Sfoglia per Autore  ABATE, CARMEN

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Mostrati risultati da 1 a 20 di 88
Titolo Data di pubblicazione Autore(i) File
N-aryl- or N-alkylpiperazine derivatives: the role of N-substituent on sigma-1, sigma-2, 5-HT1A and D2 receptor affinity 1-gen-2000 Perrone, Roberto; Berardi, Francesco; Colabufo, Nicola Antonio; Leopoldo, Marcello; Abate, CARMEN rosa; Tortorella, V.
Exploring the binding at sigma-1 receptor subtype: newly prepared heterocyclic omega-(1-alkyl)-derivatives of 3,3-dimethylpiperidine 1-gen-2003 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Pedone, M. P.; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, R; Tortorella, V.
4-(Tetralin-1-yl)- and 4-(Naphthalen-1-yl)alkyl Derivatives of 1-Cycloheylpiperazine as sigma receptor Ligands with Agonist sigma 2 Activity 1-gen-2004 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, N. C.; Contino, Marialessandra; Perrone, Roberto; Tortorella, V.
Antiproliferative and cytotoxic effects of some sigma-2 agonists and sigma-1 antagonists in tumour cell lines 1-gen-2004 Colabufo, Nicola Antonio; Berardi, Francesco; Contino, Marialessandra; Niso, Mauro; Abate, CARMEN rosa; Perrone, Roberto; Tortorella, V.
Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma1 receptor 1-gen-2005 Berardi, Francesco; Ferorelli, Savina; Abate, CARMEN rosa; M. P., Pedone; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, Roberto
Interaction of chiral MS-245 analogs at h-5-HT6 receptors 1-gen-2005 Abate, Carmen; Kolanos, R; Dukat, M; Setola, V; Roth, Bl; Glennon, Ra
Sintesi di [3H]-1-cicloesil-4-[3-(5-metossi-1,2,3,4-tetraidronaftalen-1-il)-n-propil]piperazina ([3H]-PB28) il primo potente e selettivo strumento farmacologico nella valutazione biologica di recettori sigma-2 1-gen-2006 Abate, CARMEN rosa; Colabufo, Nicola Antonio; Berardi, Francesco; Perrone, R.
Is the sigma-2 receptor a histone binding protein? 1-gen-2006 Colabufo, Nicola Antonio; Berardi, Francesco; Abate, CARMEN rosa; Niso, Mauro; Perrone, Roberto; Contino, Marialessandra
Design and evaluation of naphthol- and carbazole- containing fluorescent sigma ligands as potential probes for receptor binding studies 1-gen-2007 Ferorelli, Savina; Abate, CARMEN rosa; Colabufo, An; Niso, Mauro; Inglese, C; Berardi, Francesco; Perrone, Roberto
New potential Sigma Ligands for P.E.T.: Isosteric changes on PB28 alkyl chain 1-gen-2007 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; Colabufo, Nicola Antonio; Contino, Marialessandra; Perrone, R.
Interaction of the Sigma2 Receptor Ligand PB28 with Human Nucleosome 1-gen-2008 Abate, CARMEN rosa; Elenewski, J. E.; Glennon, R. A.
Tritium radiolabeling of [3H]-1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl)-n-propyl]piperazine ([3H]-PB28), as a potent sigma-2 receptor ligand 1-gen-2008 Abate, CARMEN rosa; Berardi, Francesco; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, R.
Novel 4-(-4-Aryl)cyclohexyl-1-(2-pyridyl)piperazines as delta8-delta7 sterol isomerase ( Emopamil Binding Protein) selective ligands with antiprolifative activity 1-gen-2008 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; DE ROBERTIS, A; Leopoldo, Marcello; Colabufo, An; Niso, Mauro; Perrone, Roberto
Tritium radiolabeling of PB28, a potent sigma-2 receptor ligand: pharmacokinetic and pharmacodynamic characterization 1-gen-2008 Colabufo, Nicola Antonio; Abate, CARMEN rosa; Contino, Marialessandra; Inglese, C; Ferorelli, Savina; Berardi, Francesco; Perrone, Roberto
PB183, a sigma receptor ligand, as a potential PET probe for the imaging of prostate adenocarcinoma 1-gen-2008 Colabufo, Nicola Antonio; Abate, CARMEN rosa; Contino, Marialessandra; Inglese, C.; Niso, Mauro; Berardi, Francesco; Perrone, Roberto
A Structure-Affinity and Comparative Molecular Field Analysis of Sigma-2 (σ2) Receptor Ligands 1-gen-2009 Abate, CARMEN rosa; PHILIP DANIEL, Mosier; Berardi, Francesco; RICHARD A., Glennon
1-Cyclohexylpiperazine and 3,3-Dimethylpiperidine Derivatives as Sigma-1 (σ1) and Sigma-2 (σ2) Receptor Ligands: A Review 1-gen-2009 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; Colabufo, Nicola Antonio; Perrone, Roberto
TRITIUM RADIOLABELING OF [3H]-1-CYCLOHEXYL-4-[3-(5-METHOXY-1,2, 3,4,-TETRAHYDRONAPHTHALEN-1-YL)-N-PROPYL]PIPERAZINE ([3H]-PB28), AS A POTENT SIGMA-2 RECEPTOR LIGAND 1-gen-2009 Abate, CARMEN rosa; Berardi, Francesco; Colabufo, Nicola Antonio; Ferorelli, Savina; Perrone, Roberto
Exploring the importance of piperazine N-atoms for sigma-2 receptor affinity and activity in a series of analogs of 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) 1-gen-2009 Berardi, Francesco; Abate, CARMEN rosa; Ferorelli, Savina; Uricchio, V; Colabufo, Nicola Antonio; Niso, Mauro; Perrone, Roberto
Interaction of the sigma-2 receptor ligand PB28 with the human nucleosome: computational and experimental probes of interaction with the H2A/H2B dimer 1-gen-2010 Abate, Carmen; Elenewski, J.; Niso, Mauro; Berardi, Francesco; Colabufo, Nicola Antonio; Azzariti, A.; Perrone, Roberto; Glennon, R. A.
Mostrati risultati da 1 a 20 di 88
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