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trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogs of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines 1-gen-2001 Perrone, R; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, Enza; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R.
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands 1-gen-2002 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands 1-gen-2002 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; DE GIORGIO, P.; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
Synthesis and Structure-affinity relationship of 1-[omega-(4-Aryl-1-piperazinyl)alkyl]-1-arylketones as 5-HT7 Receptor Ligands 1-gen-2003 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Leopoldo, Marcello; Tortorella, V.
Studies on 1-arylpiperazine derivatives with affinity for rat 5-HT7 and 5-HT1A receptors 1-gen-2004 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Perrone, Roberto; Tortorella, V.
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agent 1-gen-2004 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides as 5-HT7 receptor agents 1-gen-2005 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-phenyl-1-piperazinealkylamide derivatives, and therapeutic use thereof as 5-HT7 receptor ligands 1-gen-2005 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Contino, Marialessandra; Lacivita, Enza; Niso, Mauro; Perrone, Roberto; Tortorella, V.
Synthesis and Biological Evaluation of Potential Positron Emission Tomography (PET) Ligands for Brain Visualization of Dopamine D3 Receptors. 1-gen-2005 Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V.
First structure–activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure 1-gen-2005 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Contino, Marialessandra; Berardi, Francesco; Perrone, Roberto
Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter(SERT)and 5-HT1A receptors 1-gen-2005 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Larizza, C.; Leopoldo, Marcello; Tortorella, V.
11C-Labeling of N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors 1-gen-2005 Turolla, Ea; Matarrese, M; Belloli, S; Moresco, Rm; Simonelli, P; Todde, S; Fazio, F; Magni, F; Kienle, Mg; Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, Roberto
Design synthesis, and binding affinity of potential positron emission tomography (PET) ligands for visualitation of brain dopamine D3 receptors 1-gen-2006 Leopoldo, Marcello; Lacivita, Enza; DE GIORGIO, P; Colabufo, Nicola Antonio; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 ligands 1-gen-2006 Leopoldo, Marcello; Berardi, Francesco; Colabufo, Nicola Antonio; Lacivita, Enza; Perrone, R; Tortorella, V.
Synthesis and binding profile of constrained analogs of N-4-(4-ARYLPIPERAZIN-1-YL)BUTYL 3-METHOXYBENZAMIDES, a class of potential dopamine D3 receptor ligands 1-gen-2006 Leopoldo, Marcello; Lacivita, Enza; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto
Recent advances in the field of 5-HT7 receptor agents with 1-arylpiperazine structure. 1-gen-2006 Leopoldo, Marcello; Lacivita, Enza; De Giorgio, P; Colabufo, Nicola Antonio; Contino, Marialessandra; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors 1-gen-2006 Lacivita, Enza; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, R; Tortorella, V.
Selective Agents for Serotonin2C (5-HT2C) Receptor 1-gen-2006 Lacivita, Enza; Leopoldo, Marcello
Design and synthesis of arylpiperazine-based fluorescent ligands for serotonin 5-HT1A and dopamine D3 receptors. 1-gen-2007 Leopoldo, Marcello; Lacivita, Enza; Passafiume, E; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
Structure-activity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4aryl-1-piperazinehexanamides, a class of 5-HT7 receptor agents. 2 1-gen-2007 Leopoldo, Marcello; Lacivita, Enza; Contino, Marialessandra; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, Roberto
Mostrati risultati da 1 a 20 di 126
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