Sfoglia per Autore
Lipophilicity in Molecular Modeling of MAO Inhibitors.
1996-01-01 Barreca, Ml; Altomare, Cosimo Damiano; Leonetti, Francesco; Carotti, A; Ferappi, M; Carrupt, Pa; Testa, B.
Modeling of MAO-A/MAO-B Inhibitory Activity and Selectivity: 2D- and 3D-QSAR Studies.
1996-01-01 Barreca, M. L.; Altomare, Cosimo Damiano; Leonetti, Francesco; Carotti, A; Weber, P; Gaillard, P; Carrupt, P. A.; Testa, B.
2-D and 3-D modeling of imadazoline receptor ligands: insights into pharmacophore
1997-01-01 Carrieri, Antonio; L., Brasili; Leonetti, Francesco; M., Pigini; M., Giannella; P., Bousquet; Carotti, Angelo
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.
1998-01-01 Pigini, M; Bousquet, P; Brasili, L; Carrieri, Antonio; Cavagna, R; Dontenwill, M; Gentili, F; Giannella, M; Leonetti, Francesco; Piergentili, A; Quaglia, W; Carotti, Angelo
Binding of tracizolines to the imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models
1999-01-01 Pigini, M; Bousquet, P; Brasili, L; Carrieri, Antonio; Dontewill, M; Gentili, F; Giannella, M; Leonetti, Francesco; Piergentili, A; Quaglia, W; Carotti, Angelo
Positional Scanning Libraries of Fluorogenic Substrates for Determining Protease Specificity, Incorporating P1 Diversity.
1999-01-01 Leonetti, Francesco; Backes, B. J.; Harris, J. L.; Craik, C. S.; Ellman, J. A.
Synthesis of positional-scanning libraries of fluorogenic peptide substrates to define the extended substrate specificity of plasmin and thrombin
2000-01-01 Backes, J. B.; Harris, J. L.; Leonetti, Francesco; Craik, C. S.; Ellman, J. A.
Rapid and general profiling of protease specificity by using combinatorial fluorogenic substrate libraries
2000-01-01 Harris, J. L.; Backes, B. J.; Leonetti, Francesco; Mahrus, S.; Craik, C. S.; Ellman, J. A.
Positional Scanning Libraries of Fluorogenic Peptide Substrates for Determining Protease Specificity.
2000-01-01 Leonetti, Francesco; Harris, J. L.; Backes, B. J.; Craik, C. S.; Ellman, J. A.
Peptide-aminomethylcoumarin Positional Scanning Libraries for Determining Protease Specificity, Incorporating P1 Diversity
2000-01-01 Leonetti, Francesco; Backes, B. J.; Ellman, J. A.; Harris, J. L.; Craik, C. S.
Inhibition of monoamine oxidases by functionalized coumarin derivatives: biological activity, QSARs, and 3-D QSARs
2000-01-01 Gnerre, C; Catto, Marco; Leonetti, Francesco; Weber, P; Carrupt, Pa; Altomare, Cosimo Damiano; Carotti, A; Testa, B.
Coumarins Derivatives as Dual Inhibitors of Acetylcholinesterase and Monoamine Oxidase
2001-01-01 Bruehlmann, C; Ooms, F; Carrupt, Pa; Testa, B; Catto, Marco; Leonetti, Francesco; Altomare, Cosimo Damiano; Carotti, Angelo
Expedient solid-phase synthesis of fluorogenic protease substrates using the 7-amino-4-carbamoylmethylcoumarin (ACC)
2002-01-01 Maly, D. J.; Leonetti, Francesco; Backes, B. J.; Dauber, D. S.; Harris, J. L.; Craik, C. S.; Ellman, J. A.
Benzodiazepine-induced superoxide signals B cell apoptosis: mechanistic insight and potential therapeutic utility
2002-01-01 Blatt, N. B.; Bednarski, J. J.; Warner, R. E.; Leonetti, Francesco; Johnson, K. M.; Boitano, A.; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A.; OPIPARI JR, A. W.; Glick, G. D.
New peptidyl -beta-lactams: solution-solid phase synthesis for the preparation of antibiotic libraries
2002-01-01 Leonetti, Francesco; Maccallini, C; Cellamare, Saverio; Jabes, D; Carotti, Angelo
New peptidyl-β-lactams: solution-solid phase synthesis for the preparation of antibiotic libraries.
2002-01-01 Leonetti, Francesco; Maccallini, C; Cellammare, S; Jabes, D; Carotti, A.
New peptidyl-beta-lactams: solution-solid phase synthesis for the preparation of antibiotic libraries
2002-01-01 Leonetti, Francesco; C., Maccallini; Cellamare, Saverio; D., Jabes; A., Carotti
Convergent Solution Phase and Solid Phase Synthesis for the Preparation of β-Lactam Antibiotic Libraries
2002-01-01 Leonetti, Francesco; Cellammare, S; Maccallini, C; Jabes, D; Carotti, A.
Attenuation of autoimmune disease in fas-deficient mice by treatment with a cytotoxic benzodiazepine
2003-01-01 Bednarski, J. J.; Warner, R. E.; Rao, T.; Leonetti, Francesco; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A.; OPIPARI JR, A. W.; Glick, G. D.
