Sfoglia per Autore
Fast and highly efficient one-pot synthesis of 9-deazaxanthines
2003-01-01 Stefanachi, Angela; Leonetti, Francesco; Cappa, A.; Carotti, Angelo
Synthesis of 1-Substituted-6-methyluracils
2003-01-01 Nieto, R. M.; Coelho, A; Martinez, A; Stefanachi, Angela; Sotelo, E; Raviña, E.
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies
2003-01-01 Stefanachi, Angela
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies
2004-01-01 Carotti, A; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIÉRREZ DE TERÁN, H; Loza, M. I.; Martinez, A; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela
8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B
2004-01-01 Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues
2005-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A.
Solid-phase and Microwave Assisted Synthesis of Focused libraries of Imatinib analogues
2005-01-01 Leonetti, F; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Stefanachi, Angela; Carotti, A.
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies
2005-01-01 Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines from combined ligand- and structure-based approaches
2006-01-01 Stefanachi, Angela; Carotti, A; Brea, Jm; Cadavid, Mi; Centeno, Nb; Esteve, C; Fontaine, F; GUTIERREZ DE TRAN, H; Loza, Mi; Martinez, A; Moro, S; Nicolotti, Orazio; Nieto, R; Pastor, M; Ravina, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B.
Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor
2006-01-01 Carotti, Angelo; Cadavid, Mi; Centeno, Nb; Esteve, C; Loza, Mi; Martinez, A; Nieto, R; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela; Vidal, B.
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines from combined ligand- and structure-based approaches
2006-01-01 Stefanachi, Angela; Carotti, Angelo; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TERAN, H; Loza, M. I.; Martinez, A; Moro, S; Nicolotti, Orazio; Nieto, R; Pastor, M; Ravina, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B.
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines (9dAX) from combined ligand- and structure-based approaches
2006-01-01 Stefanachi, Angela; Carotti, A; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TÉRAN, H; Loza, M. I.; Martínez, A; Moro, S; Morizzo, E; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; AND VIDAL, B.
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications
2007-01-01 Campagna, Francesco; Cellamare, Saverio; Stefanachi, Angela; Stolfa, D. A.; Basile, T; Ferappi, M; Catto, Marco; Carotti, A.
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications
2007-01-01 Campagna, F; Cellamare, Saverio; Stefanachi, Angela; Stolfa, Ad; Basile, T; Ferappi, M; Catto, Marco; Carotti, A.
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors
2007-01-01 Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo
Synthetic Applications of Polystyrene-Supported 1,1,3,3-Tetramethylguanidine
2008-01-01 Coelho, A; Crespo, A; Fernández, F; Biagini, P. F.; Stefanachi, Angela; Sotelo, E.
1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships
2008-01-01 Stefanachi, Angela; Nicolotti, Orazio; Leonetti, Francesco; Cellamare, Saverio; Campagna, Francesco; Loza, Mi; Brea, Jm; Mazza, F; Gavuzzo, E; Carotti, Angelo
1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor
2008-01-01 Stefanachi, A; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Loza, M. I.; Martinez, A; Nieto, R; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B.; Carotti, A
Design, synthesis, and biological evaluation of glycine-based molecular tongs as inhibitors of Aβ40 aggregation in vitro
2008-01-01 Cellamare, Saverio; Stefanachi, Angela; Stolfa, D. A.; Basile, T; Catto, Marco; Campagna, Francesco; Sotelo, E; Acquafredda, Pasquale; Carotti, Angelo
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors
2008-01-01 Leonetti, Francesco; Catto, Marco; Nicolotti, Orazio; Pisani, Leonardo; Cappa, A; Stefanachi, Angela; Carotti, Angelo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Fast and highly efficient one-pot synthesis of 9-deazaxanthines | 1-gen-2003 | Stefanachi, Angela; Leonetti, Francesco; Cappa, A.; Carotti, Angelo | |
Synthesis of 1-Substituted-6-methyluracils | 1-gen-2003 | Nieto, R. M.; Coelho, A; Martinez, A; Stefanachi, Angela; Sotelo, E; Raviña, E. | |
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies | 1-gen-2003 | Stefanachi, Angela | |
9-Deazaxanthines as selective A2B AR ligands: Design, Synthesis and SAFIR studies | 1-gen-2004 | Carotti, A; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIÉRREZ DE TERÁN, H; Loza, M. I.; Martinez, A; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela | |
