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Mostrati risultati da 1 a 20 di 228
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Evaluation of reactant-based and product-based approaches to the design of combinatorial libraries 1-gen-2000 Gillet, Vj; Nicolotti, Orazio
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D QSAR predictive models 1-gen-2001 Carotti, A.; Nicolotti, Orazio; PELLEGRINI CALACE, M.; Carrieri, Antonio; Altomare, Cosimo Damiano
Neuronal Nicotinic Agonists: a Multi-approach Development of the Pharmacophore 1-gen-2001 Nicolotti, Orazio; PELLEGRINI CALACE, M. L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Centeno, N. B.; Sanz, F.; Carotti, Angelo
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D-QSAR predictive models, 1-gen-2001 Carotti, A; Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano
Multi-approach development of a new pharmacophore for neuronal nicotinic acetylcholine receptor agonists, 1-gen-2001 Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, A.
Multiobjective optimization in quantitative structure-activity relationships: Deriving accurate and interpretable QSARs 1-gen-2002 Nicolotti, Orazio; Gillet, Vj; Fleming, Pj; Green, Dvs
Ligands of neuronal nicotinic acetylcholine receptor (nAChR): inferences from the Hansch and 3-D Quantitative Structure-Activity Relationship (QSAR) models 1-gen-2002 Nicolotti, Orazio; Pellegrini Calace, M; Altomare, Cosimo Damiano; Carotti, Angelo; Carrieri, Antonio; Sanz, F.
Cytisine derivatives as high affinity nAChR ligands: Synthesis and Comparative Molecular Field Analysis 1-gen-2002 Nicolotti, Orazio; Boido, Cc; Sparatore, F; Carotti, Angelo
Insights into Diastereospecific Solvolysis of Peptidyl-β-Lactams: Combined Kinetic and Conformational Studies. 1-gen-2003 Cellamare, Saverio; Coletti, A; Leonetti, Francesco; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A; Cellamare, S.
A multi-objective approach to deriving QSAR models 1-gen-2003 Nicolotti, Orazio; Gillet, Vj; Fleming, P; Green, D.
Insight into diastereospecific solvolysis of peptidyl-beta-lactams: combined kinetic and conformational studies 1-gen-2003 Cellamare, Saverio; Coletti, C; Leonett, Fi; Maccallini, C; Marrone, A; Nicolotti, Orazio; Re, N; Altomare, Cosimo Damiano; Carotti, A.
A multiobjective approach to deriving QSAR models 1-gen-2004 Nicolotti, Orazio; Gillet, Vj; Fleming, P; Green, D.
Multi-objective approach to deriving QSAR models. 1-gen-2004 Nicolotti, Orazio; Gillet, Vj; Fleming, Pj; Green, D.
Neuronal nicotinic acetylcholine receptor agonists: Pharmacophores, evolutionary QSAR and 3D-QSAR models 1-gen-2004 Nicolotti, Orazio; Altomare, Cosimo Damiano; Pellegrini Calace, M; Carotti, Angelo
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies 1-gen-2004 Carotti, A; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIÉRREZ DE TERÁN, H; Loza, M. I.; Martinez, A; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela
8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B 1-gen-2004 Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio
Pharmacophore development and 3D-QSAR study of I1 imidazoline binding site ligands 1-gen-2004 Nicolotti, Orazio; Carotti, Angelo; Carrieri, Antonio; Pigini, M; Gentili, F; Brasili, L; Giannella, M; Quaglia, W; Piergentili, A; Bousquet, P; Dontenwill, M.
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies 1-gen-2005 Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio
A novel function for non-deterministic scouting of optimal QSAR models out of a highly-structured physicochemical space. 1-gen-2006 Nicolotti, Orazio; Miscioscia, T. F.; Leonetti, Francesco; Carotti, A.
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines (9dAX) from combined ligand- and structure-based approaches 1-gen-2006 Stefanachi, Angela; Carotti, A; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TÉRAN, H; Loza, M. I.; Martínez, A; Moro, S; Morizzo, E; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; AND VIDAL, B.
Mostrati risultati da 1 a 20 di 228
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