Sfoglia per Autore
Evaluation of reactant-based and product-based approaches to the design of combinatorial libraries
2000-01-01 Gillet, Vj; Nicolotti, Orazio
Neuronal Nicotinic Agonists: a Multi-approach Development of the Pharmacophore
2001-01-01 Nicolotti, Orazio; PELLEGRINI CALACE, M. L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Centeno, N. B.; Sanz, F.; Carotti, Angelo
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D-QSAR predictive models,
2001-01-01 Carotti, A; Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano
Multi-approach development of a new pharmacophore for neuronal nicotinic acetylcholine receptor agonists,
2001-01-01 Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, A.
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D QSAR predictive models
2001-01-01 Carotti, A.; Nicolotti, Orazio; PELLEGRINI CALACE, M.; Carrieri, Antonio; Altomare, Cosimo Damiano
Cytisine derivatives as high affinity nAChR ligands: Synthesis and Comparative Molecular Field Analysis
2002-01-01 Nicolotti, Orazio; Boido, Cc; Sparatore, F; Carotti, Angelo
Multiobjective optimization in quantitative structure-activity relationships: Deriving accurate and interpretable QSARs
2002-01-01 Nicolotti, Orazio; Gillet, Vj; Fleming, Pj; Green, Dvs
Ligands of neuronal nicotinic acetylcholine receptor (nAChR): inferences from the Hansch and 3-D Quantitative Structure-Activity Relationship (QSAR) models
2002-01-01 Nicolotti, Orazio; Pellegrini Calace, M; Altomare, Cosimo Damiano; Carotti, Angelo; Carrieri, Antonio; Sanz, F.
A multi-objective approach to deriving QSAR models
2003-01-01 Nicolotti, Orazio; Gillet, Vj; Fleming, P; Green, D.
Insight into diastereospecific solvolysis of peptidyl-beta-lactams: combined kinetic and conformational studies
2003-01-01 Cellamare, Saverio; Coletti, C; Leonett, Fi; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A.
Insights into Diastereospecific Solvolysis of Peptidyl-β-Lactams: Combined Kinetic and Conformational Studies.
2003-01-01 Cellamare, Saverio; Coletti, A; Leonetti, Francesco; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A; Cellamare, S.
A multiobjective approach to deriving QSAR models
2004-01-01 Nicolotti, Orazio; Gillet, Vj; Fleming, P; Green, D.
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies
2004-01-01 Carotti, A; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIÉRREZ DE TERÁN, H; Loza, M. I.; Martinez, A; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela
Neuronal nicotinic acetylcholine receptor agonists: Pharmacophores, evolutionary QSAR and 3D-QSAR models
2004-01-01 Nicolotti, Orazio; Altomare, Cosimo Damiano; Pellegrini Calace, M; Carotti, Angelo
8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B
2004-01-01 Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio
Multi-objective approach to deriving QSAR models.
2004-01-01 Nicolotti, Orazio; Gillet, Vj; Fleming, Pj; Green, D.
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands
2004-01-01 Nicolotti, Orazio; Carotti, Angelo; Carrieri, Antonio; Pigini, M; Gentili, F; Brasili, L; Giannella, M; Quaglia, W; Piergentili, A; Bousquet, P; Dontenwill, M.
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies
2005-01-01 Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio
A novel function for non-deterministic scouting of optimal QSAR models out of a highly-structured physicochemical space.
2006-01-01 Nicolotti, Orazio; Miscioscia, T. F.; Leonetti, Francesco; Carotti, A.
