Sfoglia per Autore
Mixed 5-HT1A/D-2 activity of a new model of arylpiperazines: 1-aryl-4-[3-(1,2-dihydronaphthalen-4-yl)-n-propyl]piperazines. 1. Synthesis and structure-activity relationships
1994-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Tortorella, V; Fiorentini, F; Olgiati, V; Vanotti, E; Govoni, S.
Conformationally restricted thiazole derivatives as novel class of 5-HT3 receptor ligands
1995-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Tortorella, V; Lograno, Md; Daniele, E; Govoni, S.
High affinity and selectivity on 5-HT1A receptor of 1-aryl-4-[(1-tetralin)alkyl]piperazines. 2
1995-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.; Fiorentini, F.; Olgiati, V.; Ghiglieri, A.; Govoni, S.
New sigma and 5-HT1A receptor ligands: omega-(tetralin-1-yl)-n-alkylamine derivatives
1996-01-01 Berardi, Francesco; Colabufo, Nicola Antonio; Giudice, G.; Perrone, Roberto; Tortorella, V.; Govoni, S.; Lucchi, L.
Structure-activity relationship studies on 5-HT1A receptor affinity of 1-phenyl-4-[(alpha- or beta- tetralinyl)-alkyl]piperazines. 4
1996-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V; Fornaretto, Mg; Caccia, C; Mcarthur, Ra
4-[omega-Tetralin-1-yl]-1-benzylpiperazines and related compounds as 5-HT1A/D-2 ligands
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lograno, M.; Tortorella, V.
5-HT3 and 5-HT4 receptor affinities of naphtho[1,2-d]thiazole derivatives with various basic side chains
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-(2-Methoxyphenyl)-4-alkylpiperazines: effect of the N-4 substituent on the affinity and selectivity for dopamine D4 receptor
1997-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
N-[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: a potent and selective dopamine D4 ligand
1998-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella,
1-Aryl-4-[N-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)alkyl]piperazines and their analogues: influence of the stereochemistry of the tetrahydronaphthalen-1-yl nucleus on 5-HT1A receptor affinity and selectivity versus alpha1 and D2 receptors. 5
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
2-(Aryloxy)ethylamine derivatives: ring opened congeners of long chain 1-arylpiperazines with high 5-HT1A receptor affinity and selectivity versus D2 and a1 receptors
1999-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
AFFINITY OF NEW CHIRAL ARYLOXYALKYLPIPERIDINES TOWARDS σ RECEPTOR SUBTYPES.
2000-01-01 Berardi, F.; Colabufo, N. A.; Fracchiolla, G.; Loiodice, Fulvio; Perrone, R.; Tortorella, V.
A structure-affinity relationship study on derivatives of N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a high-affinity and selective D4 receptor ligand
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
1-Substituted-4- 3-(1,2,3,4-tetrahydro-5- or 7-methoxynaphthalen-1-yl)propyl piperazines: influence of the N-1 piperazine substituent on 5-HT1A receptor affinity and selectivity versus D2 and alfa-1 receptors.Part 6
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Tortorella, V.
Affinity of new chiral aryloxyalkylpiperidines towards sigma receptors
2000-01-01 Fracchiolla, Giuseppe; Berardi, Francesco; Colabufo, Nicola Antonio; Loiodice, F.; Perrone, R.; Tortorella, V.
N-aryl- or N-alkylpiperazine derivatives: the role of N-substituent on sigma-1, sigma-2, 5-HT1A and D2 receptor affinity
2000-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Abate, CARMEN rosa; Tortorella, V.
trans-4,4methoxyphenyl cycloehyl piperazines: A new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogues of aryl piperazines
2001-01-01 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, E; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R.
A multireceptorial binding reinvestigation on an extended class of sigma ligands: N-[omega-(indan-1-yl and tetralin-1-yl)alkyl] derivatives of 3,3-dimethylpiperidine reveal high affinities towards sigma1 and EBP sites
2001-01-01 Berardi, Francesco; Ferorelli, Savina; Colabufo, Nicola Antonio; Leopoldo, Marcello; Perrone, Roberto; Tortorella, V.
trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogs of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines
2001-01-01 Perrone, R; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Lacivita, Enza; Tortorella, V; Leonardi, A; Poggesi, E; Testa, R.
Determination of dopamine D4 receptor density in rat striatum using PB12 as a probe
2001-01-01 Colabufo, Nicola Antonio; Berardi, Francesco; Calo', R.; Leopoldo, Marcello; Perrone, Roberto; Tortorella, V.
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