; Nicolotti, Orazio; Pisani, Leonardo; Stefanachi, Angela; Catto, Marco
Screening of benzamidine-based thrombin inhibitors via a linear interaction energy in continuum electrostatics model 1-gen-2010 Nicolotti, Orazio; Giangreco, I; Miscioscia, Tf; Convertino, M; Leonetti, Francesco; Pisani, Leonardo; Carotti, Angelo
Design, Synthesis and Biological Evaluation of Coumarin Derivatives Tethered to an Edrophonium-like Fragment as Highly Potent and Selective Dual Binding Site Acetylcholinesterase Inhibitors 1-gen-2010 Pisani, Leonardo; Catto, Marco; Giangreco, I; Leonetti, Francesco; Nicolotti, Orazio; Stefanachi, Angela; Cellamare, Saverio; Carotti, Angelo
Coumarin as a versatile scaffold to selectively target biologically relevant cytochrome P450 enzymes: aromatase, steroid 11β-hydroxylase and aldosterone synthase 1-gen-2011 Stefanachi, Angela; Favia, Ad; Nicolotti, Orazio; Leonetti, Francesco; Pisani, Leonardo; Catto, Marco; Zimmer, C; Hartmann, Rw; Cellamare, Saverio; Carotti, Angelo
6-Substituted-(E)-2-(benzofuran-3(2H)-ylidene)-N-methylacetamides as novel, potent and selective MAO inhibitors 1-gen-2011 Barletta, M.; Pisani, Leonardo; Catto, Marco; Nicolotti, Orazio; Soto Otero, R.; Carotti, Angelo
Mostrati risultati da 1 a 20 di 89
Legenda icone

  •  file ad accesso aperto
  •  file disponibili sulla rete interna
  •  file disponibili agli utenti autorizzati
  •  file disponibili solo agli amministratori
  •  file sotto embargo
  •  nessun file disponibile