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines from combined ligand- and structure-based approaches
2006-01-01 Stefanachi, Angela; Carotti, Angelo; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TERAN, H; Loza, M. I.; Martinez, A; Moro, S; Nicolotti, Orazio; Nieto, R; Pastor, M; Ravina, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Evaluation of reactant-based and product-based approaches to the design of combinatorial libraries | 1-gen-2000 | Gillet, Vj; Nicolotti, Orazio | |
Neuronal Nicotinic Agonists: a Multi-approach Development of the Pharmacophore | 1-gen-2001 | Nicolotti, Orazio; PELLEGRINI CALACE, M. L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Centeno, N. B.; Sanz, F.; Carotti, Angelo | |
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D-QSAR predictive models, | 1-gen-2001 | Carotti, A; Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano | |
Multi-approach development of a new pharmacophore for neuronal nicotinic acetylcholine receptor agonists, | 1-gen-2001 | Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, A. | |
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D QSAR predictive models | 1-gen-2001 | Carotti, A.; Nicolotti, Orazio; PELLEGRINI CALACE, M.; Carrieri, Antonio; Altomare, Cosimo Damiano | |
Cytisine derivatives as high affinity nAChR ligands: Synthesis and Comparative Molecular Field Analysis | 1-gen-2002 | Nicolotti, Orazio; Boido, Cc; Sparatore, F; Carotti, Angelo | |
Multiobjective optimization in quantitative structure-activity relationships: Deriving accurate and interpretable QSARs | 1-gen-2002 | Nicolotti, Orazio; Gillet, Vj; Fleming, Pj; Green, Dvs | |
Ligands of neuronal nicotinic acetylcholine receptor (nAChR): inferences from the Hansch and 3-D Quantitative Structure-Activity Relationship (QSAR) models | 1-gen-2002 | Nicolotti, Orazio; Pellegrini Calace, M; Altomare, Cosimo Damiano; Carotti, Angelo; Carrieri, Antonio; Sanz, F. | |
A multi-objective approach to deriving QSAR models | 1-gen-2003 | Nicolotti, Orazio; Gillet, Vj; Fleming, P; Green, D. | |
Insight into diastereospecific solvolysis of peptidyl-beta-lactams: combined kinetic and conformational studies | 1-gen-2003 | Cellamare, Saverio; Coletti, C; Leonett, Fi; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A. | |
Insights into Diastereospecific Solvolysis of Peptidyl-β-Lactams: Combined Kinetic and Conformational Studies. | 1-gen-2003 | Cellamare, Saverio; Coletti, A; Leonetti, Francesco; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A; Cellamare, S. | |
A multiobjective approach to deriving QSAR models | 1-gen-2004 | Nicolotti, Orazio; Gillet, Vj; Fleming, P; Green, D. | |
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies | 1-gen-2004 | Carotti, A; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIÉRREZ DE TERÁN, H; Loza, M. I.; Martinez, A; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela | |
Neuronal nicotinic acetylcholine receptor agonists: Pharmacophores, evolutionary QSAR and 3D-QSAR models | 1-gen-2004 | Nicolotti, Orazio; Altomare, Cosimo Damiano; Pellegrini Calace, M; Carotti, Angelo | |
8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B | 1-gen-2004 | Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio | |
Multi-objective approach to deriving QSAR models. | 1-gen-2004 | Nicolotti, Orazio; Gillet, Vj; Fleming, Pj; Green, D. | |
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands | 1-gen-2004 | Nicolotti, Orazio; Carotti, Angelo; Carrieri, Antonio; Pigini, M; Gentili, F; Brasili, L; Giannella, M; Quaglia, W; Piergentili, A; Bousquet, P; Dontenwill, M. | |
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies | 1-gen-2005 | Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio | |
A novel function for non-deterministic scouting of optimal QSAR models out of a highly-structured physicochemical space. | 1-gen-2006 | Nicolotti, Orazio; Miscioscia, T. F.; Leonetti, Francesco; Carotti, A. | |
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines from combined ligand- and structure-based approaches | 1-gen-2006 | Stefanachi, Angela; Carotti, Angelo; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TERAN, H; Loza, M. I.; Martinez, A; Moro, S; Nicolotti, Orazio; Nieto, R; Pastor, M; Ravina, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B. |
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