Fast and highly efficient one-pot synthesis of 9-deazaxanthines
2003-01-01 Stefanachi, Angela; Leonetti, Francesco; Cappa, A.; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Lipophilicity in Molecular Modeling of MAO Inhibitors. | 1-gen-1996 | Barreca, Ml; Altomare, Cosimo Damiano; Leonetti, Francesco; Carotti, A; Ferappi, M; Carrupt, Pa; Testa, B. | |
Modeling of MAO-A/MAO-B Inhibitory Activity and Selectivity: 2D- and 3D-QSAR Studies. | 1-gen-1996 | Barreca, M. L.; Altomare, Cosimo Damiano; Leonetti, Francesco; Carotti, A; Weber, P; Gaillard, P; Carrupt, P. A.; Testa, B. | |
2-D and 3-D modeling of imadazoline receptor ligands: insights into pharmacophore | 1-gen-1997 | Carrieri, Antonio; L., Brasili; Leonetti, Francesco; M., Pigini; M., Giannella; P., Bousquet; Carotti, Angelo | |
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models. | 1-gen-1998 | Pigini, M; Bousquet, P; Brasili, L; Carrieri, Antonio; Cavagna, R; Dontenwill, M; Gentili, F; Giannella, M; Leonetti, Francesco; Piergentili, A; Quaglia, W; Carotti, Angelo | |
Binding of tracizolines to the imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models | 1-gen-1999 | Pigini, M; Bousquet, P; Brasili, L; Carrieri, Antonio; Dontewill, M; Gentili, F; Giannella, M; Leonetti, Francesco; Piergentili, A; Quaglia, W; Carotti, Angelo | |
Positional Scanning Libraries of Fluorogenic Substrates for Determining Protease Specificity, Incorporating P1 Diversity. | 1-gen-1999 | Leonetti, Francesco; Backes, B. J.; Harris, J. L.; Craik, C. S.; Ellman, J. A. | |
Synthesis of positional-scanning libraries of fluorogenic peptide substrates to define the extended substrate specificity of plasmin and thrombin | 1-gen-2000 | Backes, J. B.; Harris, J. L.; Leonetti, Francesco; Craik, C. S.; Ellman, J. A. | |
Rapid and general profiling of protease specificity by using combinatorial fluorogenic substrate libraries | 1-gen-2000 | Harris, J. L.; Backes, B. J.; Leonetti, Francesco; Mahrus, S.; Craik, C. S.; Ellman, J. A. | |
Positional Scanning Libraries of Fluorogenic Peptide Substrates for Determining Protease Specificity. | 1-gen-2000 | Leonetti, Francesco; Harris, J. L.; Backes, B. J.; Craik, C. S.; Ellman, J. A. | |
Peptide-aminomethylcoumarin Positional Scanning Libraries for Determining Protease Specificity, Incorporating P1 Diversity | 1-gen-2000 | Leonetti, Francesco; Backes, B. J.; Ellman, J. A.; Harris, J. L.; Craik, C. S. | |
Inhibition of monoamine oxidases by functionalized coumarin derivatives: biological activity, QSARs, and 3-D QSARs | 1-gen-2000 | Gnerre, C; Catto, Marco; Leonetti, Francesco; Weber, P; Carrupt, Pa; Altomare, Cosimo Damiano; Carotti, A; Testa, B. | |
Coumarins Derivatives as Dual Inhibitors of Acetylcholinesterase and Monoamine Oxidase | 1-gen-2001 | Bruehlmann, C; Ooms, F; Carrupt, Pa; Testa, B; Catto, Marco; Leonetti, Francesco; Altomare, Cosimo Damiano; Carotti, Angelo | |
Expedient solid-phase synthesis of fluorogenic protease substrates using the 7-amino-4-carbamoylmethylcoumarin (ACC) | 1-gen-2002 | Maly, D. J.; Leonetti, Francesco; Backes, B. J.; Dauber, D. S.; Harris, J. L.; Craik, C. S.; Ellman, J. A. | |
Benzodiazepine-induced superoxide signals B cell apoptosis: mechanistic insight and potential therapeutic utility | 1-gen-2002 | Blatt, N. B.; Bednarski, J. J.; Warner, R. E.; Leonetti, Francesco; Johnson, K. M.; Boitano, A.; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A.; OPIPARI JR, A. W.; Glick, G. D. | |
New peptidyl -beta-lactams: solution-solid phase synthesis for the preparation of antibiotic libraries | 1-gen-2002 | Leonetti, Francesco; Maccallini, C; Cellamare, Saverio; Jabes, D; Carotti, Angelo | |
New peptidyl-β-lactams: solution-solid phase synthesis for the preparation of antibiotic libraries. | 1-gen-2002 | Leonetti, Francesco; Maccallini, C; Cellammare, S; Jabes, D; Carotti, A. | |
New peptidyl-beta-lactams: solution-solid phase synthesis for the preparation of antibiotic libraries | 1-gen-2002 | Leonetti, Francesco; C., Maccallini; Cellamare, Saverio; D., Jabes; A., Carotti | |
Convergent Solution Phase and Solid Phase Synthesis for the Preparation of β-Lactam Antibiotic Libraries | 1-gen-2002 | Leonetti, Francesco; Cellammare, S; Maccallini, C; Jabes, D; Carotti, A. | |
Attenuation of autoimmune disease in fas-deficient mice by treatment with a cytotoxic benzodiazepine | 1-gen-2003 | Bednarski, J. J.; Warner, R. E.; Rao, T.; Leonetti, Francesco; Yung, R.; Richardson, B. C.; Johnson, K. J.; Ellman, J. A.; OPIPARI JR, A. W.; Glick, G. D. | |
Fast and highly efficient one-pot synthesis of 9-deazaxanthines | 1-gen-2003 | Stefanachi, Angela; Leonetti, Francesco; Cappa, A.; Carotti, Angelo |
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