8-Substituted- 9-deazaxanthines as adenosine receptor ligands: design, synthesis and structure-affinity relationships at A2B | 1-gen-2004 | Carotti, Angelo; Stefanachi, Angela; Ravina, E; Sotelo, E; Loza, Mi; Cadavid, Mi; Centeno, Nb; Nicolotti, Orazio | |
Solid Phase and Microwave Assisted Synthesis of Focused Libraries of Imatinib Analogues | 1-gen-2005 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Catto, Marco; Stefanachi, Angela; Carotti, A. | |
Solid-phase and Microwave Assisted Synthesis of Focused libraries of Imatinib analogues | 1-gen-2005 | Leonetti, F; Capaldi, C; Pisani, Leonardo; Muncipinto, G; Stefanachi, Angela; Carotti, A. | |
In silico design and microwave-assisted solid phase synthesis of focused libraries of enzyme inhibitors with potential in cancer and neurological therapies | 1-gen-2005 | Carotti, Angelo; Leonetti, Francesco; Stefanachi, Angela; Catto, Marco; Capaldi, C.; Muncipinto, G.; Pisani, Leonardo; Nicolotti, Orazio | |
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines from combined ligand- and structure-based approaches | 1-gen-2006 | Stefanachi, Angela; Carotti, A; Brea, Jm; Cadavid, Mi; Centeno, Nb; Esteve, C; Fontaine, F; GUTIERREZ DE TRAN, H; Loza, Mi; Martinez, A; Moro, S; Nicolotti, Orazio; Nieto, R; Pastor, M; Ravina, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B. | |
Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor | 1-gen-2006 | Carotti, Angelo; Cadavid, Mi; Centeno, Nb; Esteve, C; Loza, Mi; Martinez, A; Nieto, R; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Stefanachi, Angela; Vidal, B. | |
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines from combined ligand- and structure-based approaches | 1-gen-2006 | Stefanachi, Angela; Carotti, Angelo; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TERAN, H; Loza, M. I.; Martinez, A; Moro, S; Nicolotti, Orazio; Nieto, R; Pastor, M; Ravina, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B. | |
Structural insights into hA2B affinity and selectivity of 9-deazaxanthines (9dAX) from combined ligand- and structure-based approaches | 1-gen-2006 | Stefanachi, Angela; Carotti, A; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Fontaine, F; GUTIERREZ DE TÉRAN, H; Loza, M. I.; Martínez, A; Moro, S; Morizzo, E; Nicolotti, Orazio; Nieto, R; Pastor, M; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; AND VIDAL, B. | |
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications | 1-gen-2007 | Campagna, Francesco; Cellamare, Saverio; Stefanachi, Angela; Stolfa, D. A.; Basile, T; Ferappi, M; Catto, Marco; Carotti, A. | |
Inhibiting Aβ1-40 in vitro aggregation by glycine-based molecular tongs: rational design and mechanistic implications | 1-gen-2007 | Campagna, F; Cellamare, Saverio; Stefanachi, Angela; Stolfa, Ad; Basile, T; Ferappi, M; Catto, Marco; Carotti, A. | |
Solid Phase Synthesis of Safinamide and Analogues as Potent and Selective MAO-B Inhibitors | 1-gen-2007 | Leonetti, Francesco; Capaldi, C; Pisani, Leonardo; Nicolotti, Orazio; Muncipinto, G; Stefanachi, Angela; Cellamare, Saverio; Caccia, C; Carotti, Angelo | |
Synthetic Applications of Polystyrene-Supported 1,1,3,3-Tetramethylguanidine | 1-gen-2008 | Coelho, A; Crespo, A; Fernández, F; Biagini, P. F.; Stefanachi, Angela; Sotelo, E. | |
1,3-Dialkyl-8-(hetero)aryl-9-OH-9-deazaxanthines as potent A2B adenosine receptor antagonists: design, synthesis, structure-affinity and structure-selectivity relationships | 1-gen-2008 | Stefanachi, Angela; Nicolotti, Orazio; Leonetti, Francesco; Cellamare, Saverio; Campagna, Francesco; Loza, Mi; Brea, Jm; Mazza, F; Gavuzzo, E; Carotti, Angelo | |
1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor | 1-gen-2008 | Stefanachi, A; Brea, J. M.; Cadavid, M. I.; Centeno, N. B.; Esteve, C; Loza, M. I.; Martinez, A; Nieto, R; Raviña, E; Sanz, F; Segarra, V; Sotelo, E; Vidal, B.; Carotti, A | |
Design, synthesis, and biological evaluation of glycine-based molecular tongs as inhibitors of Aβ40 aggregation in vitro | 1-gen-2008 | Cellamare, Saverio; Stefanachi, Angela; Stolfa, D. A.; Basile, T; Catto, Marco; Campagna, Francesco; Sotelo, E; Acquafredda, Pasquale; Carotti, Angelo | |
Homo- and hetero-bivalent edrophonium-like ammonium salts as highly potent, dual binding site AChE inhibitors | 1-gen-2008 | Leonetti, Francesco; Catto, Marco; Nicolotti, Orazio; Pisani, Leonardo; Cappa, A; Stefanachi, Angela; Carotti, Angelo |
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