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Lipophilicity of teicoplanin antibiotics as assessed by reversed phase high-performance liquid chromatography: quantitative structure-property and structure-activity relationships 1-gen-1994 Altomare, Cosimo Damiano; Carotti, Angelo; Cellamare, Saverio; Carrieri, Antonio; Ciabatti, R; Malabarba, A.
Papain catalyzed hydrolysis of aryl esters: a comparison of the Hansch, Docking and CoMFA methods 1-gen-1994 Carrieri, Antonio; Altomare, Cosimo Damiano; Barreca, M. L.; Contento, A; Carotti, Angelo; Hansch, C.
2-D and 3-D modeling of imadazoline receptor ligands: insights into pharmacophore 1-gen-1997 Carrieri, Antonio; L., Brasili; Leonetti, Francesco; M., Pigini; M., Giannella; P., Bousquet; Carotti, Angelo
High affinity central benzodiazepine receptor ligands: synthesis and structure-activity relationship studies of a new series of pyrazolo[4,3-c]quinolin-3-ones. 1-gen-1998 Savini, L; Massarelli, P; Nencini, C; Pellerano, C; Biggio, G; Maciocco, A; Tuligi, G; Carrieri, Antonio; Cinone, N; Carotti, Angelo
Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models. 1-gen-1998 Pigini, M; Bousquet, P; Brasili, L; Carrieri, Antonio; Cavagna, R; Dontenwill, M; Gentili, F; Giannella, M; Leonetti, Francesco; Piergentili, A; Quaglia, W; Carotti, Angelo
Comparative Molecular Field Analysis of pyridawinone-containing alfa1-antagonists 1-gen-1999 Cinone, N.; Carrieri, Antonio; Strappaghetti, G.; Corsano, S.; Barbaro, R.; Carotti, Angelo
Conformational restricted butyrophenones with mixed dopaminergic (D2) and serotoninergic (5-HT2A, 5-HT2C) affinities. Synthesis, pharmacology and 3D-QSAR 1-gen-1999 Ravina, E.; Negreira, J.; Cid, J.; Masaguer, C. F.; Rosa, E.; Rivas, M. E.; Fontenla, J. A.; Loza, M. I.; Tristan, E.; Cadavid, M. I.; Sanz, F.; Lozoya, E.; Carotti, Angelo; Carrieri, Antonio
Binding of tracizolines to the imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models 1-gen-1999 Pigini, M; Bousquet, P; Brasili, L; Carrieri, Antonio; Dontewill, M; Gentili, F; Giannella, M; Leonetti, Francesco; Piergentili, A; Quaglia, W; Carotti, Angelo
2-(2-Phenylcyclopropyl)-Imidazolines: Reversed Enantioselective Interaction At I1 and I2 Imidazoline Receptors 1-gen-1999 Quaglia, W.; Bousquet, P.; Pigini, M.; Carotti, Angelo; Carrieri, Antonio; Dontemwill, M.; Gentili, F.; Giannella, M.; Piergentili, A.; Brasili, L.
Comparative molecular field analysis (CoMFA) and docking studies of non- nucleoside HIV-1 RT inhibitors (NNIs) 1-gen-1999 Barreca, M. L.; Carotti, A.; Carrieri, A.; Chimirri, A.; Monforte, A. M.; Pellegrini Calace, M.; Rao, A.
2-(2-phenylcyclopropyl)imidazolines: Reversed enantioselective interaction at I1 and I2 imidazoline receptors [1] 1-gen-1999 Quaglia, W.; Bousquet, P.; Pigini, M.; Carotti, A.; Carrieri, A.; Dontenwill, M.; Gentili, F.; Giannella, M.; Maranca, F.; Piergentili, A.; Brasili, L.
Conformationally constrained butyrophenones with mixed dopaminergic (D(2)) and serotoninergic (5-HT(2A), 5-HT(2C)) affinities: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo- and -thienocycloalkanones as putative atypical antipsychotics. 1-gen-1999 Raviña, E; Negreira, J; Cid, J; Masaguer, Cf; Rosa, E; Rivas, Me; Fontenla, Ja; Loza, Mi; Tristán, H; Cadavid, Mi; Sanz, F; Lozoya, E; Carotti, Angelo; Carrieri, Antonio
SAR of Non-Nucleoside HIV-1 RT inhibitors (NNRTIs): Comparative Molecular field Analysis (CoMFA) and Docking Studies 1-gen-1999 Barreca, M. L.; Carotti, Angelo; Carrieri, Antonio; Chimirri, A.; Monforte, A. M.; PELLEGRINI CALACE, M.; Rao, A.
Understanding of the MAO-A and B Reversible Inhibitory Activity and Selectivity by Using 3D Descriptors of Lipophilicity 1-gen-2000 Altomare, Cosimo Damiano; Carrieri, Antonio; Summo, L; Catto, Marco; Carotti, A; Carrupt, Pa; Testa, B.
Extended form of a retro-inverso peptide stabilized by beta-sheet unidirectional H-bonds: Crystallographic and NMR evidence 1-gen-2001 Carotti, Angelo; Carrieri, Antonio; Cellamare, Saverio; Fanizzi, Fp; Gavuzzo, E; Mazza, F.
Neuronal nicotinic receptor agonists: multi-approach pharmacophore development and 3D-QSAR predictive models, 1-gen-2001 Carotti, A; Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano
Neuronal Nicotinic Agonists: a Multi-approach Development of the Pharmacophore 1-gen-2001 Nicolotti, Orazio; PELLEGRINI CALACE, M. L.; Carrieri, Antonio; Altomare, Cosimo Damiano; Centeno, N. B.; Sanz, F.; Carotti, Angelo
High affinity central benzodiazepine receptor ligands II: QSAR studies and CoMFA analysis pyrazolo(4,3-c)quinolin-3-ones 1-gen-2001 Savini, L.; Chiasserini, L.; Pellerano, C.; Biggio, G.; Maciocco, E.; Serra, M.; Cinone, N.; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, Angelo
3D-QSAR models and docking studies of reversible inhibitors of type A and B Monoamine Oxidases 1-gen-2001 Carotti, A.; Barreca, M. L.; PELLEGRINI CALACE, M.; Carrieri, Antonio; Altomare, Cosimo Damiano
Multi-approach development of a new pharmacophore for neuronal nicotinic acetylcholine receptor agonists, 1-gen-2001 Nicolotti, Orazio; Pellegrini Calace, M; Carrieri, Antonio; Altomare, Cosimo Damiano; Carotti, A.
Mostrati risultati da 1 a 20 di 129
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